Compile Data Set for Download or QSAR
Report error Found 86 Enz. Inhib. hit(s) with all data for entry = 1188
LigandChemical structure of BindingDB Monomer ID 50030266BDBM50030266(CHEMBL3339223 | US9603889, Example 8)
Affinity DataIC50: 30nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312090BDBM312090(US9603889, Example 2)
Affinity DataIC50: 30nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312102BDBM312102(US9603889, Example 13 | (S)-N-Benzyl-2- ((S)-3,3- ...)
Affinity DataIC50: 40nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312103BDBM312103(US9603889, Example 14 | (S)-2-((S)- 3,3-Dimethyl- ...)
Affinity DataIC50: 40nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312113BDBM312113(US9603889, Example 24 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 60nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312121BDBM312121(US9603889, Example 32 | N1-(((S)-2-((S)- 3,3-Dimet...)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312129BDBM312129(US9603889, Example 40)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50030266BDBM50030266(CHEMBL3339223 | US9603889, Example 8)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312130BDBM312130(US9603889, Example 41)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50030268BDBM50030268(CHEMBL3339221 | US9603889, Example 1)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312114BDBM312114(US9603889, Example 25 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312099BDBM312099(US9603889, Example 10)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312091BDBM312091(US9603889, Example 3)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312127BDBM312127(US9603889, Example 38)
Affinity DataIC50: 60nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312105BDBM312105(US9603889, Example 16 | (S)-2-((S)-3,3- Dimethyl- ...)
Affinity DataIC50: 70nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312131BDBM312131(US9603889, Example 42)
Affinity DataIC50: 70nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312100BDBM312100(US9603889, Example 11 | (S)-N-(2,3- Dichlorobenzyl...)
Affinity DataIC50: 70nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312094BDBM312094(US9603889, Example 6)
Affinity DataIC50: 70nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312128BDBM312128(US9603889, Example 39)
Affinity DataIC50: 80nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312104BDBM312104(US9603889, Example 15 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 90nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50030268BDBM50030268(CHEMBL3339221 | US9603889, Example 1)
Affinity DataIC50: 90nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312116BDBM312116(US9603889, Example 27 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 90nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312125BDBM312125(US9603889, Example 36 | N1-(((S)-2-((S)- 3,3-Dimet...)
Affinity DataIC50: 90nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312101BDBM312101(US9603889, Example 12 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 90nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312106BDBM312106(US9603889, Example 17 | N1-(((S)-2-((S)- 3,3-dimet...)
Affinity DataIC50: 100nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312115BDBM312115(US9603889, Example 26 | (3S)-N-(1-(2- Chlorophenyl...)
Affinity DataIC50: 100nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312092BDBM312092(US9603889, Example 4)
Affinity DataIC50: 100nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312130BDBM312130(US9603889, Example 41)
Affinity DataIC50: 110nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312109BDBM312109(US9603889, Example 20 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 110nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312111BDBM312111(US9603889, Example 22 | (S)-2-((S)-3,3- Dimethyl- ...)
Affinity DataIC50: 110nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312112BDBM312112(US9603889, Example 23 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 120nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312122BDBM312122(US9603889, Example 33 | N1-(((S)-2-((S)- 3,3-Dimet...)
Affinity DataIC50: 120nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312107BDBM312107(US9603889, Example 18 | (S)-N-((S)-1-(3- Chlorophe...)
Affinity DataIC50: 120nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312091BDBM312091(US9603889, Example 3)
Affinity DataIC50: 120nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312113BDBM312113(US9603889, Example 24 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 130nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312097BDBM312097(US9603889, Example 9)
Affinity DataIC50: 130nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312132BDBM312132(US9603889, Example 43)
Affinity DataIC50: 150nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312094BDBM312094(US9603889, Example 6)
Affinity DataIC50: 150nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312123BDBM312123(US9603889, Example 34 | N1-(((S)-2-((S)- 3,3-Dimet...)
Affinity DataIC50: 160nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312117BDBM312117(US9603889, Example 28 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 160nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312118BDBM312118(US9603889, Example 29 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 160nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312112BDBM312112(US9603889, Example 23 | (S)-2-((S)-3,3- Dimethyl-2...)
Affinity DataIC50: 170nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312132BDBM312132(US9603889, Example 43)
Affinity DataIC50: 180nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312092BDBM312092(US9603889, Example 4)
Affinity DataIC50: 180nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312095BDBM312095(US9603889, Example 7)
Affinity DataIC50: 190nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312107BDBM312107(US9603889, Example 18 | (S)-N-((S)-1-(3- Chlorophe...)
Affinity DataIC50: 190nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312115BDBM312115(US9603889, Example 26 | (3S)-N-(1-(2- Chlorophenyl...)
Affinity DataIC50: 190nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312093BDBM312093(US9603889, Example 5)
Affinity DataIC50: 220nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312127BDBM312127(US9603889, Example 38)
Affinity DataIC50: 220nMAssay Description:Assays were performed in white, flat-bottom, 384-well ProxiPlates (Perkin Elmer). The final assay volume was 10 μL prepared from additions of Hi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 312124BDBM312124(US9603889, Example 35 | N1-(((S)-2-((S)- 3,3-Dimet...)
Affinity DataIC50: 230nMAssay Description:Assays were performed in black, flat-bottom, 384-well plates. The final assay volume was 50 μL prepared from additions of N-His-Tb-BIR3(241-356,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

Displayed 1 to 50 (of 86 total ) | Next | Last >>
Jump to: