Compile Data Set for Download or QSAR
Report error Found 136 Enz. Inhib. hit(s) with all data for entry = 8295
LigandChemical structure of BindingDB Monomer ID 239752BDBM239752(US9394311, 35 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.150nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239785BDBM239785(US9394311, 68 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.220nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239837BDBM239837(US9394311, 119 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.230nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239812BDBM239812(US9394311, 95 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.230nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239755BDBM239755(US9394311, 38 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.280nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239826BDBM239826(US9394311, 109 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.290nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239840BDBM239840(US9394311, 122 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.350nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239838BDBM239838(US9394311, 120 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.360nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239822BDBM239822(US9394311, 105 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.440nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239793BDBM239793(US9394311, 76 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.440nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239799BDBM239799(US9394311, 82 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.480nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239786BDBM239786(US9394311, 128 | US9394311, 69 | Roche-Dataset for...)
Affinity DataIC50: 0.5nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239815BDBM239815(US9394311, 98 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.510nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239823BDBM239823(US9394311, 106 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.550nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239753BDBM239753(US9394311, 36 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.580nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239769BDBM239769(US9394311, 52 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.630nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239851BDBM239851(US9394311, 132 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.720nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239786BDBM239786(US9394311, 128 | US9394311, 69 | Roche-Dataset for...)
Affinity DataIC50: 0.720nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239778BDBM239778(US9394311, 61 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 0.720nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239825BDBM239825(US9394311, 108)
Affinity DataIC50: 0.800nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239808BDBM239808(US9394311, 91)
Affinity DataIC50: 0.880nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239849BDBM239849(US9394311, 130 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 0.890nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239744BDBM239744(US9394311, 27)
Affinity DataIC50: 0.980nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239788BDBM239788(US9394311, 71 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 1.01nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239789BDBM239789(US9394311, 72 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 1.22nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239834BDBM239834(US9394311, 117a)
Affinity DataIC50: 1.32nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239839BDBM239839(US9394311, 121 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 1.37nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239727BDBM239727(US9394311, 10)
Affinity DataIC50: 1.40nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239801BDBM239801(US9394311, 84 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 1.45nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239850BDBM239850(US9394311, 131 | Roche-Dataset for PDE10A, Compoun...)
Affinity DataIC50: 1.58nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239726BDBM239726(US9394311, 8)
Affinity DataIC50: 1.87nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239841BDBM239841(US9394311, 123a)
Affinity DataIC50: 2.03nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239844BDBM239844(US9394311, 125)
Affinity DataIC50: 2.07nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239745BDBM239745(US9394311, 28)
Affinity DataIC50: 2.13nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239791BDBM239791(US9394311, 74 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 2.16nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239796BDBM239796(US9394311, 79 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 2.22nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239735BDBM239735(US9394311, 18)
Affinity DataIC50: 2.68nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239846BDBM239846(US9394311, 127)
Affinity DataIC50: 2.71nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239779BDBM239779(US9394311, 62 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 3.23nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239827BDBM239827(US9394311, 110)
Affinity DataIC50: 3.25nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239803BDBM239803(US9394311, 86 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 3.44nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239787BDBM239787(US9394311, 70 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 3.47nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239792BDBM239792(US9394311, 75 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 3.78nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239754BDBM239754(US9394311, 37)
Affinity DataIC50: 4.21nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239802BDBM239802(US9394311, 85 | Roche-Dataset for PDE10A, Compound...)
Affinity DataIC50: 4.22nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239764BDBM239764(US9394311, 47)
Affinity DataIC50: 4.48nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239748BDBM239748(US9394311, 31)
Affinity DataIC50: 4.49nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239767BDBM239767(US9394311, 50)
Affinity DataIC50: 4.90nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239763BDBM239763(US9394311, 46)
Affinity DataIC50: 4.98nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 239737BDBM239737(US9394311, 20)
Affinity DataIC50: 5nMT: 2°CAssay Description:The human PDE10A full length assay was performed in 96-well micro titer plates. The reaction mixture of 50 μl contained 20 mM HEPES pH=7.5/10 mM M...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2017
Entry Details
US Patent

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