Compile Data Set for Download or QSAR
Report error Found 40 Enz. Inhib. hit(s) with all data for entry = 8422
TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247344BDBM247344(US9447091, 131)
Affinity DataIC50: 1.30nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247340BDBM247340(US9447091, 112)
Affinity DataIC50: 1.80nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247357BDBM247357(US9447091, 241)
Affinity DataIC50: 2.90nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247334BDBM247334(US9447091, 49)
Affinity DataIC50: 3.40nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247361BDBM247361(US9447091, 220)
Affinity DataIC50: 3.40nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247328BDBM247328(US9447091, 22)
Affinity DataIC50: 3.80nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247354BDBM247354(US9447091, 190)
Affinity DataIC50: 4.30nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247333BDBM247333(US9447091, 47)
Affinity DataIC50: 7nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247348BDBM247348(US9447091, 152)
Affinity DataIC50: 7.30nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247360BDBM247360(US9447091, 281)
Affinity DataIC50: 9nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247363BDBM247363(US9447091, 294)
Affinity DataIC50: 9.30nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247336BDBM247336(US9447091, 70)
Affinity DataIC50: 10nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247356BDBM247356(US9447091, 217)
Affinity DataIC50: 10.4nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247327BDBM247327(US9447091, 5 | US12378241, Compound A)
Affinity DataIC50: 12nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247345BDBM247345(US9447091, 133)
Affinity DataIC50: 14nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247358BDBM247358(US9447091, 244)
Affinity DataIC50: 14nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247353BDBM247353(US9447091, 178)
Affinity DataIC50: 14.9nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247338BDBM247338(US9447091, 82)
Affinity DataIC50: 16nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247331BDBM247331(US9447091, 30)
Affinity DataIC50: 16nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247364BDBM247364(US9447091, 319)
Affinity DataIC50: 18nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247355BDBM247355(US9447091, 204)
Affinity DataIC50: 20nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247330BDBM247330(US9447091, 26)
Affinity DataIC50: 21nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247335BDBM247335(US9447091, 69)
Affinity DataIC50: 22nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247350BDBM247350(US9447091, 158)
Affinity DataIC50: 22nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247337BDBM247337(US9447091, 72)
Affinity DataIC50: 32nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247362BDBM247362(US9447091, 289)
Affinity DataIC50: 32nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247332BDBM247332(US9447091, 38)
Affinity DataIC50: 33nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247329BDBM247329(US9447091, 25)
Affinity DataIC50: 34nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247339BDBM247339(US9447091, 83)
Affinity DataIC50: 37nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247366BDBM247366(US9447091, 259)
Affinity DataIC50: 45nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247347BDBM247347(US9447091, 142)
Affinity DataIC50: 48nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247352BDBM247352(US9447091, 170)
Affinity DataIC50: 59nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247342BDBM247342(US9447091, 123)
Affinity DataIC50: 61nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247349BDBM247349(US9447091, 155)
Affinity DataIC50: 62nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247343BDBM247343(US9447091, 127)
Affinity DataIC50: 62nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247365BDBM247365(US9447091, 322)
Affinity DataIC50: 65.8nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247341BDBM247341(US9447091, 119)
Affinity DataIC50: 83nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247359BDBM247359(US9447091, 280)
Affinity DataIC50: 90nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247351BDBM247351(US9447091, 169)
Affinity DataIC50: 94nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetFibroblast growth factor receptor 1(Human)
Orion

US Patent
LigandChemical structure of BindingDB Monomer ID 247346BDBM247346(US9447091, 134)
Affinity DataIC50: 98nMAssay Description:Compounds were screened in the TR-FRET assay with FGFR1 kinase. 5 ng of FGFR1 [Upstate, USA] kinase was used for assay. The compound was incubated wi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent