Compile Data Set for Download or QSAR
Report error Found 26 Enz. Inhib. hit(s) with all data for entry = 187
TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205040BDBM205040(n-(3-(2-(9h-purin-6-yl)phenylamino)-4-methylphenyl...)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205011BDBM205011(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-2-chloro...)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205010BDBM205010(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-4-chloro...)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205009BDBM205009(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-4-methyl...)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205008BDBM205008(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-4-chloro...)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205007BDBM205007(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-4-fluoro...)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 197677BDBM197677(US9216981, 5 | US9550781, 1)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 197706BDBM197706(US9216981, 35 | US9550781, 15)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205013BDBM205013(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-2,4-difl...)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205012BDBM205012(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-4-chloro...)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 197689BDBM197689(US9216981, 17 | US9550781, 24)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50165873BDBM50165873(US9550781, 19 | CHEMBL3800014)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205021BDBM205021(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-2,4-difl...)
Affinity DataIC50: 100nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205020BDBM205020(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-2,4-difl...)
Affinity DataIC50: 500nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205017BDBM205017(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-2,4-difl...)
Affinity DataIC50: 500nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50165871BDBM50165871(US9550781, 13 | CHEMBL3798635)
Affinity DataIC50: 500nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205014BDBM205014(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-2,4-difl...)
Affinity DataIC50: 500nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205038BDBM205038(n-(3-(3-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)pyridin-2...)
Affinity DataIC50: 500nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205035BDBM205035(n-(3-(3-(1h-pyrazolo[3,4-d]pyrimidin-4-yl)pyridin-...)
Affinity DataIC50: 500nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205024BDBM205024(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-2,4-difl...)
Affinity DataIC50: 500nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205005BDBM205005(n-(2,4-difluoro-3-(3-(8-methyl-9h-purin-6-yl)pyrid...)
Affinity DataIC50: 500nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205023BDBM205023(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-2,4-difl...)
Affinity DataIC50: 500nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205015BDBM205015(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-2,4-difl...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205042BDBM205042(n-(3-(2-(9h-purin-6-yl)phenylamino)-2,4-difluoroph...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 50165865BDBM50165865(US9550781, 23 | CHEMBL3798423)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent

TargetNuclear receptor coactivator 2 [740-753]()
Centaurus Biopharma

US Patent
LigandChemical structure of BindingDB Monomer ID 205025BDBM205025(n-(3-(3-(9h-purin-6-yl)pyridin-2-ylamino)-2,4-difl...)
Affinity DataIC50: 1.00E+3nMAssay Description:In vitro B-RAF Kinase Assay. To determine iIn vitro activities of recombinant B-RAF enzyme, a Homogeneous Time-Resolved Fluorescence (HTRF) assay was...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/7/2018
Entry Details
US Patent