Compile Data Set for Download or QSAR
Report error Found 210 Enz. Inhib. hit(s) with all data for entry = 131
TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254598BDBM254598(US9670136, 57 N1-((trans)-2-(4-((2-fluorobenzyl)ox...)
Affinity DataIC50: 12nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254546BDBM254546(US9670136, 5 (trans)-N1-((1R,2S)-2-phenylcycloprop...)
Affinity DataIC50: 15nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 182862BDBM182862(US9670136, 2 (cis)-N1-((1S,2R)-2-phenylcyclopropyl...)
Affinity DataIC50: 17nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 183458BDBM183458(US9670136, 52 N-(4′-((trans)-2-((4-aminocycl...)
Affinity DataIC50: 19nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254574BDBM254574(US9670136, 33 N1-(2-(naphthalen-2-yl)cyclopropyl)c...)
Affinity DataIC50: 21nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254584BDBM254584(US9670136, 43 N1-((trans)-2-(4-(1H-pyrazol-5-yl)ph...)
Affinity DataIC50: 22nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254583BDBM254583(US9670136, 42 N1-((trans)-2-(4-(1H-indazol-6-yl)ph...)
Affinity DataIC50: 27nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254568BDBM254568(US9670136, 27 N1-(2-(o-tolyl)cyclopropyl)cyclohexa...)
Affinity DataIC50: 27nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254589BDBM254589(US9670136, 48 N-(4′-((trans)-2-((4-aminocycl...)
Affinity DataIC50: 27nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 183452BDBM183452(US9670136, 51 6-amino-N-(4-((trans)-2-((4-aminocyc...)
Affinity DataIC50: 30nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254586BDBM254586(US9670136, 45 3-(5-((trans)-2-((4-aminocyclohexyl)...)
Affinity DataIC50: 32nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254546BDBM254546(US9670136, 5 (trans)-N1-((1R,2S)-2-phenylcycloprop...)
Affinity DataIC50: 33nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254596BDBM254596(US9670136, 55 N1-((trans)-2-(4-((3-(piperazin-1-yl...)
Affinity DataIC50: 33nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254561BDBM254561(US9670136, 20 N1-((trans)-2-phenylcyclopropyl)-2,3...)
Affinity DataIC50: 34nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254581BDBM254581(US9670136, 40 N1-((trans)-2-(4-cyclopropylphenyl)c...)
Affinity DataIC50: 34nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254547BDBM254547(US9670136, 6 N1-((trans)-2-(thiazol-5-yl)cycloprop...)
Affinity DataIC50: 34nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254572BDBM254572(US9670136, 31 N1-(2-(2-fluorophenyl)cyclopropyl)cy...)
Affinity DataIC50: 35nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254570BDBM254570(US9670136, 29 N1-(2-(4-methoxyphenyl)cyclopropyl)c...)
Affinity DataIC50: 36nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254569BDBM254569(US9670136, 28 N1-(2-(4-(trifluoromethyl)phenyl)cyc...)
Affinity DataIC50: 37nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254573BDBM254573(US9670136, 32 N1-(2-(3,4-difluorophenyl)cyclopropy...)
Affinity DataIC50: 37nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254551BDBM254551(US9670136, 10 N1-((trans)-2-(4-(benzyloxy)phenyl)c...)
Affinity DataIC50: 40nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254585BDBM254585(US9670136, 44 3-(5-((trans)-2-((4-aminocyclohexyl)...)
Affinity DataIC50: 41nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254599BDBM254599(US9670136, 58 N1-((trans)-2-(6-((3-methylbenzyl)am...)
Affinity DataIC50: 42nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254594BDBM254594(US9670136, 53 N1-((trans)-2-fluoro-2-phenylcyclopr...)
Affinity DataIC50: 45nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254559BDBM254559(US9670136, 18 N1-((trans)-2-phenylcyclopropyl)cycl...)
Affinity DataIC50: 45nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254582BDBM254582(US9670136, 41 N1-((trans)-2-(4-(pyridin-3-yl)pheny...)
Affinity DataIC50: 47nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254575BDBM254575(US9670136, 34 N1-(2-methyl-2-phenylcyclopropyl)cyc...)
Affinity DataIC50: 47nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254550BDBM254550(US9670136, 9 N1-((trans)-2-(3′-(trifluoromet...)
Affinity DataIC50: 48nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254546BDBM254546(US9670136, 5 (trans)-N1-((1R,2S)-2-phenylcycloprop...)
Affinity DataKi:  50nM ΔG°:  -41.7kJ/molepH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254546BDBM254546(US9670136, 5 (trans)-N1-((1R,2S)-2-phenylcycloprop...)
Affinity DataKi:  50nM ΔG°:  -41.7kJ/molepH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254553BDBM254553(US9670136, 12 4-(((trans)-2-(6-(3-(trifluoromethyl...)
Affinity DataKi:  50nM ΔG°:  -41.7kJ/molepH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 182862BDBM182862(US9670136, 2 (cis)-N1-((1S,2R)-2-phenylcyclopropyl...)
Affinity DataKi:  50nM ΔG°:  -41.7kJ/molepH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254556BDBM254556(US9670136, 15 (R)-1-(4-(((trans)-2-phenylcycloprop...)
Affinity DataKi:  50nM ΔG°:  -41.7kJ/molepH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254567BDBM254567(US9670136, 26 N1-((trans)-2-(4-bromophenyl)cyclopr...)
Affinity DataIC50: 51nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254562BDBM254562(US9670136, 21 N1-((cis)-2-phenylcyclopropyl)cycloh...)
Affinity DataIC50: 53nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254579BDBM254579(US9670136, 38 (Cis)-N1-((1R,2S)-2-(3′-(trifl...)
Affinity DataIC50: 53nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254600BDBM254600(US9670136, 59 3-((5-((trans)-2-((4-aminocyclohexyl...)
Affinity DataIC50: 54nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 183448BDBM183448(US9670136, 50 N-(4′-((trans)-2-((4-aminocycl...)
Affinity DataIC50: 62nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254558BDBM254558(US9670136, 17 4-(aminomethyl)-N-((trans)-phenylcyc...)
Affinity DataIC50: 62nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254563BDBM254563(US9670136, 22 N1-methyl-N4-((trans)-2-phenylcyclop...)
Affinity DataIC50: 66nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254560BDBM254560(US9670136, 19 N1-((trans)-2-phenylcyclopropyl)cycl...)
Affinity DataIC50: 68nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254548BDBM254548(US9670136, 7 N1-((trans)-2-(pyridin-3-yl)cycloprop...)
Affinity DataIC50: 69nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254590BDBM254590(US9670136, 49 N-(3-(5-((trans)-2-((4-aminocyclohex...)
Affinity DataIC50: 79nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254556BDBM254556(US9670136, 15 (R)-1-(4-(((trans)-2-phenylcycloprop...)
Affinity DataIC50: 81nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254588BDBM254588(US9670136, 47 5-(5-((trans)-2-((4-aminocyclohexyl)...)
Affinity DataIC50: 83nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254577BDBM254577(US9670136, 36 (Cis)-N1-((1S,2R)-2-(3′-(trifl...)
Affinity DataIC50: 86nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254580BDBM254580(US9670136, 39 (Trans)-N1-((1R,2S)-2-(3′-(tri...)
Affinity DataIC50: 89nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254553BDBM254553(US9670136, 12 4-(((trans)-2-(6-(3-(trifluoromethyl...)
Affinity DataIC50: 91nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254578BDBM254578(US9670136, 37 (Trans)-N1-((1S,2R)-2-(3′-(tri...)
Affinity DataIC50: 94nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetLysine-specific histone demethylase 1A(Human)
Oryzon Genomics

US Patent
LigandChemical structure of BindingDB Monomer ID 254597BDBM254597(US9670136, 56 N1-((trans)-2-(4-(pyridin-3-ylmethox...)
Affinity DataIC50: 94nMpH: 7.4 T: 2°CAssay Description:Briefly, a fixed amount of LSD1 was incubated on ice for 15 minutes, in the absence and/or in the presence of at least eight 3-fold serial dilutions ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

Displayed 1 to 50 (of 210 total ) | Next | Last >>
Jump to: