Compile Data Set for Download or QSAR
Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 8183
TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235902BDBM235902(US9365502, MQ-87)
Affinity DataIC50: 14nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235905BDBM235905(US9365502, MQ-85)
Affinity DataIC50: 29nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235901BDBM235901(US9365502, MQ-86)
Affinity DataIC50: 43nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235900BDBM235900(US9365502, MQ-37)
Affinity DataIC50: 46nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235898BDBM235898(US9365502, MQ-38)
Affinity DataIC50: 52nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235894BDBM235894(US9365502, MQ-31)
Affinity DataIC50: 61nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235897BDBM235897(US9365502, MQ-33)
Affinity DataIC50: 62nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235907BDBM235907(US9365502, MQ-39)
Affinity DataIC50: 65nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235896BDBM235896(US9365502, MQ-32)
Affinity DataIC50: 147nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235904BDBM235904(US9365502, MQ-48)
Affinity DataIC50: 282nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235899BDBM235899(US9365502, MQ-83)
Affinity DataIC50: 748nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235910BDBM235910(US9365502, MQ-50)
Affinity DataIC50: 1.06E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235903BDBM235903(US9365502, MQ-47)
Affinity DataIC50: 1.33E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235906BDBM235906(US9365502, MQ-49)
Affinity DataIC50: 1.58E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235895BDBM235895(US9365502, MQ-36)
Affinity DataIC50: 1.73E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235911BDBM235911(US9365502, MQ-54)
Affinity DataIC50: 1.99E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235908BDBM235908(US9365502, MQ-53)
Affinity DataIC50: 3.63E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent

TargetGamma-aminobutyric acid receptor subunit alpha-4(Rat)
Washington University

US Patent
LigandChemical structure of BindingDB Monomer ID 235909BDBM235909(US9365502, MQ-51)
Affinity DataIC50: 5.86E+3nMAssay Description:The IC50 values for non-competitive displacers of [35S]-TBPS from the picrotoxin binding site on GABAA receptors.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/3/2017
Entry Details
US Patent