Compile Data Set for Download or QSAR
Report error Found 41 Enz. Inhib. hit(s) with all data for entry = 7590
LigandChemical structure of BindingDB Monomer ID 204888BDBM204888(US9260454, 21)
Affinity DataIC50: 14nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204894BDBM204894(US9260454, 28)
Affinity DataIC50: 45nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204910BDBM204910(US9260454, 69)
Affinity DataIC50: 54nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204897BDBM204897(US9260454, 38)
Affinity DataIC50: 61nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204895BDBM204895(US9260454, 29)
Affinity DataIC50: 62nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204911BDBM204911(US9260454, 70)
Affinity DataIC50: 62nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204909BDBM204909(US9260454, 68)
Affinity DataIC50: 65nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204922BDBM204922(US9260454, 89)
Affinity DataIC50: 72nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204887BDBM204887(US9260454, 20)
Affinity DataIC50: 110nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204914BDBM204914(US9260454, 78)
Affinity DataIC50: 120nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204900BDBM204900(US9260454, 44)
Affinity DataIC50: 120nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204913BDBM204913(US9260454, 74)
Affinity DataIC50: 130nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204902BDBM204902(US9260454, 46)
Affinity DataIC50: 140nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204915BDBM204915(US9260454, 80)
Affinity DataIC50: 150nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204908BDBM204908(US9260454, 63 | US9260454, 85)
Affinity DataIC50: 200nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204899BDBM204899(US9260454, 42)
Affinity DataIC50: 240nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204921BDBM204921(US9260454, 88)
Affinity DataIC50: 250nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204884BDBM204884(US9260454, 5)
Affinity DataIC50: 270nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204898BDBM204898(US9260454, 40)
Affinity DataIC50: 340nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204892BDBM204892(US9260454, 26)
Affinity DataIC50: 340nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204891BDBM204891(US9260454, 24)
Affinity DataIC50: 370nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204893BDBM204893(US9260454, 27)
Affinity DataIC50: 420nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204896BDBM204896(US9260454, 36)
Affinity DataIC50: 430nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204917BDBM204917(US9260454, 83)
Affinity DataIC50: 750nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204890BDBM204890(US9260454, 23)
Affinity DataIC50: 800nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204906BDBM204906(US9260454, 59)
Affinity DataIC50: 1.00E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204882BDBM204882(US9260454, 6)
Affinity DataIC50: 1.10E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204912BDBM204912(US9260454, 72)
Affinity DataIC50: 1.20E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204889BDBM204889(US9260454, 22)
Affinity DataIC50: 1.40E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204919BDBM204919(US9260454, 84)
Affinity DataIC50: 1.70E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204904BDBM204904(US9260454, 53)
Affinity DataIC50: 1.70E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204905BDBM204905(US9260454, 55)
Affinity DataIC50: 2.00E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204918BDBM204918(US9260454, 86)
Affinity DataIC50: 2.10E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204903BDBM204903(US9260454, 50)
Affinity DataIC50: 2.30E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204908BDBM204908(US9260454, 63 | US9260454, 85)
Affinity DataIC50: 2.60E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204916BDBM204916(US9260454, 81)
Affinity DataIC50: 2.90E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204907BDBM204907(US9260454, 62)
Affinity DataIC50: 3.10E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204901BDBM204901(US9260454, 45)
Affinity DataIC50: 4.30E+3nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204885BDBM204885(US9260454, 10)
Affinity DataIC50: 1.20E+4nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204883BDBM204883(US9260454, 8)
Affinity DataIC50: 1.80E+4nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 204886BDBM204886(US9260454, 16)
Affinity DataIC50: 2.60E+4nMpH: 7.5 T: 2°CAssay Description:2 ul of a solution of different concentrations of the test compound in dimethyl sulfoxide was added to 28 ul of buffer (50 mM TRIS, 100 mM NaCl, 10 m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2016
Entry Details
US Patent