Compile Data Set for Download or QSAR
Report error Found 211 Enz. Inhib. hit(s) with all data for entry = 147
TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 191570BDBM191570(US9670204, 12 2-((2-ethyl-8-fluoro-6-(4-(2-(3-hydr...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192616BDBM192616(US9670204, 115 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192950BDBM192950(US9670204, 145 2-(4-(3-((5-cyano-4-(4-fluorophenyl...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192949BDBM192949(US9670204, 144 2-((2-ethyl-6-(1-(2-(3-(hydroxymeth...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192948BDBM192948(US9670204, 143 (S)-2-((2-ethyl-6-(1-(2-(3-hydroxyp...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 191618BDBM191618(US9670204, 22 2-(4-(3-((5-cyano-4-(4-fluorophenyl)...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192986BDBM192986(US9670204, 166 2-(2-((2-ethyl-6-(4-(2-(3-hydroxyaz...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192984BDBM192984(US9670204, 164 2-(2-((2-ethyl-6-(4-(2-(3-fluoroaze...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 191788BDBM191788(US9670204, 31 2-(4-(2-ethyl-3-((4-(4-fluorophenyl)...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 191784BDBM191784(US9670204, 30 1-(azetidin-1-yl)-2-(4-(2-ethyl-3-((...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192979BDBM192979(US9670204, 159 1-(2-((2-ethyl-6-(1-(2-(3-hydroxyaz...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192947BDBM192947(US9670204, 142 (R)-2-((2-ethyl-6-(1-(2-(3-hydroxyp...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192994BDBM192994(US9670204, 174 2-(4-(2-(2-cyanoethyl)-3-((4-(4-flu...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192946BDBM192946(US9670204, 141 2-((2-ethyl-6-(1-(2-(3-hydroxyazeti...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192993BDBM192993(US9670204, 173 2-(5-((2-ethyl-6-(1-(2-(3-hydroxyaz...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192945BDBM192945(US9670204, 140 2-(4-(3-((5-cyano-4-(4-fluorophenyl...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192944BDBM192944(US9670204, 139 2-((2-ethyl-6-(4-(2-(3-(hydroxymeth...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192991BDBM192991(US9670204, 171 2-(4-(3-((4-(2-cyano-4-fluorophenyl...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192943BDBM192943(US9670204, 138 2-((2-ethyl-6-(4-(2-(3-hydroxyazeti...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192990BDBM192990(US9670204, 170 2-(2-((2-ethyl-6-(1-(2-(3-hydroxyaz...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192989BDBM192989(US9670204, 169 2-(4-(3-((4-(2-cyano-4-fluorophenyl...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192988BDBM192988(US9670204, 168 2-(4-(3-((4-(2-cyano-4-fluorophenyl...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192987BDBM192987(US9670204, 167 2-(2-((6-(4-(2-(azetidin-1-yl)-2-ox...)
Affinity DataIC50: 50nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192998BDBM192998(US9670204, 178 2-(1-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 191867BDBM191867(US9670204, 72 N-(2-ethyl-6-(1-(methylsulfonyl)-1,2...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 193337BDBM193337(US9670204, 215 1-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192219BDBM192219(US9670204, 93 3-(4-(2-ethyl-3-((4-(4-fluorophenyl)...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 193359BDBM193359(US9670204, 223 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192212BDBM192212(US9670204, 89 N-(2-ethyl-6-(1-(3-(pyrrolidin-1-yl)...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192192BDBM192192(US9670204, 88 N-(2-ethyl-6-(1-(3-morpholinopropyl-...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192190BDBM192190(US9670204, 87 N-(6-(1-(3-(dimethylamino)propyl-sul...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192272BDBM192272(US9670204, 97 2-(2-((2-ethyl-6-(1-(methylsulfonyl)...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192268BDBM192268(US9670204, 96 2-(2-((2-ethyl-6-(1-(methylsulfonyl)...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192475BDBM192475(US9670204, 109 ethyl2-(4-(2-ethyl-3-((4-(4-fluorop...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192311BDBM192311(US9670204, 105 1-(2-((2-ethyl-6-(1-(methylsulfonyl...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192297BDBM192297(US9670204, 103 4-(4-fluorophenyl)-N-(2-ethyl-6-(1-...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192772BDBM192772(US9670204, 117 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192620BDBM192620(US9670204, 116 (S)-1-(2-(4-(2-ethyl-3-((4-(4-fluor...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192615BDBM192615(US9670204, 114 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192614BDBM192614(US9670204, 113 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192613BDBM192613(US9670204, 112 (S)-2-(4-(2-ethyl-3-((4-(4-fluoroph...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192576BDBM192576(US9670204, 111 (R)-2-(4-(2-ethyl-3-((4-(4-fluoroph...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192476BDBM192476(US9670204, 110 2-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192791BDBM192791(US9670204, 126 1-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192775BDBM192775(US9670204, 118 4-((4-(2-ethyl-3-((4-(4-fluoropheny...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192919BDBM192919(US9670204, 133 1-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192917BDBM192917(US9670204, 131 2-(3,3-dimethylazetidin-1-yl)-1-(4-...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192916BDBM192916(US9670204, 130 3-(dimethylamino)-1-(4-(2-ethyl-3-(...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192915BDBM192915(US9670204, 129 2-(dimethylamino)-1-(4-(2-ethyl-3-(...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

TargetAutotaxin(Human)
Galapagos

US Patent
LigandChemical structure of BindingDB Monomer ID 192914BDBM192914(US9670204, 128 1-(4-(2-ethyl-3-((4-(4-fluorophenyl...)
Affinity DataIC50: 300nMpH: 8.5 T: 2°CAssay Description:Compound IC50 values are determined in a hENPP2 (UniProtKB/SwissProt Sequence ref Q13822) biochemical assay using LPC as substrate. 5 μL of a di...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/7/2018
Entry Details
US Patent

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