Compile Data Set for Download or QSAR
Report error Found 678 Enz. Inhib. hit(s) with all data for entry = 8046
LigandChemical structure of BindingDB Monomer ID 231260BDBM231260(US9346798, 7)
Affinity DataIC50: 4.40nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231304BDBM231304(US9346798, 51)
Affinity DataIC50: 4.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231305BDBM231305(US9346798, 52)
Affinity DataIC50: 4.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231464BDBM231464(US9346798, 211)
Affinity DataIC50: 5.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231298BDBM231298(US9346798, 45)
Affinity DataIC50: 6.20nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231434BDBM231434(US9346798, 181)
Affinity DataIC50: 7.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231255BDBM231255(US9346798, 2)
Affinity DataIC50: 7.83nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231470BDBM231470(US9346798, 217)
Affinity DataIC50: 8nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231347BDBM231347(US9346798, 94)
Affinity DataIC50: 8.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231257BDBM231257(US9346798, 4)
Affinity DataIC50: 9.33nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231282BDBM231282(US9346798, 29)
Affinity DataIC50: 9.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231468BDBM231468(US9346798, 215)
Affinity DataIC50: 9.86nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231279BDBM231279(US9346798, 26)
Affinity DataIC50: 10.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231275BDBM231275(US9346798, 22)
Affinity DataIC50: 10.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231256BDBM231256(US9346798, 3)
Affinity DataIC50: 10.8nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231254BDBM231254(US9346798, 1)
Affinity DataIC50: 11.3nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231439BDBM231439(US9346798, 186)
Affinity DataIC50: 11.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231307BDBM231307(US9346798, 54)
Affinity DataIC50: 11.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231476BDBM231476(US9346798, 223)
Affinity DataIC50: 12nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231278BDBM231278(US9346798, 25)
Affinity DataIC50: 12.3nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231462BDBM231462(US9346798, 209)
Affinity DataIC50: 12.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231463BDBM231463(US9346798, 210)
Affinity DataIC50: 12.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231291BDBM231291(US9346798, 38)
Affinity DataIC50: 13nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231404BDBM231404(US9346798, 151)
Affinity DataIC50: 13.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231297BDBM231297(US9346798, 44)
Affinity DataIC50: 14nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231300BDBM231300(US9346798, 47)
Affinity DataIC50: 14.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231312BDBM231312(US9346798, 59)
Affinity DataIC50: 15nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231302BDBM231302(US9346798, 49)
Affinity DataIC50: 15nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231274BDBM231274(US9346798, 21)
Affinity DataIC50: 15.8nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231284BDBM231284(US9346798, 31)
Affinity DataIC50: 16nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231403BDBM231403(US9346798, 150)
Affinity DataIC50: 17nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231461BDBM231461(US9346798, 208)
Affinity DataIC50: 18.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231465BDBM231465(US9346798, 212)
Affinity DataIC50: 21.3nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231306BDBM231306(US9346798, 53)
Affinity DataIC50: 22.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231260BDBM231260(US9346798, 7)
Affinity DataIC50: 23.7nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231318BDBM231318(US9346798, 65)
Affinity DataIC50: 24nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231318BDBM231318(US9346798, 65)
Affinity DataIC50: 24.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231460BDBM231460(US9346798, 207)
Affinity DataIC50: 25nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231340BDBM231340(US9346798, 87)
Affinity DataIC50: 26nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231316BDBM231316(US9346798, 63)
Affinity DataIC50: 27nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231360BDBM231360(US9346798, 107)
Affinity DataIC50: 28.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231342BDBM231342(US9346798, 89)
Affinity DataIC50: 28.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231301BDBM231301(US9346798, 48)
Affinity DataIC50: 28.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231276BDBM231276(US9346798, 23)
Affinity DataIC50: 29.8nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231459BDBM231459(US9346798, 206)
Affinity DataIC50: 31.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231289BDBM231289(US9346798, 36)
Affinity DataIC50: 31.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231364BDBM231364(US9346798, 111)
Affinity DataIC50: 33.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231469BDBM231469(US9346798, 216)
Affinity DataIC50: 34nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231305BDBM231305(US9346798, 52)
Affinity DataIC50: 35.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 231478BDBM231478(US9346798, 226)
Affinity DataIC50: 36.5nMAssay Description:HEK 293 cells stably transfected with either Nav 1.7 or with Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro auto...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2017
Entry Details
US Patent

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