Compile Data Set for Download or QSAR
Report error Found 36 Enz. Inhib. hit(s) with all data for entry = 8515
LigandChemical structure of BindingDB Monomer ID 254948BDBM254948(US9505765, 38)
Affinity DataIC50: 3.10nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254963BDBM254963(US9505765, 187)
Affinity DataIC50: 4.30nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254964BDBM254964(US9505765, 188)
Affinity DataIC50: 4.40nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254968BDBM254968(US9505765, 192)
Affinity DataIC50: 5.20nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254962BDBM254962(US9505765, 186)
Affinity DataIC50: 7nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254971BDBM254971(US9505765, 195)
Affinity DataIC50: 13nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254975BDBM254975(US9505765, 199)
Affinity DataIC50: 16nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254965BDBM254965(US9505765, 189)
Affinity DataIC50: 19nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254967BDBM254967(US9505765, 191)
Affinity DataIC50: 33nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254949BDBM254949(US9505765, 39)
Affinity DataIC50: 41nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254970BDBM254970(US9505765, 194)
Affinity DataIC50: 51nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254969BDBM254969(US9505765, 193)
Affinity DataIC50: 75nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254961BDBM254961(US9505765, 184)
Affinity DataIC50: 97nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254947BDBM254947(US9505765, 37)
Affinity DataIC50: 100nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254966BDBM254966(US9505765, 190)
Affinity DataIC50: 170nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254946BDBM254946(US9505765, 36)
Affinity DataIC50: 170nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254958BDBM254958(US9505765, 181)
Affinity DataIC50: 180nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254953BDBM254953(US9505765, 176)
Affinity DataIC50: 200nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254952BDBM254952(US9505765, 175)
Affinity DataIC50: 200nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254945BDBM254945(US9505765, 35)
Affinity DataIC50: 210nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254944BDBM254944(US9505765, 23)
Affinity DataIC50: 280nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254950BDBM254950(US9505765, 93)
Affinity DataIC50: 330nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254955BDBM254955(US9505765, 178)
Affinity DataIC50: 340nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254956BDBM254956(US9505765, 179)
Affinity DataIC50: 340nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254977BDBM254977(US9505765, 201)
Affinity DataIC50: 350nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254972BDBM254972(US9505765, 196)
Affinity DataIC50: 360nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254957BDBM254957(US9505765, 180)
Affinity DataIC50: 380nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254974BDBM254974(US9505765, 198)
Affinity DataIC50: 420nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254954BDBM254954(US9505765, 177)
Affinity DataIC50: 430nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254942BDBM254942(US9505765, 1)
Affinity DataIC50: 560nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254951BDBM254951(US9505765, 96)
Affinity DataIC50: 730nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254973BDBM254973(US9505765, 197)
Affinity DataIC50: 750nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254976BDBM254976(US9505765, 200)
Affinity DataIC50: 860nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254959BDBM254959(US9505765, 182)
Affinity DataIC50: 1.60E+3nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254943BDBM254943(US9505765, 21)
Affinity DataIC50: 1.70E+3nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 254960BDBM254960(US9505765, 183)
Affinity DataIC50: 2.50E+3nMAssay Description:TAK1-TAB1 Binding Inhibitory Potency: The ability of candidate compounds to interact with TAK1-TAB1 is quantitated by a competitive binding assay usi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2017
Entry Details
US Patent