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Report error Found 114 Enz. Inhib. hit(s) with all data for entry = 126
LigandPNGBDBM164395(US9669029, 98 8-Methoxy-5-methyl-2-{2-[1-(2-morpho...)
Affinity DataIC50:  0.330nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164399(US9669029, 102 5,8-Dimethyl-2-[2-(1-methyl-4-thiop...)
Affinity DataIC50:  0.390nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164544(US9669029, 115 5,8-Dimethyl-2-[2-(1-methyl-4-thiaz...)
Affinity DataIC50:  0.400nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164545(US9669029, 116 5,8-Dimethyl-2-[2-(1-methyl-4-pyrim...)
Affinity DataIC50:  0.440nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164549(US9669029, 117 5,8-Dimethyl-2-[2-(1-methyl-4-pyraz...)
Affinity DataIC50:  0.520nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164283(US9669029, 33 5-Methyl-2-[2-(4-thiophen-2-yl-1H-im...)
Affinity DataIC50:  0.540nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164560(US9669029, 118 5,8-Dimethyl-2-[2-(1-methyl-4-pyrid...)
Affinity DataIC50:  0.550nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164284(US9669029, 34 8-Methyl-2-[2-(4-thiophen-2-yl-1H-im...)
Affinity DataIC50:  0.990nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164391(US9669029, 94 5,8-Dimethyl-2-[2-(1-methyl-4-thioph...)
Affinity DataIC50:  1nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164354(US9669029, 62 8-Methoxy-5-methyl-2-[2-(1-methyl-4-...)
Affinity DataIC50:  1.10nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164392(US9669029, 95 8-Methoxy-5-methyl-2-[2-(1-propyl-4-...)
Affinity DataIC50:  1.20nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164543(US9669029, 114 5,8-Dimethyl-2-[2-(1-methyl-4-thiaz...)
Affinity DataIC50:  1.29nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164354(US9669029, 62 8-Methoxy-5-methyl-2-[2-(1-methyl-4-...)
Affinity DataIC50:  1.5nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164396(US9669029, 99 8-Methoxy-5-methyl-2-[2-(1-methyl-4-...)
Affinity DataIC50:  1.70nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164394(US9669029, 97 4-{2-[2-(8-Methoxy-5-methyl-[1,2,4]t...)
Affinity DataIC50:  1.70nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164495(US9669029, 103 5,8-Dimethyl-2-[2-(1-methyl-4-thiaz...)
Affinity DataIC50:  2.30nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164501(US9669029, 104 5,8-Dimethyl-2-[2-(1-methyl-4-thiaz...)
Affinity DataIC50:  2.70nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164316(US9669029, 50 8-Methoxy-5-methyl-2-[(E)-2-(1-methy...)
Affinity DataIC50:  2.70nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164350(US9669029, 59 (R)-1-Chloro-3-{2-[2-(5-methyl-[1,2,...)
Affinity DataIC50:  2.80nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164536(US9669029, 111 2-[2-(4-Furan-3-yl-1-methyl-1H-imid...)
Affinity DataIC50:  2.90nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164511(US9669029, 105 8-Methoxy-5-methyl-2-{2-[1-methyl-4...)
Affinity DataIC50:  3.10nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM173102(US9096589, 5,7-Dimethyl-2-[2-(1-propyl-4-thiophen-...)
Affinity DataIC50:  3.40nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM164397(US9669029, 100 2-[2-(4-Furan-3-yl-1-methyl-1H-imid...)
Affinity DataIC50:  4nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164393(US9669029, 96 8-Methoxy-5-methyl-2-[2-(1-prop-2-yn...)
Affinity DataIC50:  4.10nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164534(US9669029, 109 5,8-Dimethyl-2-{2-[1-methyl-4-(5-me...)
Affinity DataIC50:  4.20nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164317(US9669029, 51 5,7-Dimethyl-2-[2-(1-methyl-4-thioph...)
Affinity DataIC50:  4.20nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164328(US9669029, 52 8-Methoxy-2-[2-(1-methyl-4-thiophen-...)
Affinity DataIC50:  4.5nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164532(US9669029, 107 5,8-Dimethyl-2-[2-(1-methyl-4-pyrid...)
Affinity DataIC50:  5.70nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164290(US9669029, 40 5-Methyl-2-[2-(4-thiophen-3-yl-1H-im...)
Affinity DataIC50:  5.70nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164282(US9669029, 32 1-(4-Chloro-phenyl)-2-{2-[2-(5,7-dim...)
Affinity DataIC50:  5.70nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164285(US9669029, 35 (S)-2-{2-[2-(5-Methyl-[1,2,4]triazol...)
Affinity DataIC50:  6.40nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164398(US9669029, 101 5,8-Dimethyl-2-{2-[1-methyl-4-(5-me...)
Affinity DataIC50:  6.80nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM173105(US9096589, 5,7-Dimethyl-2-{2-[1-(3-methyl-butyl)-4...)
Affinity DataIC50:  6.80nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM164539(US9669029, 113 5,8-Dimethyl-2-[2-(1-methyl-4-thiaz...)
Affinity DataIC50:  6.90nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164286(US9669029, 36 1-Methoxy-3-{2-[2-(5-methyl-[1,2,4]t...)
Affinity DataIC50:  7.5nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM173096(US9096589, 5,7-Dimethyl-2-[2-(4-thiophen-2-yl-1H-i...)
Affinity DataIC50:  7.60nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM164272(US9669029, 22 1-{2-[2-(5,7-Dimethyl-imidazo[1,2-a]...)
Affinity DataIC50:  7.90nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164380(US9669029, 83 1-Methoxy-3-{2-[2-(8-methyl-[1,2,4]t...)
Affinity DataIC50:  8.40nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM173083(US9096589, 5,7-Dimethyl-2-[(E)-2-(1-methyl-4-thiop...)
Affinity DataIC50:  8.80nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM173100(US9096589, (S)-2-{2-[2-(5,7-Dimethyl-imidazo[1,2-a...)
Affinity DataIC50:  8.80nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
In DepthDetails US Patent

LigandPNGBDBM164372(US9669029, 75 [((S)-2-Hydroxy-3-{2-[2-(5-methyl-[1...)
Affinity DataIC50:  8.80nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164533(US9669029, 108 5,8-Dimethyl-2-[2-(1-methyl-4-pyrid...)
Affinity DataIC50:  8.90nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164388(US9669029, 91 8-Methoxy-5-methyl-2-[2-(1-methyl-4-...)
Affinity DataIC50:  9.20nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164381(US9669029, 84 5-Methyl-2-[2-(1-methyl-4-thiophen-2...)
Affinity DataIC50:  9.20nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164291(US9669029, 41 5-Methyl-2-[2-(4-pyridin-3-yl-1H-imi...)
Affinity DataIC50:  9.60nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164266(US9669029, 16 5,7-Dimethyl-2-{2-[4-thiophen-2-yl-1...)
Affinity DataIC50:  9.60nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164291(US9669029, 41 5-Methyl-2-[2-(4-pyridin-3-yl-1H-imi...)
Affinity DataIC50:  9.60nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164277(US9669029, 27 2-[2-(1-Isobutyl-4-thiophen-2-yl-1H-...)
Affinity DataIC50:  12nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164531(US9669029, 106 5,8-Dimethyl-2-[2-(1-methyl-4-thiaz...)
Affinity DataIC50:  12nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

LigandPNGBDBM164371(US9669029, 74 (S)-1-{2-[2-(5-Methyl-[1,2,4]triazol...)
Affinity DataIC50:  14nMT: 25°CAssay Description:The assay is performed in 60 uL samples containing a fixed amount of the relevant PDE enzyme (sufficient to convert 20-25% of the cyclic nucleotide s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent

Displayed 1 to 50 (of 114 total ) | Next | Last >>
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