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Found 6 Enz. Inhib. hit(s) with all data for entry = 7290
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Facultes Universitaires Notre Dame De La Paix

US Patent
LigandPNGBDBM50333423(7-(Pyridin-3-ylmethoxy)-1-methyl-beta-carboline | ...)
Affinity DataIC50:  1.00E+4nMpH: 7.5Assay Description:A radiometric protein kinase assay (33PanQinase Activity Assay) was used for measuring the kinase activity of DYRK1A protein kinase. All kinase assay...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Facultes Universitaires Notre Dame De La Paix

US Patent
LigandPNGBDBM50395379(CHEMBL2164712 | US9168247, CV12)
Affinity DataIC50: >1.00E+4nMpH: 7.5Assay Description:A radiometric protein kinase assay (33PanQinase Activity Assay) was used for measuring the kinase activity of DYRK1A protein kinase. All kinase assay...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Facultes Universitaires Notre Dame De La Paix

US Patent
LigandPNGBDBM50333416(7-(2-Methoxyethoxy)-1-methyl-beta-carboline | CHEM...)
Affinity DataIC50:  1.55E+4nMpH: 7.5Assay Description:A radiometric protein kinase assay (33PanQinase Activity Assay) was used for measuring the kinase activity of DYRK1A protein kinase. All kinase assay...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Facultes Universitaires Notre Dame De La Paix

US Patent
LigandPNGBDBM50395380(CHEMBL2164709 | US9168247, JR84)
Affinity DataIC50:  1.63E+4nMpH: 7.5Assay Description:A radiometric protein kinase assay (33PanQinase Activity Assay) was used for measuring the kinase activity of DYRK1A protein kinase. All kinase assay...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Facultes Universitaires Notre Dame De La Paix

US Patent
LigandPNGBDBM50395381(CHEMBL2164716 | US9168247, JR95)
Affinity DataIC50:  2.12E+4nMpH: 7.5Assay Description:A radiometric protein kinase assay (33PanQinase Activity Assay) was used for measuring the kinase activity of DYRK1A protein kinase. All kinase assay...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Facultes Universitaires Notre Dame De La Paix

US Patent
LigandPNGBDBM50395378(CHEMBL2164696 | US9168247, CV24)
Affinity DataIC50:  4.30E+4nMpH: 7.5Assay Description:A radiometric protein kinase assay (33PanQinase Activity Assay) was used for measuring the kinase activity of DYRK1A protein kinase. All kinase assay...More data for this Ligand-Target Pair
In DepthDetails US Patent