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Target
Pantetheinase [22-493]
Ligand
BDBM510520
Substrate
n/a
Meas. Tech.
Enzymatic Assay
IC50
0.300±n/a nM
Citation
Fleck, MT; Godbout, C; Koolman, HF Heteroaromatic compounds as Vanin inhibitors US Patent US11078182 Publication Date 8/3/2021
More Info.:
Target
Name:
Pantetheinase [22-493]
Synonyms:
Pantetheinase (VNN1)(22-493) | VNN1 | VNN1_HUMAN
Type:
Enzyme Catalytic Domain
Mol. Mass.:
52490.93
Organism:
Human
Description:
aa 22-493
Residue:
472
Sequence:
QDTFTAAVYEHAAILPNATLTPVSREEALALMNRNLDILEGAITSAADQGAHIIVTPEDAIYGWNFNRDSLYPYLEDIPDPEVNWIPCNNRNRFGQTPVQERLSCLAKNNSIYVVANIGDKKPCDTSDPQCPPDGRYQYNTDVVFDSQGKLVARYHKQNLFMGENQFNVPKEPEIVTFNTTFGSFGIFTCFDILFHDPAVTLVKDFHVDTIVFPTAWMNVLPHLSAVEFHSAWAMGMRVNFLASNIHYPSKKMTGSGIYAPNSSRAFHYDMKTEEGKLLLSQLDSHPSHSAVVNWTSYASSIEALSSGNKEFKGTVFFDEFTFVKLTGVAGNYTVCQKDLCCHLSYKMSENIPNEVYALGAFDGLHTVEGRYYLQICTLLKCKTTNLNTCGDSAETASTRFEMFSLSGTFGTQYVFPEVLLSENQLAPGEFQVSTDGRLFSLKPTSGPVLTVTLFGRLYEKDWASNASSGLT