Compile Data Set for Download or QSAR
Report error Found 64 Enz. Inhib. hit(s) with all data for entry = 7589
TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204859BDBM204859(US9227979, 7)
Affinity DataKi:  1.20nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204870BDBM204870(US9227979, 19 | EA7/MRS5816)
Affinity DataKi:  2.66nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204863BDBM204863(US9227979, 12 | EA12/MRS5821)
Affinity DataKi:  2.75nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204864BDBM204864(US9227979, 13 | EA15/MRS5824)
Affinity DataKi:  3.46nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204859BDBM204859(US9227979, 7)
Affinity DataKi:  3.5nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204879BDBM204879(US9227979, 37 | MRS5846/5762 5-hex-5-ynamide)
Affinity DataKi:  4.11nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204865BDBM204865(US9227979, 14 | EA6/MRS5815)
Affinity DataKi:  4.47nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204869BDBM204869(US9227979, 18 | EA16/MRS5825)
Affinity DataKi:  6nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204861BDBM204861(US9227979, 9 | MRS5449)
Affinity DataKi:  6.40nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204880BDBM204880(US9227979, 38 | EA18(5-hept-6-ynamide)/MRS5838)
Affinity DataKi:  7.26nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204874BDBM204874(US9227979, 17 | EA13/MRS5822)
Affinity DataKi:  8.06nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204872BDBM204872(US9227979, 21 | EA10/MRS5819)
Affinity DataKi:  10.3nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204878BDBM204878(US9227979, 36 | EA19(5-pent-4-ynamide)/MRS5811)
Affinity DataKi:  11nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204881BDBM204881(US9227979, 39 | EA20(5-oct-7-ynamide)/MRS5840)
Affinity DataKi:  12.8nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204871BDBM204871(US9227979, 20 | EA4/MRS5813)
Affinity DataKi:  19.2nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 60936BDBM60936(US9227979, MRS5763)
Affinity DataKi:  31.8nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204860BDBM204860(US9227979, 8)
Affinity DataKi:  33.5nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204859BDBM204859(US9227979, 7)
Affinity DataKi:  35nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204860BDBM204860(US9227979, 8)
Affinity DataKi:  51nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204868BDBM204868(US9227979, 23 | EA17/MRS5826)
Affinity DataKi:  60.4nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204861BDBM204861(US9227979, 9 | MRS5449)
Affinity DataKi:  73nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204868BDBM204868(US9227979, 23 | EA17/MRS5826)
Affinity DataKi:  73.6nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204866BDBM204866(US9227979, 15 | EA3/MRS5812)
Affinity DataKi:  74.8nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204867BDBM204867(US9227979, 16 | EA9/MRS5818)
Affinity DataKi:  82.4nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204861BDBM204861(US9227979, 9 | MRS5449)
Affinity DataKi:  87nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 60936BDBM60936(US9227979, MRS5763)
Affinity DataKi:  90nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204877BDBM204877(US9227979, 26 | EA11/MRS5820)
Affinity DataKi:  91.5nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204876BDBM204876(US9227979, 25 | EA5/MRS5814)
Affinity DataKi:  95.7nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204875BDBM204875(US9227979, 24 | EA8/MRS5817)
Affinity DataKi:  96.7nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204873BDBM204873(US9227979, 22 | EA14/MRS5823)
Affinity DataKi:  104nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204875BDBM204875(US9227979, 24 | EA8/MRS5817)
Affinity DataKi:  106nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204873BDBM204873(US9227979, 22 | EA14/MRS5823)
Affinity DataKi:  110nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204862BDBM204862(US9227979, 11 | EA2/MRS5811)
Affinity DataKi:  128nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204878BDBM204878(US9227979, 36 | EA19(5-pent-4-ynamide)/MRS5811)
Affinity DataKi:  133nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204876BDBM204876(US9227979, 25 | EA5/MRS5814)
Affinity DataKi:  137nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204863BDBM204863(US9227979, 12 | EA12/MRS5821)
Affinity DataKi:  150nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204880BDBM204880(US9227979, 38 | EA18(5-hept-6-ynamide)/MRS5838)
Affinity DataKi:  151nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A1(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204860BDBM204860(US9227979, 8)
Affinity DataKi:  170nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204869BDBM204869(US9227979, 18 | EA16/MRS5825)
Affinity DataKi:  172nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204874BDBM204874(US9227979, 17 | EA13/MRS5822)
Affinity DataKi:  175nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204879BDBM204879(US9227979, 37 | MRS5846/5762 5-hex-5-ynamide)
Affinity DataKi:  199nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204870BDBM204870(US9227979, 19 | EA7/MRS5816)
Affinity DataKi:  203nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A3(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204877BDBM204877(US9227979, 26 | EA11/MRS5820)
Affinity DataKi:  207nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204871BDBM204871(US9227979, 20 | EA4/MRS5813)
Affinity DataKi:  267nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204864BDBM204864(US9227979, 13 | EA15/MRS5824)
Affinity DataKi:  304nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204867BDBM204867(US9227979, 16 | EA9/MRS5818)
Affinity DataKi:  327nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204872BDBM204872(US9227979, 21 | EA10/MRS5819)
Affinity DataKi:  328nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204865BDBM204865(US9227979, 14 | EA6/MRS5815)
Affinity DataKi:  376nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204866BDBM204866(US9227979, 15 | EA3/MRS5812)
Affinity DataKi:  456nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

TargetAdenosine receptor A2a(Human)
The United States of America, As Represented By The Secretary, Department of Health and Human Services

US Patent
LigandChemical structure of BindingDB Monomer ID 204855BDBM204855(US9227979, 3)
Affinity DataKi:  460nMAssay Description:Radioligand binding assays at hA1, hA2A, and hA3ARs were performed according to the procedures described in Gao, Z. G., et al., Biochem Pharmacol. 20...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

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