Compile Data Set for Download or QSAR
Report error Found 191 Enz. Inhib. hit(s) with all data for entry = 8253
TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103791BDBM103791(US8816088, I-61 | US8551978, I-61 | US9682957, I-6...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103793BDBM103793(US8816088, I-63 | US8551978, I-63 | US9682957, I-6...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 238342BDBM238342(US9394275, I-57)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103789BDBM103789(US8816088, I-59 | US8551978, I-59 | US9682957, I-5...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103776BDBM103776(US8816088, I-46 | US8551978, I-46 | US9682957, I-4...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103779BDBM103779(US8816088, I-49 | US8551978, I-49 | US9682957, I-4...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103807BDBM103807(US8816088, I-77 | US8551978, I-77 | US9682957, I-7...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103809BDBM103809(US8816088, I-79 | US8551978, I-79 | US9682957, I-7...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103799BDBM103799(US8816088, I-69 | US8551978, I-69 | US9682957, I-6...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103801BDBM103801(US8816088, I-71 | US8551978, I-71 | US9682957, I-7...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103795BDBM103795(US8816088, I-65 | US8551978, I-65 | US9682957, I-6...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 238343BDBM238343(US9394275, I-67)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103818BDBM103818(US8816088, I-89 | US8551978, I-89 | US9682957, I-8...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103816BDBM103816(US8816088, I-86 | US8551978, I-86 | US9682957, I-8...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103811BDBM103811(US8816088, I-81 | US8551978, I-81 | US9682957, I-8...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 6384BDBM6384(US8551978, I-14 | US8816088, I-15 | US8816088, 14 ...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103749BDBM103749(US8816088, I-16 | US8551978, I-16 | US9682957, I-1...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103745BDBM103745(US8816088, I-10 | US8551978, I-10 | US9682957, I-1...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103747BDBM103747(US8816088, I-12 | US8551978, I-12 | US9682957, I-1...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103742BDBM103742(US8816088, I-6 | US8551978, I-6 | US9682957, I-6 |...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 38242BDBM38242(US8551978, I-8 | US8551978, I-7 | US9682957, I-8 |...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103738BDBM103738(US8816088, I-2 | US8551978, I-2 | US9682957, I-2 |...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103740BDBM103740(US8816088, I-4 | US8551978, 266 | US9682957, I-4 |...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103763BDBM103763(US8816088, I-32 | US8551978, I-32 | US9682957, I-3...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103754BDBM103754(US8816088, I-22 | US8551978, I-22 | US9682957, I-2...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103756BDBM103756(US8816088, I-24 | US8551978, I-24 | US9682957, I-2...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 6387BDBM6387(US8816088, 18 | US9682957, I-18 | US9394275, I-18 ...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103752BDBM103752(US8816088, I-20 | US8551978, I-20 | US9682957, I-2...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103776BDBM103776(US8816088, I-46 | US8551978, I-46 | US9682957, I-4...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103774BDBM103774(US8816088, I-44 | US8551978, I-44 | US9682957, I-4...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103770BDBM103770(US8816088, I-40 | US8551978, I-40 | US9682957, I-4...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 6440BDBM6440(US9394275, I-35 | US9682957, I-35 | BDBM41533 | US...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103792BDBM103792(US8816088, I-62 | US8551978, I-62 | US9682957, I-6...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103790BDBM103790(US8816088, I-60 | US8551978, I-60 | US9682957, I-6...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103798BDBM103798(US8816088, I-68 | US8551978, I-68 | US9682957, I-6...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103823BDBM103823(US8816088, I-94 | US8551978, I-94 | US9682957, I-9...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103825BDBM103825(US8816088, I-96 | US8551978, I-96 | US9682957, I-9...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103819BDBM103819(US8816088, I-90 | US8551978, I-90 | US9682957, I-9...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103817BDBM103817(US8816088, I-88 | US8551978, I-88 | US9682957, I-8...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103812BDBM103812(US8816088, I-82 | US8551978, I-82 | US9682957, I-8...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103814BDBM103814(US8816088, I-84 | US8551978, I-84 | US9682957, I-8...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 238344BDBM238344(US9682957, I-13 | US9394275, I-13 | US9572802, Com...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103748BDBM103748(US8551978, I-15 | US9682957, I-15 | US9394275, I-1...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103744BDBM103744(US8816088, I-9 | US8551978, I-9 | US9682957, I-9 |...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103746BDBM103746(US8816088, I-11 | US8551978, I-11 | US9682957, I-1...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103741BDBM103741(US8816088, I-5 | US8551978, I-5 | US9682957, I-5 |...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 6449BDBM6449(US8551978, I-87 | US8816088, 87 | US9682957, I-87 ...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 6354BDBM6354(US8551978, I-1 | US8816088, 1 | US9682957, I-1 | U...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103739BDBM103739(US8816088, I-3 | US8551978, I-3 | US9682957, I-3 |...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Theravance Respiratory

US Patent
LigandChemical structure of BindingDB Monomer ID 103760BDBM103760(US8816088, I-29 | US8551978, I-29 | US9682957, I-2...)
Affinity DataKi:  0.100nM ΔG°:  -59.4kJ/moleT: 2°CAssay Description:Displacement assays for determination of Ki values of test compounds were performed with [3H]-NMS at 1 nM and eleven different test compound concentr...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/18/2017
Entry Details
US Patent

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