Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 10415
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533764(N-(4-cyanophenyl)-N-methyl-3-(4-(trifluoromethyl)p...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533793(2-Chloro-5-(N-methyl-3-(4-(methylcarbamoyl)phenyl)...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533865(Methyl 2-(3-(4-carbamoylphenyl)-N-methylpyrazolo[1...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533864(Methyl 2-chloro-5-(N-methyl-3-(4-(methylcarbamoyl)...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533863(WO2022079616, Example 2.1)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533861(Methyl 5-(N-methyl-3-(4-(methylcarbamoyl)phenyl)py...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533860(Methyl 5-(3-(4-carbamoylphenyl)-N-methylpyrazolo[1...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533813(Methyl 2-chloro-5-(N-methyl-3-(2-methyl-4-(carbamo...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533812(2-Morpholinoethyl 2-chloro-5-(N-methyl-3-(4-(methy...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533791(WO2022079616, Example 1.17 | t-Butyl 2-chloro-5-(N...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533790(Methyl 2-chloro-5-(N-methyl-3-(4-(methylcarbamoyl)...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533786(WO2022079616, Example 1.15 | rac-(Tetrahydrofuran-...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533782(WO2022079616, Example 1.13 | isopropyl 5-(3-(4-car...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533775(2-(Dimethylamino)-2-oxoethyl 5-(3-(4-carbamoylphen...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533774(2-Methoxyethyl 5-(3-(4-carbamoylphenyl)-N-methylpy...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533773(2,2,2-Trifluoroethyl 5-(3-(4-carbamoylphenyl)-N-me...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533772(Ethyl 5-(3-(4-carbamoylphenyl)-N-methylpyrazolo[1,...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533771(2-Morpholinoethyl 5-(3-(4-carbamoylphenyl)-N-methy...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533770(Thiazol-5-ylmethyl 5-(3-(4-carbamoylphenyl)-N-meth...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533769(2-Methoxy-2-oxoethyl 5-(3-(4-carbamoylphenyl)-N-me...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533768(Isobutyl 5-(3-(4-carbamoylphenyl)-N-methylpyrazolo...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533765(WO2022079616, Example 1.02 | tert-Butyl 5-(3-(4-ca...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533766(5-(3-(4-Carbamoylphenyl)-N-methylpyrazolo[1,5-a]py...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533767(2-(Methylthio)ethyl 5-(3-(4-carbamoylphenyl)-N-met...)
Affinity DataIC50: <100nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533790(Methyl 2-chloro-5-(N-methyl-3-(4-(methylcarbamoyl)...)
Affinity DataIC50:  550nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533865(Methyl 2-(3-(4-carbamoylphenyl)-N-methylpyrazolo[1...)
Affinity DataIC50:  550nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533793(2-Chloro-5-(N-methyl-3-(4-(methylcarbamoyl)phenyl)...)
Affinity DataIC50:  550nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533862(Methyl 5-(3-(4-carbamoylphenyl)-N-methylpyrazolo[1...)
Affinity DataIC50:  550nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533812(2-Morpholinoethyl 2-chloro-5-(N-methyl-3-(4-(methy...)
Affinity DataIC50:  550nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533837(Methyl 2-chloro-5-(N-methyl-3-(3-methyl-4-(carbamo...)
Affinity DataIC50:  550nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533783(WO2022079616, Example 1.14 | rac-1-((Ethoxycarbony...)
Affinity DataIC50:  550nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533764(N-(4-cyanophenyl)-N-methyl-3-(4-(trifluoromethyl)p...)
Affinity DataIC50:  550nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533856(Methyl 5-(3-(4-carbamoylphenyl)pyrazolo[1,5-a]pyri...)
Affinity DataIC50: >1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533856(Methyl 5-(3-(4-carbamoylphenyl)pyrazolo[1,5-a]pyri...)
Affinity DataIC50: >1.00E+3nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533837(Methyl 2-chloro-5-(N-methyl-3-(3-methyl-4-(carbamo...)
Affinity DataIC50: >1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533771(2-Morpholinoethyl 5-(3-(4-carbamoylphenyl)-N-methy...)
Affinity DataIC50: >1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPhosphatidylinositol 4-kinase()
Novartis

WIPO
LigandPNGBDBM533857(Methyl 2-chloro-5-(3-(4-(methylcarbamoyl)phenyl)py...)
Affinity DataIC50: >1.00E+3nMAssay Description: Baculovirus expression and purification of C. parvum phosphatidylinositol 4-kinase: The full-length coding sequence of C. parvum PI(4)K (cgd8_4500, ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533863(WO2022079616, Example 2.1)
Affinity DataIC50: >1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533813(Methyl 2-chloro-5-(N-methyl-3-(2-methyl-4-(carbamo...)
Affinity DataIC50: >1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533783(WO2022079616, Example 1.14 | rac-1-((Ethoxycarbony...)
Affinity DataIC50: >1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533864(Methyl 2-chloro-5-(N-methyl-3-(4-(methylcarbamoyl)...)
Affinity DataIC50: >1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533860(Methyl 5-(3-(4-carbamoylphenyl)-N-methylpyrazolo[1...)
Affinity DataIC50: >1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533862(Methyl 5-(3-(4-carbamoylphenyl)-N-methylpyrazolo[1...)
Affinity DataIC50: >1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
LigandPNGBDBM533857(Methyl 2-chloro-5-(3-(4-(methylcarbamoyl)phenyl)py...)
Affinity DataIC50: >1.00E+3nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed