Compile Data Set for Download or QSAR
Report error Found 57 Enz. Inhib. hit(s) with all data for entry = 2970
TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387172BDBM387172(3-(5-((5-chloro-2-((1-(6-methoxypyridin-3-yl)-1H-p...)
Affinity DataIC50: 0.300nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase B(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387194BDBM387194(5-((5-chloro-2-((1-(2-hydroxypropyl)-1H-pyrazol-4-...)
Affinity DataIC50: 0.600nMAssay Description:Aurora-B:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387171BDBM387171(3-(5-((5-chloro-2-((1-(pyridin-2-yl)-1H-pyrazol-4-...)
Affinity DataIC50: 0.600nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase B(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387182BDBM387182(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 0.700nMAssay Description:Aurora-B:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase B(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387192BDBM387192(5-((5-chloro-2-((1-(2-hydroxypropyl)-1H-pyrazol-4-...)
Affinity DataIC50: 0.800nMAssay Description:Aurora-B:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387186BDBM387186(1-(4-((5-chloro-4-((2-(methyl sulfonyl)octahydrocy...)
Affinity DataIC50: 0.800nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase B(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387184BDBM387184(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 0.800nMAssay Description:Aurora-B:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase B(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387193BDBM387193(1-(4-((5-chloro-4-((2-((cyclopropylmethyl)sulfonyl...)
Affinity DataIC50: 1nMAssay Description:Aurora-B:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase B(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387191BDBM387191(1-(4-((5-chloro-4-((2-(cyclopropylsulfonyl)octahyd...)
Affinity DataIC50: 1nMAssay Description:Aurora-B:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387186BDBM387186(1-(4-((5-chloro-4-((2-(methyl sulfonyl)octahydrocy...)
Affinity DataIC50: 1nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387184BDBM387184(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 1nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase B(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387181BDBM387181(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 1nMAssay Description:Aurora-B:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase B(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387187BDBM387187(1-(4-((5-chloro-4-((2-(methyl sulfonyl)octahydrocy...)
Affinity DataIC50: 1nMAssay Description:Aurora-B:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase B(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387186BDBM387186(1-(4-((5-chloro-4-((2-(methyl sulfonyl)octahydrocy...)
Affinity DataIC50: 1nMAssay Description:Aurora-B:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387182BDBM387182(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 2nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387185BDBM387185(1-(4-((5-chloro-4-((3-(methylsulfonyl)-3-azaspiro[...)
Affinity DataIC50: 2nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase B(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387177BDBM387177(ethyl 5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)am...)
Affinity DataIC50: 2nMAssay Description:Aurora-B:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387187BDBM387187(1-(4-((5-chloro-4-((2-(methyl sulfonyl)octahydrocy...)
Affinity DataIC50: 2nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387187BDBM387187(1-(4-((5-chloro-4-((2-(methyl sulfonyl)octahydrocy...)
Affinity DataIC50: 2nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase B(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387180BDBM387180(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 2nMAssay Description:Aurora-B:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387170BDBM387170(3-(5-((5-chloro-2-((1-(2-hydroxy-2-methylpropyl)-1...)
Affinity DataIC50: 2nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387184BDBM387184(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 3nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387182BDBM387182(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 3nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387172BDBM387172(3-(5-((5-chloro-2-((1-(6-methoxypyridin-3-yl)-1H-p...)
Affinity DataIC50: 4nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387175BDBM387175(5-chloro-N4-(2-(cyclopropylsulfonyl)octahydrocyclo...)
Affinity DataIC50: 5nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387192BDBM387192(5-((5-chloro-2-((1-(2-hydroxypropyl)-1H-pyrazol-4-...)
Affinity DataIC50: 5nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387191BDBM387191(1-(4-((5-chloro-4-((2-(cyclopropylsulfonyl)octahyd...)
Affinity DataIC50: 5nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387176BDBM387176((5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)p...)
Affinity DataIC50: 6nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387179BDBM387179(5-chloro-N4-(2-((cyclopropylmethyl)sulfonyl)octahy...)
Affinity DataIC50: 6nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387194BDBM387194(5-((5-chloro-2-((1-(2-hydroxypropyl)-1H-pyrazol-4-...)
Affinity DataIC50: 7nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387171BDBM387171(3-(5-((5-chloro-2-((1-(pyridin-2-yl)-1H-pyrazol-4-...)
Affinity DataIC50: 8nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387177BDBM387177(ethyl 5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)am...)
Affinity DataIC50: 8nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387181BDBM387181(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 8nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387190BDBM387190(5-((5-chloro-2-((1-(2-hydroxy-2-methylpropyl)-1H-p...)
Affinity DataIC50: 9nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387193BDBM387193(1-(4-((5-chloro-4-((2-((cyclopropylmethyl)sulfonyl...)
Affinity DataIC50: 10nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387169BDBM387169(1-(5-((5-chloro-2-((1-(2-hydroxy-2-methylpropyl)-1...)
Affinity DataIC50: 10nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387177BDBM387177(ethyl 5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)am...)
Affinity DataIC50: 10nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387180BDBM387180(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 11nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387174BDBM387174(1-(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino...)
Affinity DataIC50: 12nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387188BDBM387188(5-((5-chloro-2-((1-(pyrrolidin-3-yl)-1H-pyrazol-4-...)
Affinity DataIC50: 12nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387180BDBM387180(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 12nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387172BDBM387172(3-(5-((5-chloro-2-((1-(6-methoxypyridin-3-yl)-1H-p...)
Affinity DataIC50: 16nMAssay Description:JAK2:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387174BDBM387174(1-(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino...)
Affinity DataIC50: 17nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387189BDBM387189(5-((5-chloro-2-((1-(2-hydroxypropyl)-1H-pyrazol-4-...)
Affinity DataIC50: 19nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK2(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387171BDBM387171(3-(5-((5-chloro-2-((1-(pyridin-2-yl)-1H-pyrazol-4-...)
Affinity DataIC50: 20nMAssay Description:JAK2:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387176BDBM387176((5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)p...)
Affinity DataIC50: 21nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387181BDBM387181(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino)py...)
Affinity DataIC50: 23nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387170BDBM387170(3-(5-((5-chloro-2-((1-(2-hydroxy-2-methylpropyl)-1...)
Affinity DataIC50: 28nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetTyrosine-protein kinase JAK1(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387178BDBM387178(1-(5-((5-chloro-2-((1-methyl-1H-pyrazol-4-yl)amino...)
Affinity DataIC50: 32nMAssay Description:JAK1:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding white...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

TargetAurora kinase A(Human)
Calitor Sciences

US Patent
LigandChemical structure of BindingDB Monomer ID 387183BDBM387183(N4-(2-(tert-butylsulfonyl)octahydrocyclopenta[c]py...)
Affinity DataIC50: 50nMAssay Description:Aurora-A:Kinase assays can be performed by measurement of incorporation of γ-33P ATP into immobilized myelin basic protein (MBP). High binding w...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/2/2020
Entry Details
US Patent

Displayed 1 to 50 (of 57 total ) | Next | Last >>
Jump to: