Compile Data Set for Download or QSAR
Report error Found 19 Enz. Inhib. hit(s) with all data for entry = 8154
TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235136(US9359339, 25)
Affinity DataIC50: 0.100nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235137(US9359339, 27)
Affinity DataIC50: 0.200nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235135(US9359339, 23)
Affinity DataIC50: 0.200nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235138(US9359339, 29)
Affinity DataIC50: 0.400nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235134(US9359339, 21)
Affinity DataIC50: 0.700nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235139(US9359339, 32)
Affinity DataIC50: 1nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235130(US9359339, 13)
Affinity DataIC50: 1.10nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235131(US9359339, 14)
Affinity DataIC50: 1.30nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235132(US9359339, 15)
Affinity DataIC50: 1.70nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235142(US9359339, 45)
Affinity DataIC50: 1.80nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235129(US9359339, 8)
Affinity DataIC50: 2.20nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235126(US9359339, 3)
Affinity DataIC50: 2.30nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235127(US9359339, 4)
Affinity DataIC50: 2.5nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235141(US9359339, 43)
Affinity DataIC50: 3.40nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235125(US9359339, 2)
Affinity DataIC50: 4.70nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235124(US9359339, 1)
Affinity DataIC50: 6.20nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235133(US9359339, 19)
Affinity DataIC50: 7.80nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235140(US9359339, 40)
Affinity DataIC50: 11.8nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent

TargetGlucagon receptor(Human)
Merck Sharp & Dohme

US Patent
LigandPNGBDBM235128(US9359339, 6)
Affinity DataIC50: 28nMpH: 7.5 T: 2°CAssay Description:A stable CHO (Chinese hamster ovary) cell line expressing cloned human glucagon receptor was maintained as described (Chicchi, et. al. J Biol Chem 27...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details
US Patent