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Report error Found 18 Enz. Inhib. hit(s) with all data for entry = 8547
TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257517BDBM257517(US9505773, 10)
Affinity DataKi:  4.20nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 92863BDBM92863(mTOR Inhibitor, Rapamycin | US9505773, Rapamycin)
Affinity DataKi:  5.40nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257515BDBM257515(US9505773, 8)
Affinity DataKi:  5.90nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257521BDBM257521(US9505773, 14)
Affinity DataKi:  6.5nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257524BDBM257524(US9505773, 19)
Affinity DataKi:  7.70nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257513BDBM257513(US9505773, 5)
Affinity DataKi:  7.90nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257519BDBM257519(US9505773, 12)
Affinity DataKi:  9.5nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257529BDBM257529(US9505773, Meridamycin)
Affinity DataKi:  10nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257528BDBM257528(US9505773, FK506)
Affinity DataKi:  10nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257527BDBM257527(US9505773, 22)
Affinity DataKi:  12nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257520BDBM257520(US9505773, 13)
Affinity DataKi:  13nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257525BDBM257525(US9505773, 20)
Affinity DataKi:  18nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257523BDBM257523(US9505773, 18)
Affinity DataKi:  45nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257526BDBM257526(US9505773, 21)
Affinity DataKi:  95nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257516BDBM257516(US9505773, 9)
Affinity DataKi:  180nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257514BDBM257514(US9505773, 6)
Affinity DataKi:  370nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257518BDBM257518(US9505773, 11)
Affinity DataKi:  430nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent

TargetPeptidyl-prolyl cis-trans isomerase FKBP1A(Human)
Isomerase Therapeutics

US Patent
LigandChemical structure of BindingDB Monomer ID 257522BDBM257522(US9505773, 16)
Affinity DataKi:  460nMAssay Description:The assay was conducted at 10° C. in 50 mM Tris buffer at pH8.0, 50 μM DTT, 100 mM NaCl, 0.005% NP40 with 6 nM FKBP12 and 60 μM substrate (...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/6/2017
Entry Details
US Patent