Compile Data Set for Download or QSAR
Report error Found 48 Enz. Inhib. hit(s) with all data for entry = 393
TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264699(US9718771, 2-45)
Affinity DataIC50: 0.800nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264702(US9718771, 2-49)
Affinity DataIC50: 0.900nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264671(US9718771, 2-6)
Affinity DataIC50: 1nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264676(US9718771, 2-11)
Affinity DataIC50: 1.10nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264691(US9718771, 2-32)
Affinity DataIC50: 1.10nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264672(US9718771, 2-7)
Affinity DataIC50: 1.20nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264688(US9718771, 2-29)
Affinity DataIC50: 1.20nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264712(US9718771, 6-5)
Affinity DataIC50: 1.20nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264706(US9718771, 4-1)
Affinity DataIC50: 1.20nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264693(US9718771, 2-34)
Affinity DataIC50: 1.5nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264679(US9718771, 2-14)
Affinity DataIC50: 1.70nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264701(US9718771, 2-47)
Affinity DataIC50: 1.80nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264684(US9718771, 2-21)
Affinity DataIC50: 1.90nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264700(US9718771, 2-46)
Affinity DataIC50: 1.90nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264696(US9718771, 2-41)
Affinity DataIC50: 1.90nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264680(US9718771, 2-15)
Affinity DataIC50: 2.5nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264710(US9718771, 6-2)
Affinity DataIC50: 2.5nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264675(US9718771, 2-10)
Affinity DataIC50: 2.5nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264669(US9718771, 2-3)
Affinity DataIC50: 2.80nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264711(US9718771, 6-3)
Affinity DataIC50: 2.80nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264673(US9718771, 2-8)
Affinity DataIC50: 2.90nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264707(US9718771, 4-2)
Affinity DataIC50: 3.10nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264681(US9718771, 2-16)
Affinity DataIC50: 3.30nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264695(US9718771, 2-39)
Affinity DataIC50: 3.40nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264697(US9718771, 2-43)
Affinity DataIC50: 3.5nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264686(US9718771, 2-24)
Affinity DataIC50: 3.70nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264670(US9718771, 2-4)
Affinity DataIC50: 3.90nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264708(US9718771, 5-1)
Affinity DataIC50: 4.40nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264683(US9718771, 2-18)
Affinity DataIC50: 4.70nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264685(US9718771, 2-22)
Affinity DataIC50: 5nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264667(US9718771, 2-1)
Affinity DataIC50: 5.30nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264690(US9718771, 2-31)
Affinity DataIC50: 5.70nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264687(US9718771, 2-25)
Affinity DataIC50: 6.70nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264668(US9718771, 2-2)
Affinity DataIC50: 6.70nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264677(US9718771, 2-12)
Affinity DataIC50: 6.80nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264689(US9718771, 2-30)
Affinity DataIC50: 6.90nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264666(US9718771, 1-2)
Affinity DataIC50: 7.60nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264692(US9718771, 2-33)
Affinity DataIC50: 7.80nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264694(US9718771, 2-37)
Affinity DataIC50: 8.60nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264703(US9718771, 3-1)
Affinity DataIC50: 8.90nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264698(US9718771, 2-44)
Affinity DataIC50: 9nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264709(US9718771, 6-1)
Affinity DataIC50: 11.2nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264705(US9718771, 3-7)
Affinity DataIC50: 12.8nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264704(US9718771, 3-4)
Affinity DataIC50: 15.3nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264678(US9718771, 2-13)
Affinity DataIC50: 21.5nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264674(US9718771, 2-9)
Affinity DataIC50: 22.2nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264682(US9718771, 2-17)
Affinity DataIC50: 27.3nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent

TargetSphingosine 1-phosphate receptor 1(Human)
Kissei Pharmaceutical

US Patent
LigandPNGBDBM264713(US9718771, Comparative1)
Affinity DataIC50: 441nMpH: 7.4 T: 2°CAssay Description:Inhibitory activity evaluation was performed by multi-screen (registered trademark) HTS 96-well plate (Millipore) using the cell membrane fraction st...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/16/2018
Entry Details
US Patent