Compile Data Set for Download or QSAR
Report error Found 37 Enz. Inhib. hit(s) with all data for entry = 1820
LigandChemical structure of BindingDB Monomer ID 342149BDBM342149(US9771359, EX-56 | 1-((2-(tert-butyl)-4-(3-chlorop...)
Affinity DataKi:  0.100nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342128BDBM342128(US9771359, EX-20 | N-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  0.300nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342122BDBM342122(US9771359, EX-14 | US9771359, EX-15 | US9771359, E...)
Affinity DataKi:  0.400nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342117BDBM342117(US9771359, EX-03 | N-((2-(tert-butyl)-4-(3-chlorop...)
Affinity DataKi:  0.600nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342122BDBM342122(US9771359, EX-14 | US9771359, EX-15 | US9771359, E...)
Affinity DataKi:  0.700nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342121BDBM342121(US9771359, EX-13 | US9771359, EX-18 | N-((4-(3-chl...)
Affinity DataKi:  0.700nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342119BDBM342119(US9771359, EX-06 | N-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  0.700nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342120BDBM342120(US9771359, EX-12 | N-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  1.10nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342115BDBM342115(US9771359, EX-01 | N-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  1.40nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342151BDBM342151(US9771359, EX-58 | N-(4-(3-((2-(tert-butyl)-4-(m-t...)
Affinity DataKi:  2.30nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342130BDBM342130(US9771359, EX-24 | N-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  2.35nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342129BDBM342129(US9771359, EX-23 | N-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  4.70nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342121BDBM342121(US9771359, EX-13 | US9771359, EX-18 | N-((4-(3-chl...)
Affinity DataKi:  5.20nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342147BDBM342147(US9771359, EX-54 | 1-((2-(tert-butyl)-4-(3-chlorop...)
Affinity DataKi:  5.90nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342150BDBM342150(US9771359, EX-57 | N-(4-(3-((2-(tert-butyl)-4-(3-c...)
Affinity DataKi:  6.60nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342118BDBM342118(US9771359, EX-05 | N-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  7.5nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342144BDBM342144(US9771359, EX-45 | N-((5-(3-chlorophenyl)-2-(tertb...)
Affinity DataKi:  9.10nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342148BDBM342148(US9771359, EX-55 | 1-((2-(tert-butyl)-4-(3-chlorop...)
Affinity DataKi:  12.3nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342127BDBM342127(US9771359, EX-19 | N-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  13.8nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342138BDBM342138(US9771359, EX-39 | N-(4-(3-((2-(tert-butyl)-4-(3-f...)
Affinity DataKi:  17.6nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342132BDBM342132(US9771359, EX-28 | 1-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  19.4nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
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Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342135BDBM342135(US9771359, EX-33 | 1-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  24.6nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342140BDBM342140(US9771359, EX-41 | 1-((2-(tert-butyl)-4-(3-chlorop...)
Affinity DataKi:  27.5nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342116BDBM342116(US9771359, EX-02 | N-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  28.4nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342142BDBM342142(US9771359, EX-43 | 1-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  29.8nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342143BDBM342143(US9771359, EX-44 | N-((5-(3-chlorophenyl)-2-(tertb...)
Affinity DataKi:  29.9nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342145BDBM342145(US9771359, EX-47 | 1-((2-(tert-butyl)-4-(3-chlorop...)
Affinity DataKi:  33.3nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342146BDBM342146(US9771359, EX-49 | 1-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  35nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342122BDBM342122(US9771359, EX-14 | US9771359, EX-15 | US9771359, E...)
Affinity DataKi:  41.9nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342139BDBM342139(US9771359, EX-40 | 1-((2-(tert-butyl)-4-(3-chlorop...)
Affinity DataKi:  43.6nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342133BDBM342133(US9771359, EX-31 | 1-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  48.8nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342137BDBM342137(US9771359, EX-38 | N-(4-(3-((2-(tert-butyl)-4-(3-c...)
Affinity DataKi:  52.6nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342134BDBM342134(US9771359, EX-32 | 1-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  60.8nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342131BDBM342131(US9771359, EX-27 | 1-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  62.5nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342136BDBM342136(US9771359, EX-35 | 1-((2-(tert-butyl)-4-(3-chlorop...)
Affinity DataKi:  78.4nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342121BDBM342121(US9771359, EX-13 | US9771359, EX-18 | N-((4-(3-chl...)
Affinity DataKi:  96.7nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 342141BDBM342141(US9771359, EX-42 | 1-((4-(3-chlorophenyl)-2-(trifl...)
Affinity DataKi:  103nMAssay Description:The FLIPR protocol consists of 2 substance additions during a kinetic measurement. First the compounds to be tested (5 μM) are pipetted onto the...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/6/2019
Entry Details
US Patent