Compile Data Set for Download or QSAR
Report error Found 297 Enz. Inhib. hit(s) with all data for entry = 7975
TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227334BDBM227334(US9328106, 285)
Affinity DataKi:  0.00100nM ΔG°:  -68.5kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227253BDBM227253(US9328106, 204)
Affinity DataKi:  0.00100nM ΔG°:  -68.5kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227278BDBM227278(US9328106, 229)
Affinity DataKi:  0.00100nM ΔG°:  -68.5kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227362BDBM227362(US9328106, 313)
Affinity DataKi:  0.00200nM ΔG°:  -66.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227169BDBM227169(US9328106, 117)
Affinity DataKi:  0.00200nM ΔG°:  -66.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227443BDBM227443(US9328106, 396)
Affinity DataKi:  0.00200nM ΔG°:  -66.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227267BDBM227267(US9328106, 218)
Affinity DataKi:  0.00224nM ΔG°:  -66.5kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227173BDBM227173(US9328106, 121)
Affinity DataKi:  0.00300nM ΔG°:  -65.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227266BDBM227266(US9328106, 217)
Affinity DataKi:  0.00300nM ΔG°:  -65.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227381BDBM227381(US9328106, 332)
Affinity DataKi:  0.00300nM ΔG°:  -65.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227361BDBM227361(US9328106, 312)
Affinity DataKi:  0.00300nM ΔG°:  -65.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 50053685BDBM50053685(US9328106, 341 | CHEMBL3318855)
Affinity DataKi:  0.00300nM ΔG°:  -65.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227440BDBM227440(US9328106, 393)
Affinity DataKi:  0.00300nM ΔG°:  -65.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227227BDBM227227(US9328106, 177)
Affinity DataKi:  0.00342nM ΔG°:  -65.4kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227445BDBM227445(US9328106, 398)
Affinity DataKi:  0.00400nM ΔG°:  -65.1kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227230BDBM227230(US9328106, 181)
Affinity DataKi:  0.00400nM ΔG°:  -65.1kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227309BDBM227309(US9328106, 260)
Affinity DataKi:  0.00400nM ΔG°:  -65.1kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227366BDBM227366(US9328106, 317)
Affinity DataKi:  0.00509nM ΔG°:  -64.5kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227171BDBM227171(US9328106, 129 | US9328106, 119)
Affinity DataKi:  0.00600nM ΔG°:  -64.1kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 50053679BDBM50053679(US9328106, 115 | CHEMBL3318853)
Affinity DataKi:  0.00600nM ΔG°:  -64.1kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227245BDBM227245(US9328106, 196)
Affinity DataKi:  0.00600nM ΔG°:  -64.1kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227322BDBM227322(US9328106, 273)
Affinity DataKi:  0.00700nM ΔG°:  -63.7kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227407BDBM227407(US9328106, 359)
Affinity DataKi:  0.00700nM ΔG°:  -63.7kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227304BDBM227304(US9328106, 255)
Affinity DataKi:  0.00700nM ΔG°:  -63.7kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227387BDBM227387(US9328106, 338)
Affinity DataKi:  0.00700nM ΔG°:  -63.7kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227330BDBM227330(US9328106, 281)
Affinity DataKi:  0.00700nM ΔG°:  -63.7kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227235BDBM227235(US9328106, 186)
Affinity DataKi:  0.00700nM ΔG°:  -63.7kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227264BDBM227264(US9328106, 215)
Affinity DataKi:  0.00762nM ΔG°:  -63.5kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227354BDBM227354(US9328106, 305)
Affinity DataKi:  0.00800nM ΔG°:  -63.3kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227160BDBM227160(US9328106, 107)
Affinity DataKi:  0.00800nM ΔG°:  -63.3kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227205BDBM227205(US9328106, 154)
Affinity DataKi:  0.00800nM ΔG°:  -63.3kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227421BDBM227421(US9328106, 373)
Affinity DataKi:  0.00900nM ΔG°:  -63.0kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227406BDBM227406(US9328106, 358)
Affinity DataKi:  0.00900nM ΔG°:  -63.0kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227170BDBM227170(US9328106, 118)
Affinity DataKi:  0.00900nM ΔG°:  -63.0kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227389BDBM227389(US9328106, 340)
Affinity DataKi:  0.0100nM ΔG°:  -62.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 50053683BDBM50053683(US9328106, 135 | CHEMBL3318854)
Affinity DataKi:  0.0100nM ΔG°:  -62.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227311BDBM227311(US9328106, 262)
Affinity DataKi:  0.0100nM ΔG°:  -62.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227308BDBM227308(US9328106, 259)
Affinity DataKi:  0.0100nM ΔG°:  -62.8kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227447BDBM227447(US9328106, 400)
Affinity DataKi:  0.0110nM ΔG°:  -62.5kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227249BDBM227249(US9328106, 200)
Affinity DataKi:  0.0110nM ΔG°:  -62.5kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227265BDBM227265(US9328106, 216)
Affinity DataKi:  0.0110nM ΔG°:  -62.5kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227257BDBM227257(US9328106, 208)
Affinity DataKi:  0.0120nM ΔG°:  -62.3kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227212BDBM227212(US9328106, 161)
Affinity DataKi:  0.0130nM ΔG°:  -62.1kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227352BDBM227352(US9328106, 303)
Affinity DataKi:  0.0130nM ΔG°:  -62.1kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227219BDBM227219(US9328106, 168)
Affinity DataKi:  0.0130nM ΔG°:  -62.1kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227339BDBM227339(US9328106, 290)
Affinity DataKi:  0.0131nM ΔG°:  -62.1kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227370BDBM227370(US9328106, 321)
Affinity DataKi:  0.0137nM ΔG°:  -62.0kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227388BDBM227388(US9328106, 339)
Affinity DataKi:  0.0140nM ΔG°:  -62.0kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227353BDBM227353(US9328106, 304)
Affinity DataKi:  0.0140nM ΔG°:  -62.0kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetSerine/threonine-protein kinase pim-1(Human)
Genentech

US Patent
LigandChemical structure of BindingDB Monomer ID 227239BDBM227239(US9328106, 190)
Affinity DataKi:  0.0140nM ΔG°:  -62.0kJ/molepH: 7.2 T: 2°CAssay Description:LC3K assay: PIM-1, -2, and -3 enzymes were generated as fusion proteins expressed in bacteria and purified by IMAC column chromatography (Sun, X., Ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

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