Compile Data Set for Download or QSAR
Report error Found 342 Enz. Inhib. hit(s) with all data for entry = 159
TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 193371BDBM193371(2-(((4-(difluoromethoxy)phenyl)amino)methyl)-5-(4-...)
Affinity DataIC50: 334nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 196331BDBM196331(2-(((3,4-difluorophenyl)amino)methyl)-5-(4-fluorop...)
Affinity DataIC50: 462nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197278BDBM197278(5-(4-fluorophenyl)-2-(((4-fluorophenyl)(methyl)ami...)
Affinity DataIC50: 467nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 196596BDBM196596(2-(((4-(difluoromethoxy)-3-fluorophenyl)amino)meth...)
Affinity DataIC50: 489nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 191594BDBM191594(2-(((3-(difluoromethoxy)phenyl)amino)methyl)-5-(4-...)
Affinity DataIC50: 505nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 196291BDBM196291(2-(((2,5-difluorophenyl)amino)methyl)-5-(4-fluorop...)
Affinity DataIC50: 508nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197965BDBM197965(2-(((4-(difluoromethoxy)-2-fluorophenyl)amino)meth...)
Affinity DataIC50: 578nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197329BDBM197329(5-(4-chlorophenyl)-2-(((4-methoxyphenyl)(methyl)am...)
Affinity DataIC50: 585nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 193379BDBM193379(2-(((2,3-difluorophenyl)amino)methyl)-5-(4-fluorop...)
Affinity DataIC50: 586nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197328BDBM197328(US9676782, 95)
Affinity DataIC50: 588nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197324BDBM197324(2-(((4-bromophenyl)(methyl)amino)methyl)-5-(4-fluo...)
Affinity DataIC50: 592nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197196BDBM197196(5-(4-fluorophenyl)-2-(((3-fluorophenyl)(methyl)ami...)
Affinity DataIC50: 594nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 198682BDBM198682(2-(((5-chloropyridin-2-yl)amino)methyl)-5-(4-fluor...)
Affinity DataIC50: 602nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197950BDBM197950(2-(((4-(difluoromethoxy)-2-fluorophenyl)amino)meth...)
Affinity DataIC50: 624nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197327BDBM197327(2-(((3,5-difluorophenyl)(methyl)amino)methyl)-5-(4...)
Affinity DataIC50: 660nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197331BDBM197331(5-(3-chlorophenyl)-2-(((4-methoxyphenyl)(methyl)am...)
Affinity DataIC50: 668nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197332BDBM197332(2-(((4-methoxyphenyl)(methyl)amino)methyl)-5-(p-to...)
Affinity DataIC50: 675nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197956BDBM197956(2-(((4-(difluoromethoxy)-2-fluorophenyl)amino)meth...)
Affinity DataIC50: 706nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 193371BDBM193371(2-(((4-(difluoromethoxy)phenyl)amino)methyl)-5-(4-...)
Affinity DataIC50: 709nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 196309BDBM196309(2-(((3,5-difluorophenyl)amino)methyl)-5-(4-fluorop...)
Affinity DataIC50: 738nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 196750BDBM196750((r)-2-(((2,4-difluorophenyl)amino)methyl)-5-(4-flu...)
Affinity DataIC50: 771nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 198263BDBM198263(2-(((4-(difluoromethoxy)-2-fluorophenyl)amino)meth...)
Affinity DataIC50: 772nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197333BDBM197333(5-(2-chlorophenyl)-2-(((4-methoxyphenyl)(methyl)am...)
Affinity DataIC50: 777nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197334BDBM197334(5-(3-fluorophenyl)-2-(((4-methoxyphenyl)(methyl)am...)
Affinity DataIC50: 783nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 196567BDBM196567(2-(((2-fluoro-4-methylphenyl)amino)methyl)-5-(4-fl...)
Affinity DataIC50: 799nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197963BDBM197963(2-(((4-(difluoromethoxy)-2-fluorophenyl)amino)meth...)
Affinity DataIC50: 800nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197335BDBM197335(2-(((4-methoxyphenyl)(methyl)amino)methyl)-5-(2,4,...)
Affinity DataIC50: 801nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197231BDBM197231(2-(((3-chlorophenyl)(methyl)amino)methyl)-5-(4-flu...)
Affinity DataIC50: 805nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197338BDBM197338(2-(((4-methoxyphenyl)(methyl)amino)methyl)-5-(m-to...)
Affinity DataIC50: 805nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197945BDBM197945(2-(((4-(difluoromethoxy)-2-fluorophenyl)amino)meth...)
Affinity DataIC50: 821nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 196552BDBM196552(2-(((4-chloro-2-fluorophenyl)amino)methyl)-5-(4-fl...)
Affinity DataIC50: 856nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197339BDBM197339(5-(3,5-difluorophenyl)-2-(((4-methoxyphenyl)(methy...)
Affinity DataIC50: 856nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197957BDBM197957(2-(((4-(difluoromethoxy)-2-fluorophenyl)amino)meth...)
Affinity DataIC50: 863nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 196608BDBM196608((r)-5-(4-fluorophenyl)-2-(((2-fluorophenyl)amino)m...)
Affinity DataIC50: 871nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197346BDBM197346(5-(2-fluorophenyl)-2-(((4-methoxyphenyl)(methyl)am...)
Affinity DataIC50: 871nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 196832BDBM196832(5-(4-fluorophenyl)-2-(((2-fluorophenyl)(methyl)ami...)
Affinity DataIC50: 876nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197323BDBM197323(2-(((4-chlorophenyl)(methyl)amino)methyl)-5-(4-flu...)
Affinity DataIC50: 885nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 193377BDBM193377(2-(4-(((5-(4-fluorophenyl)-4-oxo-4,5,6,7-tetrahydr...)
Affinity DataIC50: 890nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197636BDBM197636(5-(5-chloropyridin-2-yl)-2-(((4-methoxyphenyl)(met...)
Affinity DataIC50: 917nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197969BDBM197969(5-(5-chloropyridin-2-yl)-2-(((4-(difluoromethoxy)-...)
Affinity DataIC50: 930nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197972BDBM197972(2-(((4-(difluoromethoxy)-2-fluorophenyl)amino)meth...)
Affinity DataIC50: 943nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 191566BDBM191566(5-(4-fluorophenyl)-2-(((2-fluorophenyl)amino)methy...)
Affinity DataIC50: 944nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197958BDBM197958(2-(((4-(difluoromethoxy)-2-fluorophenyl)amino)meth...)
Affinity DataIC50: 950nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197325BDBM197325(5-(4-fluorophenyl)-2-(((4-methoxyphenyl)(methyl)am...)
Affinity DataIC50: 986nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197347BDBM197347(US9676782, 110 | 5-(2,5-difluorophenyl)-2-(((4-met...)
Affinity DataIC50: 1.02E+3nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197243BDBM197243(5-(4-fluorophenyl)-2-(((3-methoxyphenyl)(methyl)am...)
Affinity DataIC50: 1.02E+3nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197369BDBM197369(5-(2,3-difluorophenyl)-2-(((4-methoxyphenyl)(methy...)
Affinity DataIC50: 1.03E+3nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 197635BDBM197635(5-(4-(difluoromethoxy)phenyl)-2-(((4-methoxyphenyl...)
Affinity DataIC50: 1.03E+3nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 191575BDBM191575(5-(4-fluorophenyl)-2-(((3-fluorophenyl)amino)methy...)
Affinity DataIC50: 1.04E+3nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

TargetMetabotropic glutamate receptor 3(Rat)
Vanderbilt University

US Patent
LigandChemical structure of BindingDB Monomer ID 196363BDBM196363(2-(((2,6-difluorophenyl)amino)methyl)-5-(4-fluorop...)
Affinity DataIC50: 1.05E+3nMT: 2°CAssay Description:HEK 293A cells stably expressing rat mGlu5 were plated in black-walled, clear-bottomed, poly-D-lysine coated 384-well plates in 20 μL of assay m...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/7/2018
Entry Details
US Patent

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