Compile Data Set for Download or QSAR
maximum 50k data
Found 9 Enz. Inhib. hit(s) with all data for entry = 2404
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Orca Pharmaceuticals

US Patent
LigandPNGBDBM364365(4-[3-[2-chloro-6-(trifluoromethyl)benzoyl]-7-fluor...)
Affinity DataIC50:  17.9nMAssay Description:The assay was run in black 384 well plates (Greiner cat no: 784900). Various concentrations of test ligands in 0.1 microlitres DMSO were dispensed to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Orca Pharmaceuticals

US Patent
LigandPNGBDBM364366(4-[3-[2-chloro-6-(trifluoromethyl)benzoyl]-7-fluor...)
Affinity DataIC50:  37.9nMAssay Description:The assay was run in black 384 well plates (Greiner cat no: 784900). Various concentrations of test ligands in 0.1 microlitres DMSO were dispensed to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Orca Pharmaceuticals

US Patent
LigandPNGBDBM364366(4-[3-[2-chloro-6-(trifluoromethyl)benzoyl]-7-fluor...)
Affinity DataIC50:  42.9nMAssay Description:The assay was run in black 384 well plates (Greiner cat no: 784900). Various concentrations of test ligands in 0.1 microlitres DMSO were dispensed to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Orca Pharmaceuticals

US Patent
LigandPNGBDBM364364(4-[3-[2-chloro-6-(trifluoromethyl)benzoyl]-7-fluor...)
Affinity DataIC50:  43.6nMAssay Description:The assay was run in black 384 well plates (Greiner cat no: 784900). Various concentrations of test ligands in 0.1 microlitres DMSO were dispensed to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Orca Pharmaceuticals

US Patent
LigandPNGBDBM364371(4-[3-[2-chloro-6-(trifluoromethyl)benzoyl]-1 H-ind...)
Affinity DataIC50:  59.6nMAssay Description:The assay was run in black 384 well plates (Greiner cat no: 784900). Various concentrations of test ligands in 0.1 microlitres DMSO were dispensed to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Orca Pharmaceuticals

US Patent
LigandPNGBDBM364369(4-[7-fluoro-3-[2-fluoro-6-(trifluoromethyl)benzoyl...)
Affinity DataIC50:  61.9nMAssay Description:The assay was run in black 384 well plates (Greiner cat no: 784900). Various concentrations of test ligands in 0.1 microlitres DMSO were dispensed to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Orca Pharmaceuticals

US Patent
LigandPNGBDBM364370(4-[3-(2,6-dichlorobenzoyl)-7-fluoro-1H-indol-1-yl]...)
Affinity DataIC50:  91.6nMAssay Description:The assay was run in black 384 well plates (Greiner cat no: 784900). Various concentrations of test ligands in 0.1 microlitres DMSO were dispensed to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Orca Pharmaceuticals

US Patent
LigandPNGBDBM364364(4-[3-[2-chloro-6-(trifluoromethyl)benzoyl]-7-fluor...)
Affinity DataIC50:  97.4nMAssay Description:The assay was run in black 384 well plates (Greiner cat no: 784900). Various concentrations of test ligands in 0.1 microlitres DMSO were dispensed to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
Orca Pharmaceuticals

US Patent
LigandPNGBDBM364372(3-fluoro-4-[7-fluoro-3-[2-fluoro-6-(trifluoromethy...)
Affinity DataIC50:  111nMAssay Description:The assay was run in black 384 well plates (Greiner cat no: 784900). Various concentrations of test ligands in 0.1 microlitres DMSO were dispensed to...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent