Compile Data Set for Download or QSAR
Report error Found 98 Enz. Inhib. hit(s) with all data for entry = 676
TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286349BDBM286349(US9518060, Example K7 | US11220518, Ex. No. K7 | U...)
Affinity DataKi:  0.165nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286350BDBM286350(US9518060, Example K8 | US11220518, Ex. No. K8 | U...)
Affinity DataKi:  0.181nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286348BDBM286348(US9518060, Example K6 | US11220518, Ex. No. K6 | U...)
Affinity DataKi:  0.376nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286347BDBM286347(US9518060, Example K5 | US11220518, Ex. No. K5 | U...)
Affinity DataKi:  0.683nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286345BDBM286345(US9518060, Example K3 | US11220518, Ex. No. K3 | U...)
Affinity DataKi:  0.912nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286246BDBM286246(5-{[(8S)-6,8-dimethyl-6,9-diazaspiro[4.5]dec-9-yl]...)
Affinity DataKi:  1.01nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286343BDBM286343(N-(2-ethoxy-5-fluoropyrimidin-4-yl)-6,6-dimethyl-5...)
Affinity DataKi:  1.12nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286320BDBM286320(US9518060, Example J6)
Affinity DataKi:  1.17nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286270BDBM286270(US9518060, Example E2 | US11220518, Ex. No. E2 | U...)
Affinity DataKi:  1.64nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286377BDBM286377(US9518060, Example L4 | US11220518, Ex. No. L4 | U...)
Affinity DataKi:  1.71nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286310BDBM286310(N-(5-fluoro-2-propylpyrimidin-4-yl)-6,6-dimethyl-5...)
Affinity DataKi:  1.73nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286260BDBM286260(US9518060, Example B3 | US11220518, Ex. No. B3 | U...)
Affinity DataKi:  2.03nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286327BDBM286327(N-[5-fluoro-2-(methoxymethyl)pyrimidin-4-yl]-6,6-d...)
Affinity DataKi:  2.10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286344BDBM286344(US9518060, Example K2 | US11220518, Ex. No. K2 | U...)
Affinity DataKi:  2.11nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286264BDBM286264(US9518060, Example B6 | US11220518, Ex. No. B6 | U...)
Affinity DataKi:  2.43nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286316BDBM286316(US9518060, Example J3)
Affinity DataKi:  2.63nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286227BDBM286227(N4-(6,6-dimethyl-5-{[(2S)-2,4,5,5-tetramethylpiper...)
Affinity DataKi:  2.69nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286346BDBM286346(US9518060, Example K4 | US11220518, Ex. No. K4 | U...)
Affinity DataKi:  3.33nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286244BDBM286244(US9518060, Example A8 | US11220518, Ex. No. A8 | U...)
Affinity DataKi:  3.39nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286311BDBM286311(US9518060, Example I2 | US11220518, Ex. No. I2 | U...)
Affinity DataKi:  3.67nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286242BDBM286242(US9518060, Example A7 | US11220518, Ex. No. A7 | U...)
Affinity DataKi:  3.81nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286239BDBM286239(US9518060, Example A5 | US11220518, Ex. No. A5 | U...)
Affinity DataKi:  3.95nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286380BDBM286380(N-(4-ethoxypyrimidin-2-yl)-6,6-dimethyl-5-{[(2S,5R...)
Affinity DataKi:  4.24nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286257BDBM286257(N2-ethyl-5-fluoro-N4-(5-{[(2S,5R)-4-(3-methoxyprop...)
Affinity DataKi:  5.09nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286267BDBM286267(N-(2-ethyl-5-fluoropyrimidin-4-yl)-6,6-dimethyl-5-...)
Affinity DataKi:  5.43nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286318BDBM286318(US9518060, Example J5 | US11220518, Ex. No. J5 | U...)
Affinity DataKi:  6.43nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286279BDBM286279(US9518060, Example H3 | US11220518, Ex. No. H3 | U...)
Affinity DataKi:  7.21nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286317BDBM286317(US9518060, Example J4 | US11220518, Ex. No. J4 | U...)
Affinity DataKi:  8.64nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286231BDBM286231(US9518060, Example A2 | US11780853, Example A2)
Affinity DataKi:  8.75nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286245BDBM286245(US9518060, Example A9 | US11220518, Ex. No. A9 | U...)
Affinity DataKi:  9.73nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286273BDBM286273(2-((5S)-4-{[3-[(2-ethyl-5-fluoropyrimidin-4-yl)ami...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286384BDBM286384(5-{[(2S,5R)-2,5-dimethyl-4-(tetrahydro-2H-pyran-4-...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286385BDBM286385(US9518060, Example N3 | US9518060, Example N2 | US...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286368BDBM286368(US9518060, Example K24 | US9518060, Example K23 | ...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286330BDBM286330(US9518060, Example J10 | US11220518, Ex. No. J10 |...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286331BDBM286331(US9518060, Example J11 | US11220518, Ex. No. J11 |...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286332BDBM286332(US9518060, Example J12 | US11220518, Ex. No. J12 |...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286335BDBM286335(US9518060, Example J13 | US11220518, Ex. No. J13 |...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286340BDBM286340(US9518060, Example J15 | US11220518, Ex. No. J15 |...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286362BDBM286362(US9518060, Example K19 | US11220518, Ex. No. K19 |...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286365BDBM286365(5-{[(2S,5R)-2,5-dimethyl-4-(tetrahydro-2H-pyran-4-...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286368BDBM286368(US9518060, Example K24 | US9518060, Example K23 | ...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286248BDBM286248(N4-(5-{[(2S,5R)-2,5-dimethyl-4-(tetrahydro-2H-pyra...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286251BDBM286251(US9518060, Example A12 | US11220518, Ex. No. A12 |...)
Affinity DataKi: <10nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286269BDBM286269(N-(2-ethyl-5-fluoropyrimidin-4-yl)-6,6-dimethyl-5-...)
Affinity DataKi:  10.5nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286241BDBM286241(US9518060, Example A6 | US11220518, Ex. No. A6 | U...)
Affinity DataKi:  10.8nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286342BDBM286342(US9518060, Example J16 | US11220518, Ex. No. J16 |...)
Affinity DataKi:  11.1nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286357BDBM286357(US9518060, Example K15 | US11220518, Ex. No. K15 |...)
Affinity DataKi:  11.2nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286351BDBM286351(US9518060, Example K9)
Affinity DataKi:  12.8nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

TargetProtein-tyrosine kinase 2-beta(Human)
Pfizer

US Patent
LigandChemical structure of BindingDB Monomer ID 286271BDBM286271(US9518060, Example E3)
Affinity DataKi:  13.1nMpH: 7.4Assay Description:Protein Kinase C beta 2 (PKCβII) catalyzes the production of ADP from ATP that accompanies the phosphoryl transfer to the PKC Pseudosubstrate pe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/14/2019
Entry Details
US Patent

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