Compile Data Set for Download or QSAR
Report error Found 6 Enz. Inhib. hit(s) with all data for entry = 8426
TargetPhospholipase D1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 247410BDBM247410(US9453017, 2)
Affinity DataIC50: 15nMAssay Description:In vitro PLD activity is measured with an exogenous substrate assay as previously described (Brown, H. A. et al. (1993) Cell 75:1137-1144). Briefly, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetPhospholipase D1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 87245BDBM87245(VU0155056-2 | N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[...)
Affinity DataIC50: 80nMAssay Description:In vitro PLD activity is measured with an exogenous substrate assay as previously described (Brown, H. A. et al. (1993) Cell 75:1137-1144). Briefly, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetPhospholipase D2(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 247409BDBM247409(US9453017, 1)
Affinity DataIC50: 100nMAssay Description:In vitro PLD activity is measured with an exogenous substrate assay as previously described (Brown, H. A. et al. (1993) Cell 75:1137-1144). Briefly, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetPhospholipase D2(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 87245BDBM87245(VU0155056-2 | N-(2-(4-(2-Oxo-2,3-dihydro-1H-benzo[...)
Affinity DataIC50: 240nMAssay Description:In vitro PLD activity is measured with an exogenous substrate assay as previously described (Brown, H. A. et al. (1993) Cell 75:1137-1144). Briefly, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetPhospholipase D2(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 247410BDBM247410(US9453017, 2)
Affinity DataIC50: 1.10E+3nMAssay Description:In vitro PLD activity is measured with an exogenous substrate assay as previously described (Brown, H. A. et al. (1993) Cell 75:1137-1144). Briefly, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent

TargetPhospholipase D1(Human)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 247409BDBM247409(US9453017, 1)
Affinity DataIC50: 7.40E+3nMAssay Description:In vitro PLD activity is measured with an exogenous substrate assay as previously described (Brown, H. A. et al. (1993) Cell 75:1137-1144). Briefly, ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/5/2017
Entry Details
US Patent