Compile Data Set for Download or QSAR
Report error Found 34 Enz. Inhib. hit(s) with all data for entry = 84
TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 50296329BDBM50296329((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(2-phe...)
Affinity DataIC50: 2.70nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228865BDBM228865(Ipratropium | US9333195, IPRATROPIUM)
Affinity DataIC50: 3nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228855BDBM228855(US9687478, 77 | US9333195, 77)
Affinity DataIC50: 3.10nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 200229BDBM200229(Atropine | AB00694549-11 | cid_174174)
Affinity DataIC50: 3.20nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 50296330BDBM50296330((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(4-phe...)
Affinity DataIC50: 3.80nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 50296331BDBM50296331((3R)-3-{[Hydroxy(di-2-thienyl)acetyl]oxy}-1-(3-phe...)
Affinity DataIC50: 4.40nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228848BDBM228848(US9687478, 8 | US9333195, 8)
Affinity DataIC50: 4.80nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228856BDBM228856(US9687478, 78 | US9333195, 78)
Affinity DataIC50: 5nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 50296341BDBM50296341((3R)-3-{[Hydroxy(di-3-thienyl)acetyl]oxy}-1-(3-phe...)
Affinity DataIC50: 5.40nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228852BDBM228852(US9687478, 53 | US9333195, 53)
Affinity DataIC50: 5.60nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162552BDBM162552(US9687478, 129)
Affinity DataIC50: 6.30nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228850BDBM228850(US9687478, 18 | US9333195, 18)
Affinity DataIC50: 6.60nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228851BDBM228851(US9687478, 20 | US9333195, 20)
Affinity DataIC50: 6.80nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162554BDBM162554(US9687478, 137)
Affinity DataIC50: 6.90nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162484BDBM162484(US9687478, 100)
Affinity DataIC50: 7.60nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228853BDBM228853(US9687478, 71 | US9333195, 71)
Affinity DataIC50: 8.20nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162551BDBM162551(US9687478, 128)
Affinity DataIC50: 8.80nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228857BDBM228857(US9687478, 84 | US9333195, 84)
Affinity DataIC50: 9.90nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162553BDBM162553(US9687478, 136)
Affinity DataIC50: 11nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162549BDBM162549(US9687478, 126)
Affinity DataIC50: 13nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 50296340BDBM50296340((3R)-3-[(Di-2-thienylacetyl)oxy]-1-(3-phenoxypropy...)
Affinity DataIC50: 13nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162556BDBM162556(US9687478, 146)
Affinity DataIC50: 13nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162520BDBM162520(US9687478, 114)
Affinity DataIC50: 14nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228849BDBM228849(US9687478, 17 | US9333195, 17)
Affinity DataIC50: 14nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162483BDBM162483(US9687478, 101)
Affinity DataIC50: 14nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 50296335BDBM50296335((3R)-3-{[Hydroxy(diphenyl)acetyl]oxy}-1-(3-phenoxy...)
Affinity DataIC50: 15nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162550BDBM162550(US9687478, 127)
Affinity DataIC50: 16nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228854BDBM228854(US9687478, 74 | US9333195, 74)
Affinity DataIC50: 16nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162555BDBM162555(US9687478, 138)
Affinity DataIC50: 19nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 228847BDBM228847(US9687478, 7 | US9333195, 7)
Affinity DataIC50: 22nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162543BDBM162543(US9687478, 116)
Affinity DataIC50: 23nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162519BDBM162519(US9687478, 109)
Affinity DataIC50: 31nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162478BDBM162478(US9687478, 99)
Affinity DataIC50: 31nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent

TargetMuscarinic acetylcholine receptor M3(Human)
Almirall

US Patent
LigandChemical structure of BindingDB Monomer ID 162365BDBM162365(US9687478, 1)
Affinity DataIC50: 31nMT: 2°CAssay Description:Assays were carried out at 25° C. Membrane preparations from stably transfected chinese hamster ovary-K1 cells (CHO) expressing the genes for the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/10/2018
Entry Details
US Patent