Compile Data Set for Download or QSAR
Report error Found 431 Enz. Inhib. hit(s) with all data for entry = 1516
LigandChemical structure of BindingDB Monomer ID 329283BDBM329283(US9663508, Example 784 | 4-(5-chloro-6-(3,5-dichlo...)
Affinity DataIC50: 14nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329279BDBM329279(US9663508, Example 782 | 4-(5-chloro-6-(2,4-dichlo...)
Affinity DataIC50: 16.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329192BDBM329192(US9663508, Example 694 | 4-(5-cyano-6-(3,6-dichlor...)
Affinity DataIC50: 17.2nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329097BDBM329097(US9663508, Example 598 | 5-chloro-4-(5-chloro-6-(2...)
Affinity DataIC50: 18.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329191BDBM329191(US9663508, Example 693 | 4-(5-cyano-6-(2,6-dichlor...)
Affinity DataIC50: 22.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329298BDBM329298(US9663508, Example 799 | 4-(5-chloro-6-(2,4-dichlo...)
Affinity DataIC50: 23.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329287BDBM329287(US9663508, Example 788 | 4-(5-chloro-6-(2,4-dichlo...)
Affinity DataIC50: 24.8nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329293BDBM329293(US9663508, Example 794 | 3-bromo-4-(5-chloro-6-(2,...)
Affinity DataIC50: 27.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329187BDBM329187(US9663508, Example 689 | 4-(5-cyano-6-(2,4-dichlor...)
Affinity DataIC50: 28.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329077BDBM329077(US9663508, Example 578 | 4-(5-chloro-6-(2,4-dichlo...)
Affinity DataIC50: 29.6nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329082BDBM329082(US9663508, Example 583 | 4-(5-chloro-6-(2,3-dichlo...)
Affinity DataIC50: 30.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329039BDBM329039(US9663508, Example 422 | 4-(5-chloro-6-(3,5-dichlo...)
Affinity DataIC50: 31.3nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329042BDBM329042(US9663508, Example 425 | 4-(5-chloro-6-(3-chloro-4...)
Affinity DataIC50: 32.2nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329206BDBM329206(US9663508, Example 708 | 4-(6-(1,3-benzothiazol-2-...)
Affinity DataIC50: 32.6nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329054BDBM329054(US9663508, Example 461 | 4-(5-chloro-6-(3,5-dichlo...)
Affinity DataIC50: 33.7nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329015BDBM329015(US9663508, Example 348 | 4-(5-chloro-6-(3,5-dichlo...)
Affinity DataIC50: 34.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329273BDBM329273(US9663508, Example 776 | 3-chloro-4-(5-chloro-6-(2...)
Affinity DataIC50: 34.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329085BDBM329085(US9663508, Example 586 | 4-(5-chloro-6-(3-chloro-2...)
Affinity DataIC50: 34.6nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329146BDBM329146(US9663508, Example 647 | Mixture of 4-(6-((1R)-1-(...)
Affinity DataIC50: 34.9nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329163BDBM329163(US9663508, Example 665 | 4-(5-chloro-6-(2,4-dichlo...)
Affinity DataIC50: 35.7nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329261BDBM329261(US9663508, Example 764 | 4-(5-chloro-6-(2,6-dichlo...)
Affinity DataIC50: 36.7nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329250BDBM329250(US9663508, Example 753 | 4-(5-chloro-6-(4-chloro-2...)
Affinity DataIC50: 36.9nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329235BDBM329235(US9663508, Example 738 | 4-(5-chloro-6-(2,4-dichlo...)
Affinity DataIC50: 37nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329040BDBM329040(US9663508, Example 423 | 4-(5-chloro-6-(2-chloro-5...)
Affinity DataIC50: 38.6nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329290BDBM329290(US9663508, Example 791 | 4-(5-chloro-6-(2,3,6-trif...)
Affinity DataIC50: 39.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329274BDBM329274(US9663508, Example 777 | 3-chloro-4-(5-chloro-6-(3...)
Affinity DataIC50: 40nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329249BDBM329249(US9663508, Example 752 | 4-(5-chloro-6-(2-chloro-5...)
Affinity DataIC50: 42.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329074BDBM329074(US9663508, Example 575 | 4-(5-bromo-6-(2,4-dichlor...)
Affinity DataIC50: 42.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329277BDBM329277(US9663508, Example 780 | 4-(5-chloro-6-(3-chloro-2...)
Affinity DataIC50: 44.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329104BDBM329104(US9663508, Example 605 | 4-(5-chloro-6-(2,5-difluo...)
Affinity DataIC50: 45.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329037BDBM329037(US9663508, Example 413 | 4-(5-chloro-6-(4-chloro-3...)
Affinity DataIC50: 46.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329171BDBM329171(US9663508, Example 673 | 4-(5-chloro-6-((1R)-1-(2,...)
Affinity DataIC50: 46.2nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329202BDBM329202(US9663508, Example 704 | 4-(5-chloro-6-(3-chloro-2...)
Affinity DataIC50: 46.8nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329188BDBM329188(US9663508, Example 690 | 4-(6-(3-chloro-2-methylph...)
Affinity DataIC50: 46.9nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329260BDBM329260(US9663508, Example 763 | 4-(5-chloro-6-(4-chloro-3...)
Affinity DataIC50: 47.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329084BDBM329084(US9663508, Example 585 | 4-(5-chloro-6-(2,4-dichlo...)
Affinity DataIC50: 47.2nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329254BDBM329254(US9663508, Example 757 | 4-(5-chloro-6-((7-fluoro-...)
Affinity DataIC50: 47.7nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329107BDBM329107(US9663508, Example 608 | 4-(5-chloro-6-((2-methyl-...)
Affinity DataIC50: 48.1nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329122BDBM329122(US9663508, Example 623 | 4-(5-chloro-6-(3-fluoro-4...)
Affinity DataIC50: 48.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329066BDBM329066(US9663508, Example 568 | 4-(5-chloro-6-(2,4,6-tric...)
Affinity DataIC50: 48.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329078BDBM329078(US9663508, Example 579 | 4-(5-chloro-6-(3-chloro-2...)
Affinity DataIC50: 48.6nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329093BDBM329093(US9663508, Example 594 | 5-chloro-4-(5-chloro-6-((...)
Affinity DataIC50: 48.8nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329225BDBM329225(US9663508, Example 728 | 4-(5-chloro-6-((4-methylp...)
Affinity DataIC50: 49.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329164BDBM329164(US9663508, Example 666 | 4-(5-chloro-6-(2-chloro-4...)
Affinity DataIC50: 49.7nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329088BDBM329088(US9663508, Example 589 | 5-chloro-4-(5-chloro-6-(2...)
Affinity DataIC50: 49.9nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329229BDBM329229(4-(5-chloro-6-((1R)-1-cyclobutylethoxy)-3-pyridiny...)
Affinity DataIC50: 50nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329292BDBM329292(US9663508, Example 793 | 4-(5-chloro-6-(3,4-dichlo...)
Affinity DataIC50: 50.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329028BDBM329028(US9663508, Example 372 | 4-(5-chloro-6-(3-chloro-5...)
Affinity DataIC50: 50.4nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329165BDBM329165(US9663508, Example 667 | US9663508, Example 668 | ...)
Affinity DataIC50: 50.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 329063BDBM329063(US9663508, Example 829 | 4-(6-(3-chloro-4- methylp...)
Affinity DataIC50: 50.5nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2019
Entry Details
US Patent

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