Compile Data Set for Download or QSAR
Report error Found 77 Enz. Inhib. hit(s) with all data for entry = 250
LigandChemical structure of BindingDB Monomer ID 253625BDBM253625(US9701672, 56)
Affinity DataIC50: 0.200nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253635BDBM253635(US9701672, 66)
Affinity DataIC50: 0.5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253632BDBM253632(US9701672, 63)
Affinity DataIC50: 0.700nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247150BDBM247150(US9701672, 4 | (S,E)-2-Methyl-N-(2,2,2-trifluoro-1...)
Affinity DataIC50: 0.900nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247150BDBM247150(US9701672, 4 | (S,E)-2-Methyl-N-(2,2,2-trifluoro-1...)
Affinity DataIC50: 1.10nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253633BDBM253633(US9701672, 64)
Affinity DataIC50: 1.10nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247168BDBM247168(1-(5-Cyclopropylthiazol-2-yl)ethanone | US9701672,...)
Affinity DataIC50: 1.20nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253628BDBM253628(US9701672, 59)
Affinity DataIC50: 1.40nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253626BDBM253626(US9701672, 57)
Affinity DataIC50: 1.40nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247154BDBM247154(1-(5-Methylthiazol-2-yl)ethanone | US9701672, 8)
Affinity DataIC50: 1.5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253649BDBM253649((S)—N-(4-(5-Ethylthiophen-2-yl)-2-oxo-6-(4-((...)
Affinity DataIC50: 1.5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247169BDBM247169(1-(5-Ethylthiazol-2-yl)ethanone | US9701672, 23)
Affinity DataIC50: 2.10nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253631BDBM253631(US9701672, 62)
Affinity DataIC50: 2.10nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247152BDBM247152(1-(5-Cyclopropylthiophen-2-yl)ethanone | US9701672...)
Affinity DataIC50: 2.20nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253627BDBM253627(US9701672, 58)
Affinity DataIC50: 2.20nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247056BDBM247056((S,E)-2-Methyl-N-(2,2,2-trifluoro-1-(4-(4,4,4-trif...)
Affinity DataIC50: 2.5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 252410BDBM252410(US9701672, 47)
Affinity DataIC50: 2.70nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 249008BDBM249008(US9701672, 30)
Affinity DataIC50: 2.70nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 249861BDBM249861(US9701672, 42)
Affinity DataIC50: 3nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253621BDBM253621(US9701672, 52)
Affinity DataIC50: 3.20nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 251745BDBM251745(US9701672, 45)
Affinity DataIC50: 3.5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253652BDBM253652(US9701672, 76)
Affinity DataIC50: 4.20nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253618BDBM253618(US9701672, 49)
Affinity DataIC50: 4.5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 249850BDBM249850(US9701672, 40)
Affinity DataIC50: 6.70nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253624BDBM253624(US9701672, 55)
Affinity DataIC50: 7.80nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247151BDBM247151((S,E)-2-Methyl-N-(1,1,1-trifluorodec-3-yn-2-yliden...)
Affinity DataIC50: 7.80nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253634BDBM253634(US9701672, 65)
Affinity DataIC50: 8.80nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 251746BDBM251746(US9701672, 48 | US9701672, 46)
Affinity DataIC50: 8.80nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247153BDBM247153(1-(5-((Dimethylamino)methyl)thiophen-2-yl)ethanone...)
Affinity DataIC50: 9nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253619BDBM253619(US9701672, 50)
Affinity DataIC50: 9.40nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253643BDBM253643(US9701672, 72)
Affinity DataIC50: 10.3nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 251746BDBM251746(US9701672, 48 | US9701672, 46)
Affinity DataIC50: 11.4nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 249130BDBM249130(US9701672, 35)
Affinity DataIC50: 11.5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 249535BDBM249535(US9701672, 36 | US9701672, 37)
Affinity DataIC50: 12.5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247172BDBM247172(US9701672, 32 | US9701672, 26)
Affinity DataIC50: 12.6nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247161BDBM247161(1-(1-Isopropyl-1H-pyrazol-3-yl)ethanone | US970167...)
Affinity DataIC50: 14.5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253645BDBM253645((S)-4-(5-Cyclopropylthiophen-2-yl)-2-oxo-6-(4-(4,4...)
Affinity DataIC50: 15nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 251563BDBM251563(US9701672, 44)
Affinity DataIC50: 15.2nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 249801BDBM249801(US9701672, 39)
Affinity DataIC50: 16.6nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247163BDBM247163((S,E)-2-Methyl-N-(2,2,2-trifluoro-1-(4-(5,5,5-trif...)
Affinity DataIC50: 16.6nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247174BDBM247174(US9701672, 28)
Affinity DataIC50: 17.6nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247159BDBM247159(1-(1-Cyclobutyl-1H-pyrazol-3-yl)ethanone | US97016...)
Affinity DataIC50: 19.4nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 251547BDBM251547(US9701672, 43)
Affinity DataIC50: 20.2nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247170BDBM247170(US9701672, 24)
Affinity DataIC50: 22.9nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247164BDBM247164((S,E)-N-(1-(2-Chloro-4-(4,4,4-trifluorobutoxy)phen...)
Affinity DataIC50: 24.5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253637BDBM253637(US9701672, 68)
Affinity DataIC50: 30.2nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253642BDBM253642(US9701672, 71)
Affinity DataIC50: 31.5nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247165BDBM247165((S,E)-2-Methyl-N-(2,2,2-trifluoro-1-(2-methoxy-4-(...)
Affinity DataIC50: 31.8nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 247155BDBM247155(1-(6-(Dimethylamino)pyridin-3-yl)ethanone | US9701...)
Affinity DataIC50: 32nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 253641BDBM253641(US9701672, 70)
Affinity DataIC50: 32.3nMpH: 7.4Assay Description:The MGAT enzyme reactions were performed in Corning FALCON 96-well polypropylene plates, in a total volume of 60 μL of 50 mM potassium phosphate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/30/2018
Entry Details
US Patent

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