Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 4 Enz. Inhib. hit(s) with all data for entry = 514
TargetFibroblast growth factor receptor 2(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM142256(US8933099, 22 | US9951047, Compound (I))
Affinity DataIC50:  5.10nMT: 25°CAssay Description:To a flat bottom 96 well white plate (Sumitomo Bakelite Co., Ltd., MS-8496W), 10 μl of FGFR1 protein (Carna Biosciences, Inc., 08-133) solution ...More data for this Ligand-Target Pair
In DepthDetails US Patent
PDB3D3D Structure (crystal)

TargetFibroblast growth factor receptor 1(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM142256(US8933099, 22 | US9951047, Compound (I))
Affinity DataIC50:  5.70nMT: 25°CAssay Description:To a flat bottom 96 well white plate (Sumitomo Bakelite Co., Ltd., MS-8496W), 10 μl of FGFR1 protein (Carna Biosciences, Inc., 08-133) solution ...More data for this Ligand-Target Pair
In DepthDetails US Patent
PDB3D3D Structure (crystal)

TargetFibroblast growth factor receptor 3(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM142256(US8933099, 22 | US9951047, Compound (I))
Affinity DataIC50:  6nMT: 25°CAssay Description:To a flat bottom 96 well white plate (Sumitomo Bakelite Co., Ltd., MS-8496W), 10 μl of FGFR1 protein (Carna Biosciences, Inc., 08-133) solution ...More data for this Ligand-Target Pair
In DepthDetails US Patent


TargetFibroblast growth factor receptor 4(Human)
Eisai R&D Management

US Patent
LigandPNGBDBM142256(US8933099, 22 | US9951047, Compound (I))
Affinity DataIC50:  683nMT: 25°CAssay Description:To a flat bottom 96 well white plate (Sumitomo Bakelite Co., Ltd., MS-8496W), 10 μl of FGFR1 protein (Carna Biosciences, Inc., 08-133) solution ...More data for this Ligand-Target Pair
In DepthDetails US Patent