Compile Data Set for Download or QSAR
Report error Found 374 Enz. Inhib. hit(s) with all data for entry = 249
TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247123BDBM247123(3-((4-((4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
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Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247059BDBM247059(3-((4-((4-(3-(3-(tert-Butyl)-1-(p-tolyl)-1H-pyrazo...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247091BDBM247091(N-(2-(dimethylamino)ethyl)-4-((4-((4-(3-(3-isoprop...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247123BDBM247123(3-((4-((4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
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TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247091BDBM247091(N-(2-(dimethylamino)ethyl)-4-((4-((4-(3-(3-isoprop...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247106BDBM247106(3-methoxy-5-((4-((4-(3-(3-(1-methylcyclopropyl)-1-...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
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Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247090BDBM247090(N-(2-hydroxyethyl)-3-((4-((4-(3-(3-isopropyl-1-(4-...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247061BDBM247061(N-(2-(Dimethylamino)ethyl)-3-((4-((4-(3-(3-isoprop...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247108BDBM247108(3-((4-((4-(3-(3-isopropyl-1-(4-methoxyphenyl)-1H-p...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247124BDBM247124(1-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)-3-(4-(...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247079BDBM247079(3-((4-((4-(3-(1-(4-methoxyphenyl)-3-(3-methyloxeta...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
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Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247111BDBM247111(3-((4-((4-(3-(1-(3,4-dimethylphenyl)-3-isopropyl-1...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247127BDBM247127(3-((6-((4-(3-(3-(tert-butyl)-1-(p-tolyl)-1H-pyrazo...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247079BDBM247079(3-((4-((4-(3-(1-(4-methoxyphenyl)-3-(3-methyloxeta...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247126BDBM247126(3-((6-((4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247078BDBM247078(3-((4-((4-(3-(3-(3-methyloxetan-3-yl)-1-(p-tolyl)-...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247062BDBM247062(N-(2-(Dimethylamino)ethyl)-3-((4-((4-(3-(3-isoprop...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247078BDBM247078(3-((4-((4-(3-(3-(3-methyloxetan-3-yl)-1-(p-tolyl)-...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247113BDBM247113(3-methoxy-5-((4-((4-(3-(1-(4-methoxyphenyl)-3-(tet...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
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TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247113BDBM247113(3-methoxy-5-((4-((4-(3-(1-(4-methoxyphenyl)-3-(tet...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247112BDBM247112(3-((4-((4-(3-(3-(tert-butyl)-1-(6-methoxypyridin-3...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247064BDBM247064(3-((4-((4-(3-(3-Isopropyl-1-(p-tolyl)-1H-pyrazol-5...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247080BDBM247080(3-((4-((4-(3-(3-(tert-butyl)-1-(4-methylthiophen-2...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247114BDBM247114(3-methoxy-5-((4-((4-(3-(1-(4-methoxyphenyl)-3-(tet...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247085BDBM247085(3-((4-((4-(3-(3-(tert-butyl)-1-(p-tolyl)-1H-pyrazo...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247085BDBM247085(3-((4-((4-(3-(3-(tert-butyl)-1-(p-tolyl)-1H-pyrazo...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247084BDBM247084(N-(2-(dimethylamino)ethyl)-3-((4-((4-(3-(3-isoprop...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247084BDBM247084(N-(2-(dimethylamino)ethyl)-3-((4-((4-(3-(3-isoprop...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247100BDBM247100(3-((4-((4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247086BDBM247086(3-((4-((4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247070BDBM247070(3-((6-((4-(3-(3-isopropyl-1-(4-methoxyphenyl)-1H-p...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247105BDBM247105(3-((4-((4-(3-(3-cyclopropyl-1-(p-tolyl)-1H-pyrazol...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247104BDBM247104(3-((4-((4-(3-(3-ethyl-1-(p-tolyl)-1H-pyrazol-5-yl)...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247088BDBM247088(N-(2-hydroxyethyl)-3-((4-((4-(3-(3-isopropyl-1-(p-...)
Affinity DataIC50: 1nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247129BDBM247129(3-((6-(4-(3-(3-(tert-Butyl)-1-(4-methoxyphenyl)-1H...)
Affinity DataIC50: 1.30nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247075BDBM247075(3-((4-((4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247099BDBM247099(3-((4-((4-(3-(3-(tert-butyl)-1-(p-tolyl)-1H-pyrazo...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247075BDBM247075(3-((4-((4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247066BDBM247066(3-((4-((4-(3-(3-Isopropyl-1-(6-methoxypyridin-3-yl...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247090BDBM247090(N-(2-hydroxyethyl)-3-((4-((4-(3-(3-isopropyl-1-(4-...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247114BDBM247114(3-methoxy-5-((4-((4-(3-(1-(4-methoxyphenyl)-3-(tet...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247109BDBM247109(3-((4-((4-(3-(3-(tert-butyl)-1-(4-methoxyphenyl)-1...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247125BDBM247125(5-((4-((4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247061BDBM247061(N-(2-(Dimethylamino)ethyl)-3-((4-((4-(3-(3-isoprop...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247069BDBM247069(5-((4-((4-(3-(3-(tert-Butyl)-1-(p-tolyl)-1H-pyrazo...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247076BDBM247076(3-((4-((4-(3-(3-isopropyl-1-(4-methoxyphenyl)-1H-p...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247108BDBM247108(3-((4-((4-(3-(3-isopropyl-1-(4-methoxyphenyl)-1H-p...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetMitogen-activated protein kinase 14(Human)
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LigandChemical structure of BindingDB Monomer ID 247124BDBM247124(1-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5-yl)-3-(4-(...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of test compounds against the p38 MAPKα isoform (MAPK14: Invitrogen), are evaluated indirectly by determining the leve...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetTyrosine-protein kinase SYK(Human)
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LigandChemical structure of BindingDB Monomer ID 247123BDBM247123(3-((4-((4-(3-(3-isopropyl-1-(p-tolyl)-1H-pyrazol-5...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of compounds of the invention against Syk enzymes (Invitrogen), are evaluated in a similar fashion to that described herein...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

TargetProto-oncogene tyrosine-protein kinase Src(Human)
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LigandChemical structure of BindingDB Monomer ID 247119BDBM247119(3-((4-((4-(3-(3-(tert-butyl)-1-(p-tolyl)-1H-pyrazo...)
Affinity DataIC50: 2nMAssay Description:The inhibitory activities of compounds of the invention against c-Src and Syk enzymes (Invitrogen), are evaluated in a similar fashion to that descri...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

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