Compile Data Set for Download or QSAR
Report error Found 516 Enz. Inhib. hit(s) with all data for entry = 1209
TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312471BDBM312471(US9604977, Example 217 | 2-[5-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 9nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312344BDBM312344(US9604977, Example 90 | 2-[3-(4-Trifluoromethyl-th...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312490BDBM312490(US9604977, Example 236 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312313BDBM312313(US9604977, Example 61 | 2-[3-(3-Trifluoromethyl-[1...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312340BDBM312340(US9604977, Example 86 | 2-[3-(4-Trifluoromethyl-th...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312389BDBM312389(US9604977, Example 135 | 2-[3-(3-Trifluoromethyl-[...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312453BDBM312453(US9604977, Example 199 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312356BDBM312356(US9604977, Example 102 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312342BDBM312342(US9604977, Example 88 | 2-[3-(3-Cyclopropyl-[1,2,4...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312447BDBM312447(US9604977, Example 193 | 2-[6-Ethyl-3-(4-methyl-th...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312401BDBM312401(US9604977, Example 147 | 2-[6,6-Difluoro-3-(3-trif...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312380BDBM312380(US9604977, Example 126 | 2-[3-(3-Trifluoromethyl-[...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312314BDBM312314(US9604977, Example 62 | 3-[3-(3-Trifluoromethyl-[1...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312347BDBM312347(US9604977, Example 93 | 3-[3-(3-Cyclopropyl-[1,2,4...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312350BDBM312350(US9604977, Example 96 | 2-[3-(4-Cyclopropyl-thiazo...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312382BDBM312382(US9604977, Example 128 | 3-[3-(3-Trifluoromethyl-[...)
Affinity DataIC50: 10nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312493BDBM312493(US9604977, Example 239 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 11nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312465BDBM312465(US9604977, Example 211 | 3-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 12nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312510BDBM312510(US9604977, Example 256 | (R)-1-[[3-[3-(trifluorome...)
Affinity DataIC50: 12nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312472BDBM312472(US9604977, Example 218 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 13nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312420BDBM312420(US9604977, Example 166 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 13nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312421BDBM312421(US9604977, Example 167 | 2-[(S)-3-(3-Cyclopropyl-[...)
Affinity DataIC50: 13nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312460BDBM312460(US9604977, Example 206 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 16nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312500BDBM312500(US9604977, Example 246 | 4-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 17nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312473BDBM312473(US9604977, Example 219 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 18nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312454BDBM312454(US9604977, Example 200 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 18nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312422BDBM312422(US9604977, Example 168 | 2-[(R)-3-(3-Cyclopropyl-[...)
Affinity DataIC50: 18nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312472BDBM312472(US9604977, Example 218 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 19nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312346BDBM312346(US9604977, Example 92 | 2-[3-(3-Cyclopropyl-[1,2,4...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312378BDBM312378(US9604977, Example 124 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312379BDBM312379(US9604977, Example 125 | 3-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312346BDBM312346(US9604977, Example 92 | 2-[3-(3-Cyclopropyl-[1,2,4...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312388BDBM312388(US9604977, Example 134 | 3-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312404BDBM312404(US9604977, Example 150 | 2-[6,6-Difluoro-3-(4-meth...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312338BDBM312338(US9604977, Example 85 | 2-[3-(4-Trifluoromethyl-th...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312485BDBM312485(US9604977, Example 231 | 2-[6,6-Difluoro-3-(4-isop...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312340BDBM312340(US9604977, Example 86 | 2-[3-(4-Trifluoromethyl-th...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312342BDBM312342(US9604977, Example 88 | 2-[3-(3-Cyclopropyl-[1,2,4...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312405BDBM312405(US9604977, Example 151 | 2-[6,6-Difluoro-3-(4-meth...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312343BDBM312343(US9604977, Example 89 | 2-[3-(4-Trifluoromethyl-th...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312391BDBM312391(US9604977, Example 137 | 3-[3-(3-Trifluoromethyl-[...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312319BDBM312319(US9604977, Example 67 | 2-[3-(3-Isopropyl-[1,2,4]o...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312386BDBM312386(US9604977, Example 132 | 2-[3-(3-Cyclopropyl-[1,2,...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312320BDBM312320(US9604977, Example 68 | 3-[3-(3-Isopropyl-[1,2,4]o...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312401BDBM312401(US9604977, Example 147 | 2-[6,6-Difluoro-3-(3-trif...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312338BDBM312338(US9604977, Example 85 | 2-[3-(4-Trifluoromethyl-th...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein, adipocyte(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312331BDBM312331(US9604977, Example 78 | 2-[3-(4-Methyl-oxazol-2-yl...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312330BDBM312330(US9604977, Example 77 | 2-[4,4-Dimethyl-3-(3-methy...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312363BDBM312363(US9604977, Example 109 | (−)-2-[3-(3-Cyclopr...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

TargetFatty acid-binding protein 5(Human)
Hoffmann-La Roche

US Patent
LigandChemical structure of BindingDB Monomer ID 312313BDBM312313(US9604977, Example 61 | 2-[3-(3-Trifluoromethyl-[1...)
Affinity DataIC50: 20nMAssay Description:Compounds were profiled for activity against human FABP4 (huFABP4) and/or human FABP5 (huFABP5) in Terbium (Tb) time resolved-fluorescence energy tra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/23/2019
Entry Details
US Patent

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