Compile Data Set for Download or QSAR
Report error Found 25 Enz. Inhib. hit(s) with all data for entry = 7470
LigandChemical structure of BindingDB Monomer ID 196826BDBM196826(US9212186, 23)
Affinity DataKi:  0.300nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196827BDBM196827(US9212186, 24)
Affinity DataKi:  0.600nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50448126BDBM50448126(CHEMBL3122105 | US9212186, 22)
Affinity DataKi:  0.900nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196820BDBM196820(US9212186, 13 | US9212186, 14)
Affinity DataKi:  1.20nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196822BDBM196822(US9212186, 18 | US9212186, 21 | US9212186, 20 | US...)
Affinity DataKi:  1.80nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50448125BDBM50448125(CHEMBL3122106 | US9212186, 17)
Affinity DataKi:  2.30nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196818BDBM196818(US9212186, 11 | US9212186, 12)
Affinity DataKi:  2.60nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50448123BDBM50448123(CHEMBL3122108 | US9212186, 16)
Affinity DataKi:  3nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196816BDBM196816(US9212186, 9)
Affinity DataKi:  4.90nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196822BDBM196822(US9212186, 18 | US9212186, 21 | US9212186, 20 | US...)
Affinity DataKi:  5.70nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196810BDBM196810(US9212186, 3)
Affinity DataKi:  7.5nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196814BDBM196814(US9212186, 7)
Affinity DataKi:  9.5nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196833BDBM196833(US9212186, 30)
Affinity DataKi:  10.9nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196812BDBM196812(US9212186, 5)
Affinity DataKi:  20nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196828BDBM196828(US9212186, 25)
Affinity DataKi:  31.2nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196829BDBM196829(US9212186, 26)
Affinity DataKi:  33.5nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196817BDBM196817(US9212186, 10)
Affinity DataKi:  44.4nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196820BDBM196820(US9212186, 13 | US9212186, 14)
Affinity DataKi:  47.7nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196822BDBM196822(US9212186, 18 | US9212186, 21 | US9212186, 20 | US...)
Affinity DataKi:  61.3nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196815BDBM196815(US9212186, 8)
Affinity DataKi:  144nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196813BDBM196813(US9212186, 6)
Affinity DataKi:  184nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196818BDBM196818(US9212186, 11 | US9212186, 12)
Affinity DataKi:  212nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50448123BDBM50448123(CHEMBL3122108 | US9212186, 16)
Affinity DataKi:  279nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196822BDBM196822(US9212186, 18 | US9212186, 21 | US9212186, 20 | US...)
Affinity DataKi:  390nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 196830BDBM196830(US9212186, 27)
Affinity DataKi:  819nMAssay Description:This assay was used to determine a compound's potency in inhibiting activity of LRRK2 by determining, Kiapp, IC50, or percent inhibition values. In 3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2016
Entry Details
US Patent