Compile Data Set for Download or QSAR
Report error Found 108 Enz. Inhib. hit(s) with all data for entry = 8357
TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242783BDBM242783(US9422331, 1)
Affinity DataIC50: 3nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242789BDBM242789(US9422331, 7)
Affinity DataIC50: 5nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242790BDBM242790(US9422331, 8)
Affinity DataIC50: 5nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242784BDBM242784(US9422331, 2)
Affinity DataIC50: 6nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242787BDBM242787(US9422331, 5)
Affinity DataIC50: 6nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 50441827BDBM50441827(CHEMBL2436217 | US9422331, 11)
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242791BDBM242791(US9422331, 9)
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242805BDBM242805(US9422331, 26)
Affinity DataIC50: 9nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242821BDBM242821(US9422331, 49)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242810BDBM242810(US9422331, 34)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 50441821BDBM50441821(CHEMBL2436223 | US9422331, 27)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 50441826BDBM50441826(CHEMBL2436216 | US9422331, 10)
Affinity DataIC50: 10nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242796BDBM242796(US9422331, 17)
Affinity DataIC50: 11nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242785BDBM242785(US9422331, 3)
Affinity DataIC50: 12nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242822BDBM242822(US9422331, 50)
Affinity DataIC50: 12nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242803BDBM242803(US9422331, 24)
Affinity DataIC50: 12nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242786BDBM242786(US9422331, 4)
Affinity DataIC50: 13nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242820BDBM242820(US9422331, 48)
Affinity DataIC50: 13nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242811BDBM242811(US9422331, 35)
Affinity DataIC50: 15nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242802BDBM242802(US9422331, 23)
Affinity DataIC50: 16nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242804BDBM242804(US9422331, 25)
Affinity DataIC50: 17nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242788BDBM242788(US9422331, 6)
Affinity DataIC50: 17nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242800BDBM242800(US9422331, 21)
Affinity DataIC50: 18nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 50441809BDBM50441809(CHEMBL2436218 | US9422331, 13)
Affinity DataIC50: 19nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 50441807BDBM50441807(CHEMBL2436225 | US9422331, 31)
Affinity DataIC50: 22nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242823BDBM242823(US9422331, 52)
Affinity DataIC50: 23nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242807BDBM242807(US9422331, 29)
Affinity DataIC50: 23nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242825BDBM242825(US9422331, 54)
Affinity DataIC50: 23nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 50441824BDBM50441824(CHEMBL2436224 | US9422331, 51)
Affinity DataIC50: 27nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242809BDBM242809(US9422331, 33)
Affinity DataIC50: 28nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242817BDBM242817(US9422331, 42)
Affinity DataIC50: 29nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242797BDBM242797(US9422331, 18)
Affinity DataIC50: 30nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 50441813BDBM50441813(CHEMBL2436222 | US9422331, 44)
Affinity DataIC50: 32nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242824BDBM242824(US9422331, 53)
Affinity DataIC50: 33nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242808BDBM242808(US9422331, 30)
Affinity DataIC50: 34nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242794BDBM242794(US9422331, 15)
Affinity DataIC50: 43nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242819BDBM242819(US9422331, 47)
Affinity DataIC50: 43nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242798BDBM242798(US9422331, 19)
Affinity DataIC50: 44nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 50441806BDBM50441806(CHEMBL2436226 | US9422331, 32)
Affinity DataIC50: 46nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242793BDBM242793(US9422331, 14)
Affinity DataIC50: 54nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242799BDBM242799(US9422331, 20)
Affinity DataIC50: 55nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242801BDBM242801(US9422331, 22)
Affinity DataIC50: 56nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 50441808BDBM50441808(CHEMBL2436219 | US9422331, 45)
Affinity DataIC50: 58nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242806BDBM242806(US9422331, 28)
Affinity DataIC50: 75nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 50441814BDBM50441814(CHEMBL2436221 | US9422331, 46)
Affinity DataIC50: 83nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242812BDBM242812(US9422331, 36)
Affinity DataIC50: 120nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242818BDBM242818(US9422331, 43)
Affinity DataIC50: 125nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242795BDBM242795(US9422331, 16)
Affinity DataIC50: 179nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 50441815BDBM50441815(CHEMBL2436220 | US9422331, 39)
Affinity DataIC50: 182nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

TargetE3 ubiquitin-protein ligase XIAP [124-214,C202A,C213G](Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 242813BDBM242813(US9422331, 37)
Affinity DataIC50: 189nMpH: 7.5 T: 2°CAssay Description:The peptide AVPIAQKSEK-(ε-biotin)-OH 1:2 TFA ("Peptide A") was identified as a substrate for the TR-FRET assay by screening the 6× Hist...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2017
Entry Details
US Patent

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