Compile Data Set for Download or QSAR
Report error Found 127 Enz. Inhib. hit(s) with all data for entry = 2144
LigandChemical structure of BindingDB Monomer ID 355969BDBM355969(US9815842, Example 93 | (S)-1-(5-chloro-6- (difluo...)
Affinity DataIC50: 0.00100nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355889BDBM355889(US9815842, Example 13 | (S)-methyl 3-chloro- 5-(3-...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355886BDBM355886(US9815842, Example 10 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355950BDBM355950(US9815842, Example 74 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355967BDBM355967(US9815842, Example 91 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355892BDBM355892(US9815842, Example 16 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50169049BDBM50169049(CHEMBL3806155 | US9815842, Example 1 | US10442808,...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355970BDBM355970(US9815842, Example 94 | (S)-1-(6-(2H-1,2,3- triazo...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355971BDBM355971(US9815842, Example 95 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355980BDBM355980(US9815842, Example 104 | 1-(5-chloro-6-(2H- 1,2,3-...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355885BDBM355885(US9815842, Example 9 | (S)-1-(5-chloro-6- methoxyp...)
Affinity DataIC50: 0.00200nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355973BDBM355973(US9815842, Example 97 | (S)-1-(5-chloro-6- (difluo...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355906BDBM355906(US9815842, Example 30 | 1-(2-chloro-7- isopropylpy...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355896BDBM355896(US9815842, Example 20 | 1-(3-chloro-4-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355897BDBM355897(US9815842, Example 21 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355894BDBM355894(US9815842, Example 18 | 1-(5-chloro-6- methoxypyri...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355895BDBM355895(US9815842, Example 19 | 1-(2-chloro-7- isopropylpy...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355965BDBM355965(US9815842, Example 89 | (S)-1-(2-chloro-7-(1- meth...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355921BDBM355921(US9815842, Example 45 | (R)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355925BDBM355925(US9815842, Example 49 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355890BDBM355890(US9815842, Example 14 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355987BDBM355987(US9815842, Example 111 | (R)-1-(6-(2H-1,2,3- triaz...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355911BDBM355911(US9815842, Example 35 | 1-(7-(sec-butyl)-2- chloro...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355948BDBM355948(US9815842, Example 72 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355978BDBM355978(US9815842, Example 102 | 1-(5-chloro-6-(2H- 1,2,3-...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355915BDBM355915(US9815842, Example 39 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00300nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355920BDBM355920(US9815842, Example 44 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00400nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355929BDBM355929(US9815842, Example 53 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00400nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355878BDBM355878((S)-1-(2-chloro-7-(1-methoxyethyl)pyrazolo[1,5-a]p...)
Affinity DataIC50: 0.00400nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355910BDBM355910(US9815842, Example 34 | 1-(7-(tert-butyl)-2- chlor...)
Affinity DataIC50: 0.00400nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355898BDBM355898(US9815842, Example 22 | 1-(5-chloro-6-(4- methyl-2...)
Affinity DataIC50: 0.00400nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 50169052BDBM50169052(CHEMBL3806235 | US9815842, Example 54 | US10442808...)
Affinity DataIC50: 0.00400nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355899BDBM355899(US9815842, Example 23 | 1-(4-(2- aminopyrimidin-4-...)
Affinity DataIC50: 0.00400nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355902BDBM355902(US9815842, Example 26 | 1-(5-bromopyridin-3- yl)-3...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 356002BDBM356002(US9815842, Example 126 | (R)-1-(5-chloro-6-(2H-1,2...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355928BDBM355928(US9815842, Example 52 | 1-(4-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355961BDBM355961(US9815842, Example 85 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355900BDBM355900(US9815842, Example 24 | 1-(5-chloro-1- methyl-6-ox...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355932BDBM355932(US9815842, Example 56 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355901BDBM355901(US9815842, Example 25 | 1-(5-chloro-6- ethoxypyrid...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355931BDBM355931(US9815842, Example 55 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355951BDBM355951(US9815842, Example 75 | (S)-1-(2-chloro-7-(1- meth...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355957BDBM355957(US9815842, Example 81 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355891BDBM355891(US9815842, Example 15 | 1-(2-chloro-7-(2- methoxyp...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355881BDBM355881(US9815842, Example 5 | (R)-1-(5-chloro-6-(2H-1,2,3...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355977BDBM355977(US9815842, Example 101 | 1-(5-chloro-6-(2H- 1,2,3-...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355974BDBM355974(US9815842, Example 98 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355914BDBM355914(US9815842, Example 38 | 1-(5-chloro-6-(2H- 1,2,3-t...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355947BDBM355947(US9815842, Example 71 | (S)-1-(5-chloro-6- (2H-1,2...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

LigandChemical structure of BindingDB Monomer ID 355979BDBM355979(US9815842, Example 103 | 1-(5-chloro-6-(2H- 1,2,3-...)
Affinity DataIC50: 0.00500nMAssay Description:IC50 values of test compounds were determined with an enzyme activity assay using the C-domain of MALT1 (amino acids 329-824). The readout parameter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/14/2019
Entry Details
US Patent

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