Compile Data Set for Download or QSAR
Report error Found 162 Enz. Inhib. hit(s) with all data for entry = 8494
TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135770BDBM135770(US8846601, 155 | US9458201, 155 | US10179804, Exam...)
Affinity DataEC50:  0.189nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135775BDBM135775(US8846601, 160 | US9458201, 160 | US10179804, Exam...)
Affinity DataEC50:  0.245nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135765BDBM135765(US8846601, 150 | US9458201, 150 | US10179804, Exam...)
Affinity DataEC50:  0.300nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135736BDBM135736(US8846601, 121 | US9458201, 121 | US10179804, Exam...)
Affinity DataKi:  0.400nM ΔG°:  -55.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135752BDBM135752(US8846601, 137 | US9458201, 137 | US10179804, Exam...)
Affinity DataKi:  0.400nM ΔG°:  -55.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135776BDBM135776(US8846601, 161 | US9458201, 161 | US10179804, Exam...)
Affinity DataEC50:  0.413nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135767BDBM135767(US8846601, 152 | US9458201, 152 | US10179804, Exam...)
Affinity DataEC50:  0.5nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135690BDBM135690(US8846601, 75 | US9458201, 75 | US10179804, Exampl...)
Affinity DataKi:  0.600nM ΔG°:  -54.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135769BDBM135769(US8846601, 202 | US8846601, 154 | US9458201, 154 |...)
Affinity DataEC50:  0.625nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135717BDBM135717(US8846601, 102 | US9458201, 102 | US10179804, Exam...)
Affinity DataKi:  0.700nM ΔG°:  -54.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135630BDBM135630(US8846601, 15 | US9458201, 15 | US10179804, Exampl...)
Affinity DataKi:  0.700nM ΔG°:  -54.4kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135753BDBM135753(US8846601, 138 | US9458201, 138 | US10179804, Exam...)
Affinity DataKi:  0.800nM ΔG°:  -54.0kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135774BDBM135774(US8846601, 159 | US9458201, 159 | US10179804, Exam...)
Affinity DataEC50:  0.825nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135777BDBM135777(US8846601, 162 | US9458201, 162 | US10179804, Exam...)
Affinity DataEC50:  0.850nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135754BDBM135754(US8846601, 139 | US9458201, 139 | US10179804, Exam...)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135629BDBM135629(US8846601, 14 | US9458201, 14 | US10179804, Exampl...)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135679BDBM135679(US8846601, 64 | US9458201, 64 | US10179804, Exampl...)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 253650BDBM253650(US9458201, 96 | US10632171, Peptide No. 96)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135725BDBM135725(US8846601, 110 | US9458201, 110 | US10179804, Exam...)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135741BDBM135741(US8846601, 126 | US9458201, 126 | US10179804, Exam...)
Affinity DataKi:  1nM ΔG°:  -53.4kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135687BDBM135687(US8846601, 72 | US9458201, 72 | US10179804, Exampl...)
Affinity DataKi:  2nM ΔG°:  -51.6kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135755BDBM135755(US8846601, 140 | US9458201, 140 | US10179804, Exam...)
Affinity DataKi:  2nM ΔG°:  -51.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135771BDBM135771(US8846601, 156 | US9458201, 156 | US10179804, Exam...)
Affinity DataEC50:  2nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135742BDBM135742(US8846601, 127 | US9458201, 127 | US10179804, Exam...)
Affinity DataKi:  2nM ΔG°:  -51.6kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135743BDBM135743(US8846601, 128 | US9458201, 128 | US10179804, Exam...)
Affinity DataKi:  2nM ΔG°:  -51.6kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135686BDBM135686(US8846601, 71 | US9458201, 71 | US10179804, Exampl...)
Affinity DataEC50:  2nMpH: 7.5 T: 2°CAssay Description:Accumulation of intracellular cAMP was examined as a measure of the ability of the peptides of the present invention to elicit a functional response ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135737BDBM135737(US8846601, 122 | US9458201, 122 | US10632171, Pept...)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135734BDBM135734(US8846601, 119 | US9458201, 119 | US10179804, Exam...)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135716BDBM135716(US8846601, 101 | US9458201, 101 | US10179804, Exam...)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 253653BDBM253653(US9458201, 132 | US10179804, Example 132 | US10632...)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 253656BDBM253656(US9458201, 146)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135633BDBM135633(US8846601, 18 | US9458201, 55 | US10179804, Exampl...)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135669BDBM135669(US8846601, 54 | US9458201, 54 | US10179804, Exampl...)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135634BDBM135634(US8846601, 19 | US9458201, 19 | US10179804, Exampl...)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135689BDBM135689(US8846601, 74 | US9458201, 74 | US10179804, Exampl...)
Affinity DataKi:  3nM ΔG°:  -50.6kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135766BDBM135766(US8846601, 151 | US9458201, 151 | US10179804, Exam...)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135697BDBM135697(US8846601, 82 | US9458201, 82 | US10179804, Exampl...)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135694BDBM135694(US8846601, 79 | US9458201, 79 | US10179804, Exampl...)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 253651BDBM253651(US9458201, 98 | US10179804, Example 98 | US1063217...)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135643BDBM135643(US8846601, 28 | US9458201, 28 | US10179804, Exampl...)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135744BDBM135744(US8846601, 129 | US9458201, 136 | US10179804, Exam...)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/moleT: 2°CAssay Description:A competitive inhibition binding assay was performed employing Eu-NDP-α-MSH (PerkinElmer Life Sciences catalog No. AD0225) with determination b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135760BDBM135760(US8846601, 145 | US9458201, 145 | US10179804, Exam...)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135774BDBM135774(US8846601, 159 | US9458201, 159 | US10179804, Exam...)
Affinity DataKi:  4nM ΔG°:  -49.9kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135770BDBM135770(US8846601, 155 | US9458201, 155 | US10179804, Exam...)
Affinity DataKi:  5nM ΔG°:  -49.3kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135765BDBM135765(US8846601, 150 | US9458201, 150 | US10179804, Exam...)
Affinity DataKi:  5nM ΔG°:  -49.3kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135695BDBM135695(US8846601, 80 | US9458201, 80 | US10179804, Exampl...)
Affinity DataKi:  5nM ΔG°:  -49.3kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135777BDBM135777(US8846601, 162 | US9458201, 162 | US10179804, Exam...)
Affinity DataKi:  5nM ΔG°:  -49.3kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135616BDBM135616(US8846601, 51 | US8846601, 115 | US8846601, 1 | US...)
Affinity DataKi:  5nM ΔG°:  -49.3kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135720BDBM135720(US8846601, 105 | US9458201, 105 | US10179804, Exam...)
Affinity DataKi:  6nM ΔG°:  -48.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

TargetMelanocortin receptor 4(Human)
Palatin Technologies

US Patent
LigandChemical structure of BindingDB Monomer ID 135767BDBM135767(US8846601, 152 | US9458201, 152 | US10179804, Exam...)
Affinity DataKi:  6nM ΔG°:  -48.8kJ/molepH: 7.5 T: 2°CAssay Description:A competitive inhibition binding assay is performed using membrane homogenates prepared from HEK-293 cells that express recombinant hMC4-R, hMC3-R, o...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2017
Entry Details
US Patent

Displayed 1 to 50 (of 162 total ) | Next | Last >>
Jump to: