Compile Data Set for Download or QSAR
Report error Found 31 Enz. Inhib. hit(s) with all data for entry = 2120
TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354702BDBM354702(US9809583, Example 10 | Preparation of t-butyl(4-h...)
Affinity DataIC50: 6.30nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354706BDBM354706(US9809583, Example 19 | Preparation of 4-((2R,5S)-...)
Affinity DataIC50: 7.60nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354712BDBM354712(US9809583, Example 25 | Preparation of N-(4-(((2R,...)
Affinity DataIC50: 8.5nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354721BDBM354721(US9809583, Example 33 | Preparation of ((2S,5S)-3-...)
Affinity DataIC50: 10.4nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354703BDBM354703(US9809583, Example 11 | Preparation of 4-((2R,5S)-...)
Affinity DataIC50: 10.5nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354698BDBM354698(US9809583, Example 6 | Preparation of ((2R,5S)-3-(...)
Affinity DataIC50: 11nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354700BDBM354700(US9809583, Example 8 | Preparation of ((2R,5S)-3-(...)
Affinity DataIC50: 13.7nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354719BDBM354719(US9809583, Example 31 | Preparation of 4-(2R,5S)-5...)
Affinity DataIC50: 14.1nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354717BDBM354717(US9809583, Example 29 | Preparation of (S)-2-hydro...)
Affinity DataIC50: 14.1nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354705BDBM354705(US9809583, Example 13 | Preparation of (S)-3-((4-c...)
Affinity DataIC50: 14.5nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354699BDBM354699(US9809583, Example 7 | Preparation of (S)-3-((4-ni...)
Affinity DataIC50: 15.7nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354715BDBM354715(US9809583, Example 27 | Preparation of 4-((2R,5S)-...)
Affinity DataIC50: 22.4nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354694BDBM354694(US9809583, Example 2 | Preparation of 4-((2S,5S)-5...)
Affinity DataIC50: 23.9nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354722BDBM354722(US9809583, Example 34 | Preparation of 4-(((2R,5S)...)
Affinity DataIC50: 24.1nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354720BDBM354720(US9809583, Example 32 | Preparation of (2R,5S)-3-(...)
Affinity DataIC50: 32.7nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354714BDBM354714(US9809583, Example 26 | Preparation of ethyl(S)-3-...)
Affinity DataIC50: 43.6nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354710BDBM354710(US9809583, Example 23 | Preparation of 4-((2R,5S)-...)
Affinity DataIC50: 44.3nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354693BDBM354693(US9809583, Example 1 | Preparation of (S)-4-((2,3-...)
Affinity DataIC50: 64.4nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354713BDBM354713(US9809583, Example 56 | Preparation of 4-((2R,5S)-...)
Affinity DataIC50: 75.1nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354716BDBM354716(US9809583, Example 28 | Preparation of 4-((2R,5S)-...)
Affinity DataIC50: 77.2nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354697BDBM354697(US9809583, Example 5 | Preparation of 4-((2R,5R)-5...)
Affinity DataIC50: 91.6nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354711BDBM354711(US9809583, Example 24 | Preparation of (2R,5S)-3-(...)
Affinity DataIC50: 141nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354718BDBM354718(US9809583, Example 30 | Preparation of N-(4-(((2S,...)
Affinity DataIC50: 142nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354704BDBM354704(US9809583, Example 12 | Preparation of 4-((2R,5R)-...)
Affinity DataIC50: 145nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354723BDBM354723(US9809583, Example 35 | Preparation of 4-((2S,5S)-...)
Affinity DataIC50: 185nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354701BDBM354701(US9809583, Example 9 | Preparation of 4-(((2R,5S)-...)
Affinity DataIC50: 367nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354696BDBM354696(US9809583, Example 4 | Preparation of (S)-3-((3-me...)
Affinity DataIC50: 657nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354708BDBM354708(US9809583, Example 21 | Preparation of 4-((2S,5R)-...)
Affinity DataIC50: 1.06E+3nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354707BDBM354707(US9809583, Example 20 | Preparation of 4-((2S,5R)-...)
Affinity DataIC50: 1.08E+3nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354695BDBM354695(US9809583, Example 3 | 4-((2S,5R)-5-(hydroxymethyl...)
Affinity DataIC50: 1.09E+3nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent

TargetAndrogen receptor(Green monkey)
Dong-A St

US Patent
LigandChemical structure of BindingDB Monomer ID 354709BDBM354709(US9809583, Example 22 | Preparation of 4-((2S,5R)-...)
Affinity DataIC50: 1.87E+3nMAssay Description:In order to examine binding ability of the agonists of the present invention to androgen receptors, the following in-vitro experiment was performed. ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2019
Entry Details
US Patent