Compile Data Set for Download or QSAR
Report error Found 35 Enz. Inhib. hit(s) with all data for entry = 220
TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151617BDBM151617(US8987335, 18)
Affinity DataIC50: 13nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151611BDBM151611(US8987335, 12 | SP-2509 | US9555024, 12 | US114330...)
Affinity DataIC50: 13nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151608BDBM151608(US8987335, 9 | US9555024, 9)
Affinity DataIC50: 13nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151623BDBM151623(US8987335, 24)
Affinity DataIC50: 28nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151624BDBM151624(US8987335, 25)
Affinity DataIC50: 49nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151610BDBM151610(US8987335, 11 | US9555024, 11)
Affinity DataIC50: 128nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 50445343BDBM50445343(CHEMBL3104348 | US9555024, 4)
Affinity DataIC50: 196nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151605BDBM151605(US8987335, 1 | US9555024, 1)
Affinity DataIC50: 218nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 50445341BDBM50445341(CHEMBL3104346 | US9555024, 2)
Affinity DataIC50: 275nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151606BDBM151606(US8987335, 3 | US9555024, 3)
Affinity DataIC50: 291nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 50445339BDBM50445339(CHEMBL3104349 | US9555024, 5)
Affinity DataIC50: 333nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151622BDBM151622(US8987335, 23)
Affinity DataIC50: 519nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetAmine oxidase [flavin-containing] B(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151605BDBM151605(US8987335, 1 | US9555024, 1)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetAmine oxidase [flavin-containing] A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151625BDBM151625(US8987335, --)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151619BDBM151619(US8987335, 20)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 50445334BDBM50445334(CHEMBL3104247 | US9555024, 7)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 50445335BDBM50445335(CHEMBL3104246 | US9555024, 6)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151620BDBM151620(US8987335, 21)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151618BDBM151618(US8987335, 19 | US9555024, 19)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151615BDBM151615(US8987335, 16 | US9555024, 16)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151621BDBM151621(US8987335, 22)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151614BDBM151614(US8987335, 15 | US9555024, 15)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151613BDBM151613(US8987335, 14 | US9555024, 14)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151612BDBM151612(US8987335, 13 | US9555024, 13)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151616BDBM151616(US8987335, 17)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151607BDBM151607(US8987335, 8 | US9555024, 8)
Affinity DataIC50: 3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetAmine oxidase [flavin-containing] B(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151625BDBM151625(US8987335, --)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151609BDBM151609(US8987335, 10 | US9555024, 10)
Affinity DataIC50: 1.00E+4nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetAmine oxidase [flavin-containing] A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151605BDBM151605(US8987335, 1 | US9555024, 1)
Affinity DataIC50: 8.85E+4nMAssay Description:Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetAmine oxidase [flavin-containing] A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151611BDBM151611(US8987335, 12 | SP-2509 | US9555024, 12 | US114330...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetAmine oxidase [flavin-containing] A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151617BDBM151617(US8987335, 18)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetAmine oxidase [flavin-containing] B(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151611BDBM151611(US8987335, 12 | SP-2509 | US9555024, 12 | US114330...)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetAmine oxidase [flavin-containing] A(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151623BDBM151623(US8987335, 24)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetAmine oxidase [flavin-containing] B(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151617BDBM151617(US8987335, 18)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent

TargetAmine oxidase [flavin-containing] B(Human)
University of Utah

US Patent
LigandChemical structure of BindingDB Monomer ID 151623BDBM151623(US8987335, 24)
Affinity DataIC50: 3.00E+5nMAssay Description:Inhibition of monoamine oxidase activity was carried used using the MAO-GIo Assay Kit according to the manufacturer's suggested protocol. Briefly...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2018
Entry Details
US Patent