Compile Data Set for Download or QSAR
Report error Found 150 Enz. Inhib. hit(s) with all data for entry = 103
TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174126BDBM174126(US9688668, 1a)
Affinity DataKi:  100nMAssay Description:SLR080811, prepared as the HCl salt, was tested first at recombinant SphK1 and SphK2 using a broken cell assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174053BDBM174053(US9688668, 20)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174050BDBM174050(US9688668, 17)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174059BDBM174059(US9688668, 24)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174056BDBM174056(US9688668, 23)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174055BDBM174055(US9688668, 22)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174054BDBM174054(US9688668, 21)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174064BDBM174064(US9688668, 28)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174063BDBM174063(US9688668, 27)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174061BDBM174061(US9688668, 26)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174060BDBM174060(US9688668, 25)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174049BDBM174049(US9688668, 16)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174068BDBM174068(US9688668, 32)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174114BDBM174114(US9688668, 64)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174047BDBM174047(US9688668, 15)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174067BDBM174067(US9688668, 31)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174046BDBM174046(US9688668, 14)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174066BDBM174066(US9688668, 30)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174044BDBM174044(US9688668, 13)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174065BDBM174065(US9688668, 29)
Affinity DataKi: <1.00E+3nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 50443388BDBM50443388(CHEMBL3086782 | US9688668, SLR080811)
Affinity DataKi:  1.30E+3nMAssay Description:SLR080811, prepared as the HCl salt, was tested first at recombinant SphK1 and SphK2 using a broken cell assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174126BDBM174126(US9688668, 1a)
Affinity DataKi:  1.50E+3nMAssay Description:SLR080811, prepared as the HCl salt, was tested first at recombinant SphK1 and SphK2 using a broken cell assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174052BDBM174052(US9688668, 19)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174052BDBM174052(US9688668, 19)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174051BDBM174051(US9688668, 18)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174051BDBM174051(US9688668, 18)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174049BDBM174049(US9688668, 16)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174072BDBM174072(US9688668, 36)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174071BDBM174071(US9688668, 35)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174071BDBM174071(US9688668, 35)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174070BDBM174070(US9688668, 34)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174069BDBM174069(US9688668, 33)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174069BDBM174069(US9688668, 33)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174076BDBM174076(US9688668, 40)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174075BDBM174075(US9688668, 39)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174075BDBM174075(US9688668, 39)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174074BDBM174074(US9688668, 38)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174074BDBM174074(US9688668, 38)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174073BDBM174073(US9688668, 37)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174073BDBM174073(US9688668, 37)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174072BDBM174072(US9688668, 36)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174083BDBM174083(US9688668, 44)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174082BDBM174082(US9688668, 43)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174082BDBM174082(US9688668, 43)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174080BDBM174080(US9688668, 42)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174080BDBM174080(US9688668, 42)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174079BDBM174079(US9688668, 41)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 1(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174079BDBM174079(US9688668, 41)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174076BDBM174076(US9688668, 40)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

TargetSphingosine kinase 2(Human)
University of Virginia Patent Foundation

US Patent
LigandChemical structure of BindingDB Monomer ID 174085BDBM174085(US9688668, 46)
Affinity DataKi: >1.00E+4nMAssay Description:SphK activity was measured by a scintillation proximity assay as previously described [1], the disclosure of which is incorporated herein. Briefly, r...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2018
Entry Details
US Patent

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