Compile Data Set for Download or QSAR
Report error Found 808 Enz. Inhib. hit(s) with all data for entry = 1093
LigandChemical structure of BindingDB Monomer ID 308636BDBM308636(trans-N-[2-chloro-4-(trifluoromethyl)benzyl]-4-(4-...)
Affinity DataKi: <1nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308767BDBM308767(trans-N-[2-chloro-4-(trifluoromethyl)benzyl]-1-[(1...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309277BDBM309277(US9656955, Example 800 | Trans-4-(3-fluoropyridin-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309148BDBM309148(US9656955, Example 670 | (3R,4S)-1-[(1-methyl-1H-i...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309278BDBM309278((3R,4S)-4-(4-fluorophenyl)-1-[(1-methyl-1H-imidazo...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308646BDBM308646(trans-N-(3-chloro-4-fluorophenyl)-4-(4-fluoropheny...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308645BDBM308645(US9656955, Example 159 | trans-4-(4-fluorophenyl)-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308773BDBM308773(US9656955, Example 287 | N-{trans-4-(4-fluoropheny...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309280BDBM309280(US9656955, Example 803 | 5-fluoro-N-{(3R,4S)-1-[(1...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308884BDBM308884(US9656955, Example 398 | (3R,4S)-1-[(1-methyl-1H-i...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309143BDBM309143(US9656955, Example 665 | (3R,4S)-4-(4-fluorophenyl...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308766BDBM308766(US9656955, Example 280 | trans-N-(2,4-dichlorobenz...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309272BDBM309272(US9656955, Example 795 | 5-fluoro-N-{(3R,4S)-4-(4-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308784BDBM308784(US9656955, Example 298 | trans-N-[4-fluoro-3-(trif...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309163BDBM309163(BDBM309164 | US9656955, Example 685 | Trans-1-[(1-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309291BDBM309291(US9656955, Example 816 | Trans-1-[(1-methyl-1H-imi...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308783BDBM308783(US9656955, Example 297 | (3-chlorophenyl){trans-4-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309293BDBM309293(US9656955, Example 818 | Trans-N-[2-chloro-4-(trif...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308910BDBM308910(US9656955, Example 425 | Trans-4-cyclohexyl-1-[(1-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309163BDBM309163(BDBM309164 | US9656955, Example 685 | Trans-1-[(1-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308662BDBM308662(US9656955, Example 176 | trans-4-(4-fluorophenyl)-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309283BDBM309283(US9656955, Example 807 | N-{(3R,4S)-4-(4-fluorophe...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309027BDBM309027(US9656955, Example 548 | (3R,4S)-N-hexyl-1-[(1-met...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309282BDBM309282(US9656955, Example 806 | 5-chloro-N-{(3R,4S)-4-(4-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309285BDBM309285(US9656955, Example 809 | N-{((3R,4S)-1-[(1-methyl-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308902BDBM308902(US9656955, Example 417 | (3R,4S)-N-(3-chloro-4-flu...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309284BDBM309284(US9656955, Example 808 | 5-chloro-N-{(3R,4S)-1-[(1...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308780BDBM308780(US9656955, Example 294 | 4-{[trans-3-{[2-chloro-4-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309159BDBM309159(US9656955, Example 681 | Trans-1-[(1-methyl-1H-imi...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309286BDBM309286(US9656955, Example 810 | 5-fluoro-N-{(3R,4S)-4-(4-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309311BDBM309311(US9656955, Example 836 | trans-4-(4-fluorophenyl)-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308806BDBM308806(US9656955, Example 320 | trans-N-[2-chloro-4-(trif...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309313BDBM309313(US9656955, Example 838 | (3R,4S)-4-(4-fluorophenyl...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309312BDBM309312(US9656955, Example 837 | (3R,4S)-4-(4-fluorophenyl...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308791BDBM308791(US9656955, Example 305 | trans-4-(4-fluorophenyl)-...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309049BDBM309049(US9656955, Example 570 | (3R,4S)-N-[(2,5-dichlorot...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308815BDBM308815(US9656955, Example 329 | (3R,4S)-4-(4-fluorophenyl...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308815BDBM308815(US9656955, Example 329 | (3R,4S)-4-(4-fluorophenyl...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309199BDBM309199(US9656955, Example 722 | N-{(3R,4S)-4-(4-fluorophe...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308808BDBM308808(US9656955, Example 322 | (3R,4S)-N-[2-chloro-4-(tr...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309315BDBM309315(US9656955, Example 840 | (3R,4S)-4-(4-fluorophenyl...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309314BDBM309314(US9656955, Example 839 | (3R,4S)-4-(4-fluorophenyl...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309317BDBM309317(US9656955, Example 842 | (3R,4S)-N-(3-chloro-4-flu...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309316BDBM309316(US9656955, Example 841 | (3R,4S)-N-(3-chlorophenyl...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308813BDBM308813(US9656955, Example 327 | (3R,4S)-4-(4-fluorophenyl...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309210BDBM309210(US9656955, Example 733 | (3R,4S)-N-(2,2-difluorohe...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308706BDBM308706(US9656955, Example 220 | trans-1-[(1-methyl-1H-imi...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 308582BDBM308582(US9656955, Example 67 | trans-1-[(1-methyl-1H-imid...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309202BDBM309202(US9656955, Example 725 | N-{(3R,4S)-4-(4-fluorophe...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 309205BDBM309205(US9656955, Example 728 | 6-(4-fluorophenyl)-N-{(3R...)
Affinity DataKi: <10nMAssay Description:Radioligand binding assays using recombinant CHO cell membranes expressing human GlyT1: Radioligand binding to human GlyT1c transporter-expressing me...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/8/2019
Entry Details
US Patent

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