Compile Data Set for Download or QSAR
Report error Found 17 Enz. Inhib. hit(s) with all data for entry = 51
LigandChemical structure of BindingDB Monomer ID 107635BDBM107635(US9695179, 1)
Affinity DataIC50: 2.43E+3nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111137BDBM111137(US9695179, 132)
Affinity DataIC50: 3.70E+3nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111102BDBM111102(US9695179, 97)
Affinity DataIC50: 5.80E+3nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111103BDBM111103(US9695179, 98)
Affinity DataIC50: 6.70E+3nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111126BDBM111126(US9695179, 121)
Affinity DataIC50: 7.30E+3nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111094BDBM111094(US9695179, 90)
Affinity DataIC50: 1.12E+4nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111133BDBM111133(US9695179, 128)
Affinity DataIC50: 1.63E+4nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111129BDBM111129(US9695179, 124)
Affinity DataIC50: 1.73E+4nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111131BDBM111131(US9695179, 126)
Affinity DataIC50: 2.36E+4nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 89915BDBM89915((6-chloro-2-oxo-4-phenyl-1H-quinolin-3-yl) N,N-die...)
Affinity DataIC50: 2.68E+4nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111090BDBM111090(US9695179, 87)
Affinity DataIC50: 1.39E+5nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111087BDBM111087(US9695179, 84)
Affinity DataIC50: 3.72E+5nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111086BDBM111086(US9695179, 83)
Affinity DataIC50: 4.42E+5nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111093BDBM111093(US9695179, 89)
Affinity DataIC50: 5.86E+5nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111089BDBM111089(US9695179, 86)
Affinity DataIC50: 6.70E+5nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111092BDBM111092(US9695179, 88)
Affinity DataIC50: 8.64E+5nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 111088BDBM111088(US9695179, 85)
Affinity DataIC50: 8.76E+5nMT: 2°CAssay Description:The interactions between test compounds and BRD4 protein containing both bromodomain 1 and bromodomain 2 were measured with human BRD4 protein with N...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent