Compile Data Set for Download or QSAR
Report error Found 171 Enz. Inhib. hit(s) with all data for entry = 132
TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183615BDBM183615(US9670142, A79 fluoro-4'-trifluoromethoxy-biph...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183609BDBM183609(US9670142, A78 biphenyl-4,4'-dicarboxylic acid...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183604BDBM183604(US9670142, A77 cyano-2'-fluoro-biphenyl-4-carb...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183588BDBM183588(US9670142, A76 4-(1H-benzimidazol-5-yl)-N-methyl-N...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183578BDBM183578(US9670142, A75 N-methyl-4-(1-methyl-1H-indazol-5-y...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183576BDBM183576(US9670142, A74 N-methyl-4-(1-methyl-1H-indazol-6-y...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183575BDBM183575(US9670142, A73 4'-methyl-biphenyl-4-carboxylic...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183572BDBM183572(US9670142, A72 N-methyl-N-((1R,3S)-3-propionylamin...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183634BDBM183634(US9670142, A87 4-(2,3-dihydro-benzo[1,4]dioxin-6-y...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183633BDBM183633(US9670142, A86 4'-chloro-3'-fluoro-bipheny...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183632BDBM183632(US9670142, A85 4'-difluoromethoxy-biphenyl-4-c...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183628BDBM183628(US9670142, A84 4-(1H-indazol-5-yl)-N-methyl-N-((1R...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183626BDBM183626(US9670142, A83 2',4'-difluoro-biphenyl-4-c...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183625BDBM183625(US9670142, A82 4'-methoxy-biphenyl-4-carboxyli...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183624BDBM183624(US9670142, A81 4'-(2H-pyrazol-3-yl)-biphenyl-4...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183616BDBM183616(US9670142, A80 N-methyl-4-(1-methyl-1H-indol-5-yl)...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184410BDBM184410(US9670142, A95 4-(1H-indol-5-yl)-N-methyl-N-((1R,3...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184409BDBM184409(US9670142, A94 N-methyl-4-(2-oxo-2,3-dihydro-1H-in...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184408BDBM184408(US9670142, A93 N-methyl-4-(2-oxo-2,3-dihydro-1H-be...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184407BDBM184407(US9670142, A92 4'-chloro-2'-fluoro-bipheny...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184406BDBM184406(US9670142, A91 4-(1H-benzotriazol-5-yl)-N-methyl-N...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184405BDBM184405(US9670142, A90 2',4'-dimethyl-biphenyl-4-c...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183639BDBM183639(US9670142, A88 2',4'-dimethoxy-biphenyl-4-...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184478BDBM184478(US9670142, A102 N-methyl-4-(6-methyl-1H-indazol-5-...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184418BDBM184418(US9670142, A101 4-(1H-indol-5-yl)-3,N-dimethyl-N-(...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184416BDBM184416(US9670142, A100 N-methyl-4-(3-methyl-1H-indazol-5-...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184415BDBM184415(US9670142, A99a 4-(3-cyano-1H-indol-5-yl)-N-methyl...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184414BDBM184414(US9670142, A99 2'-fluoro-4'-methoxy-biphen...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 183615BDBM183615(US9670142, A79 fluoro-4'-trifluoromethoxy-biph...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184412BDBM184412(US9670142, A97 2-fluoro-4'-[methyl-((1R,3S)-3-...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184540BDBM184540(US9670142, A110 5-(1-methyl-1H-indol-5-yl)-pyridin...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184539BDBM184539(US9670142, A109 5-(1H-indol-5-yl)-pyridine-2-carbo...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184538BDBM184538(US9670142, A108 3-fluoro-N-methyl-4-(1-methyl-1H-i...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184537BDBM184537(US9670142, A107 N-methyl-4-(7-methyl-1H-indazol-5-...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184499BDBM184499(US9670142, A106 2-fluoro-4-(1H-indol-5-yl)-N-methy...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184493BDBM184493(US9670142, A105 5-(3-methyl-1H-indazol-5-yl)-pyrid...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184492BDBM184492(US9670142, A104 5-(7-methyl-1H-indazol-5-yl)-pyrid...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 185360BDBM185360(US9670142, A118 6-(1-methyl-1H-indol-5-yl)-pyridaz...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 185359BDBM185359(US9670142, A117 6-(1H-indol-5-yl)-N-methyl-N-((1R,...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184615BDBM184615(US9670142, A116 4-(4-fluoro-1H-indol-5-yl)-N-methy...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184585BDBM184585(US9670142, A115 N-methyl-4-(3-methyl-1H-indol-5-yl...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184573BDBM184573(US9670142, A114 3,N-dimethyl-4-(1-methyl-1H-indol-...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184550BDBM184550(US9670142, A113 6-(1H-indol-5-yl)-pyridazine-3-car...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184547BDBM184547(US9670142, A112 3-fluoro-4-(1H-indol-5-yl)-N-methy...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 184541BDBM184541(US9670142, A111 2-fluoro-N-methyl-4-(1-methyl-1H-i...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 185540BDBM185540(US9670142, A126 N-methyl-4-(4-methyl-1H-indazol-5-...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 185537BDBM185537(US9670142, A125 5-(1-methyl-1H-indol-5-yl)-pyrazin...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 185533BDBM185533(US9670142, A124 3,N-dimethyl-4-(4-methyl-1H-indazo...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 185520BDBM185520(US9670142, A123 N-methyl-4-(1-methyl-1H-benzimidaz...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

TargetFatty acid synthase(Human)
Merck Patent

US Patent
LigandChemical structure of BindingDB Monomer ID 185518BDBM185518(US9670142, A122 4-(6-fluoro-1H-indol-5-yl)-N-methy...)
Affinity DataIC50: 300nMpH: 7.0 T: 2°CAssay Description:The biochemical FASN activity testing was performed as 384 well two-time-point kinetic fluorescence intensity assay format in Greiner low volume medi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2018
Entry Details
US Patent

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