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Target
Non-receptor tyrosine-protein kinase TYK2 [833-1187]
Ligand
BDBM174018
Substrate
n/a
Meas. Tech.
TYK2 Kinase Assay
IC50
1.00±n/a nM
Citation
Brasca, MG; Bindi, S; Caldarelli, M; Nesi, M; Orrenius, SC; Panzeri, A Substituted pyrroles active as kinases inhibitors US Patent US9688661 Publication Date 6/27/2017
More Info.:
Target
Name:
Non-receptor tyrosine-protein kinase TYK2 [833-1187]
Synonyms:
Non-receptor tyrosine-protein kinase TYK2 (TYK2) | TYK2 | TYK2_HUMAN
Type:
Protein
Mol. Mass.:
40613.06
Organism:
Human
Description:
Human TYK2 variant (833-1187 aa)
Residue:
355
Sequence:
LPEPSCPQLATLTSQCLTYEPTQRPSFRTILRDLTRLQPHNLADVLTVNPDSPASDPTVFHKRYLKKIRDLGEGHFGKVSLYCYDPTNDGTGEMVAVKALKADCGPQHRSGWKQEIDILRTLYHEHIIKYKGCCEDQGEKSLQLVMEYVPLGSLRDYLPRHSIGLAQLLLFAQQICEGMAYLHAQHYIHRDLAARNVLLDNDRLVKIGDFGLAKAVPEGHEYYRVREDGDSPVFWYAPECLKEYKFYYASDVWSFGVTLYELLTHCDSSQSPPTKFLELIGIAQGQMTVLRLTELLERGERLPRPDKCPCEVYHLMKNCWETEASFRPTFENLIPILKTVHEKYQGQAPSVFSVC