Reaction Details Report a problem with these data
Target
Receptor-interacting serine/threonine-protein kinase 1 [2-375]
Ligand
BDBM509402
Substrate
n/a
Meas. Tech.
Biochemical Assay
Ki
<5.00±n/a nM
Citation
Patel, S; Hamilton, G; Stivala, C; Chen, H; Daniels, B Bicyclic sulfones and sulfoxides and methods of use thereof US Patent US11072617 Publication Date 7/27/2021
More Info.:
Target
Name:
Receptor-interacting serine/threonine-protein kinase 1 [2-375]
Synonyms:
RIP | RIP1 | RIPK1 | RIPK1_HUMAN | Receptor-interacting serine/threonine-protein kinase (RIPK1)(2-375)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
42278.41
Organism:
Human
Description:
Q13546[2-375]
Residue:
374
Sequence:
QPDMSLNVIKMKSSDFLESAELDSGGFGKVSLCFHRTQGLMIMKTVYKGPNCIEHNEALLEEAKMMNRLRHSRVVKLLGVIIEEGKYSLVMEYMEKGNLMHVLKAEMSTPLSVKGRIILEIIEGMCYLHGKGVIHKDLKPENILVDNDFHIKIADLGLASFKMWSKLNNEEHNELREVDGTAKKNGGTLYYMAPEHLNDVNAKPTEKSDVYSFAVVLWAIFANKEPYENAICEQQLIMCIKSGNRPDVDDITEYCPREIISLMKLCWEANPEARPTFPGIEEKFRPFYLSQLEESVEEDVKSLKKEYSNENAVVKRMQSLQLDCVAVPSSRSNSATEQPGSLHSSQGLGMGPVEESWFAPSLEHPQEENEPSLQ