Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 7977
TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Nerviano Medical Sciences

US Patent
LigandPNGBDBM227457(US9333205, 61)
Affinity DataIC50: 240nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of putative kinase inhibitors and the potency of selected compounds were determined using a trans-phosphorylation assay. Spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetDual specificity protein kinase TTK(Human)
Nerviano Medical Sciences

US Patent
LigandPNGBDBM227457(US9333205, 61)
Affinity DataIC50: 360nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of putative kinase inhibitors and the potency of selected compounds were determined using a trans-phosphorylation assay. Spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Nerviano Medical Sciences

US Patent
LigandPNGBDBM227455(US9333205, 30)
Affinity DataIC50: 400nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of putative kinase inhibitors and the potency of selected compounds were determined using a trans-phosphorylation assay. Spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetEukaryotic translation initiation factor 2-alpha kinase 3(Human)
Nerviano Medical Sciences

US Patent
LigandPNGBDBM227456(US9333205, 55)
Affinity DataIC50: 510nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of putative kinase inhibitors and the potency of selected compounds were determined using a trans-phosphorylation assay. Spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetDual specificity protein kinase TTK(Human)
Nerviano Medical Sciences

US Patent
LigandPNGBDBM227455(US9333205, 30)
Affinity DataIC50: 680nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of putative kinase inhibitors and the potency of selected compounds were determined using a trans-phosphorylation assay. Spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent

TargetDual specificity protein kinase TTK(Human)
Nerviano Medical Sciences

US Patent
LigandPNGBDBM227456(US9333205, 55)
Affinity DataIC50: 3.44E+3nMpH: 7.5 T: 2°CAssay Description:The inhibitory activity of putative kinase inhibitors and the potency of selected compounds were determined using a trans-phosphorylation assay. Spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/15/2017
Entry Details
US Patent