Compile Data Set for Download or QSAR
Report error Found 87 Enz. Inhib. hit(s) with all data for entry = 10913
LigandChemical structure of BindingDB Monomer ID 577560BDBM577560(WO2022263472, Example 10 | 7-[(3R,4R)-4-Methyltetr...)
Affinity DataIC50: 1nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577575BDBM577575(WO2022263472, Example 44 | 2-((1-Methyl-3-(oxetan-...)
Affinity DataIC50: 1nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577554BDBM577554(WO2022263472, Example 4 | 2-[[1-[(1 R)-2,2-Difluor...)
Affinity DataIC50: 1nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577560BDBM577560(WO2022263472, Example 10 | 7-[(3R,4R)-4-Methyltetr...)
Affinity DataIC50: 1nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577571BDBM577571(WO2022263472, Example 21 | 2-((1-Methyl-3-(((R)-1 ...)
Affinity DataIC50: 1nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577554BDBM577554(WO2022263472, Example 4 | 2-[[1-[(1 R)-2,2-Difluor...)
Affinity DataIC50: 1nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577571BDBM577571(WO2022263472, Example 21 | 2-((1-Methyl-3-(((R)-1 ...)
Affinity DataIC50: 1nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577557BDBM577557(WO2022263472, Example 7 | WO2022263472, Example 15...)
Affinity DataIC50: 2nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577564BDBM577564(WO2022263472, Example 14 | 2-[[1-(Methylsulfonylme...)
Affinity DataIC50: 2nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577557BDBM577557(WO2022263472, Example 7 | WO2022263472, Example 15...)
Affinity DataIC50: 2nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577568BDBM577568(WO2022263472, Example 18 | 2-((3-(((S)-1-acetyl-2,...)
Affinity DataIC50: 2nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577568BDBM577568(WO2022263472, Example 18 | 2-((3-(((S)-1-acetyl-2,...)
Affinity DataIC50: 2nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577564BDBM577564(WO2022263472, Example 14 | 2-[[1-(Methylsulfonylme...)
Affinity DataIC50: 2nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577556BDBM577556(WO2022263472, Example 6 | 2-((1-Methyl-3-(((2R,3S)...)
Affinity DataIC50: 3nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577567BDBM577567(WO2022263472, Example 17 | 2-((3-(((R)-1 -Acetyl-2...)
Affinity DataIC50: 3nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577567BDBM577567(WO2022263472, Example 17 | 2-((3-(((R)-1 -Acetyl-2...)
Affinity DataIC50: 3nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577570BDBM577570(WO2022263472, Example 20 | 2-((4-(2-Hydroxypropan-...)
Affinity DataIC50: 3nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577570BDBM577570(WO2022263472, Example 20 | 2-((4-(2-Hydroxypropan-...)
Affinity DataIC50: 3nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577558BDBM577558(WO2022263472, Example 8 | WO2022263472, Example 19)
Affinity DataIC50: 4nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577574BDBM577574(WO2022263472, Example 24 | 2-((1 -(methyl-d3)-3-((...)
Affinity DataIC50: 4nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577587BDBM577587(WO2022263472, Example 56 | 2-((1-((S)-1-Cyanoethyl...)
Affinity DataIC50: 4nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577556BDBM577556(WO2022263472, Example 6 | 2-((1-Methyl-3-(((2R,3S)...)
Affinity DataIC50: 4nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577553BDBM577553(WO2022263472, Example 3 | 2-[[1 -methyl-3-[(3S,4R)...)
Affinity DataIC50: 4nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577555BDBM577555(WO2022263472, Example 5 | 2-[[1 -[(1 S)-2,2-difluo...)
Affinity DataIC50: 4nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577556BDBM577556(WO2022263472, Example 6 | 2-((1-Methyl-3-(((2R,3S)...)
Affinity DataIC50: 4nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577582BDBM577582(WO2022263472, Example 51 | (R)-2-((1-Methyl-3-(oxe...)
Affinity DataIC50: 5nMAssay Description: LRRK2(human) is incubated with 50 mM HEPES pH 8.0, 0.2 mM EDTA, 0.01 %Brij-35, 1% (w/v) BSA, 5 mM DTT, 250 Mm RLGRDKYKTLRQIRQ, 10 mM Magnesium aceta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577556BDBM577556(WO2022263472, Example 6 | 2-((1-Methyl-3-(((2R,3S)...)
Affinity DataIC50: 5nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577559BDBM577559(WO2022263472, Example 9 | 2-[[1-[2-Hydroxy-1-methy...)
Affinity DataIC50: 5nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577552BDBM577552(WO2022263472, Example 2 | 2-[[1-Methyl-3-[(3R,4S)-...)
Affinity DataIC50: 5nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577574BDBM577574(WO2022263472, Example 24 | 2-((1 -(methyl-d3)-3-((...)
Affinity DataIC50: 5nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577559BDBM577559(WO2022263472, Example 9 | 2-[[1-[2-Hydroxy-1-methy...)
Affinity DataIC50: 5nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577551BDBM577551(WO2022263472, Example 1 | 2-[[3-(1-acetylazetidin-...)
Affinity DataIC50: 5nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577553BDBM577553(WO2022263472, Example 3 | 2-[[1 -methyl-3-[(3S,4R)...)
Affinity DataIC50: 5nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577558BDBM577558(WO2022263472, Example 8 | WO2022263472, Example 19)
Affinity DataIC50: 5nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577552BDBM577552(WO2022263472, Example 2 | 2-[[1-Methyl-3-[(3R,4S)-...)
Affinity DataIC50: 5nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577558BDBM577558(WO2022263472, Example 8 | WO2022263472, Example 19)
Affinity DataIC50: 5nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577555BDBM577555(WO2022263472, Example 5 | 2-[[1 -[(1 S)-2,2-difluo...)
Affinity DataIC50: 5nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577551BDBM577551(WO2022263472, Example 1 | 2-[[3-(1-acetylazetidin-...)
Affinity DataIC50: 6nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577558BDBM577558(WO2022263472, Example 8 | WO2022263472, Example 19)
Affinity DataIC50: 6nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577562BDBM577562(WO2022263472, Example 12 | 2-[[3-[(3R,4R)-4-Methox...)
Affinity DataIC50: 6nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577599BDBM577599(WO2022263472, Example 80)
Affinity DataIC50: 6nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577557BDBM577557(WO2022263472, Example 7 | WO2022263472, Example 15...)
Affinity DataIC50: 7nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577557BDBM577557(WO2022263472, Example 7 | WO2022263472, Example 15...)
Affinity DataIC50: 7nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577587BDBM577587(WO2022263472, Example 56 | 2-((1-((S)-1-Cyanoethyl...)
Affinity DataIC50: 7nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577581BDBM577581(WO2022263472, Example 50 | 2-((1-((S)-1-cyanoethyl...)
Affinity DataIC50: 7nMAssay Description: LRRK2(human) is incubated with 50 mM HEPES pH 8.0, 0.2 mM EDTA, 0.01 %Brij-35, 1% (w/v) BSA, 5 mM DTT, 250 Mm RLGRDKYKTLRQIRQ, 10 mM Magnesium aceta...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577573BDBM577573(WO2022263472, Example 23 | 2-((1-(Methyl-d3)-3-(((...)
Affinity DataIC50: 8nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577562BDBM577562(WO2022263472, Example 12 | 2-[[3-[(3R,4R)-4-Methox...)
Affinity DataIC50: 8nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577599BDBM577599(WO2022263472, Example 80)
Affinity DataIC50: 9nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577563BDBM577563(WO2022263472, Example 13 | 2-[[3-[(3S,4S)-4-methox...)
Affinity DataIC50: 9nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

LigandChemical structure of BindingDB Monomer ID 577573BDBM577573(WO2022263472, Example 23 | 2-((1-(Methyl-d3)-3-(((...)
Affinity DataIC50: 10nMAssay Description:The measurements of the activities were made using a LRRK2-G2019S(human) Kinase activity assay as described hereunder. The potency of compounds was e...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/30/2022
Entry Details
WIPO WO2022263472

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