Reaction Details Report a problem with these data
Target
NAD(+) hydrolase SARM1 [50-724]
Ligand
BDBM600555
Substrate
n/a
Meas. Tech.
Biological Assay
IC50
<1000±n/a nM
Citation
Kolluri, R; Tegley, CM; Zhu, L; Brown, SP; Reynolds, CH; Tasker, AS; Grice, CA Substituted pyridine derivatives as SARM1 inhibitors US Patent US11629136 Publication Date 4/18/2023
More Info.:
Target
Name:
NAD(+) hydrolase SARM1 [50-724]
Synonyms:
KIAA0524 | NAD(+) hydrolase SARM1 (50-724) | SAMD2 | SARM | SARM1 | SARM1_HUMAN
Type:
Protein
Mol. Mass.:
74398.52
Organism:
Human
Description:
aa 50-724
Residue:
675
Sequence:
PREVSPGAGTEVQDALERALPELQQALSALKQAGGARAVGAGLAEVFQLVEEAWLLPAVGREVAQGLCDAIRLDGGLDLLLRLLQAPELETRVQAARLLEQILVAENRDRVARIGLGVILNLAKEREPVELARSVAGILEHMFKHSEETCQRLVAAGGLDAVLYWCRRTDPALLRHCALALGNCALHGGQAVQRRMVEKRAAEWLFPLAFSKEDELLRLHACLAVAVLATNKEVEREVERSGTLALVEPLVASLDPGRFARCLVDASDTSQGRGPDDLQRLVPLLDSNRLEAQCIGAFYLCAEAAIKSLQGKTKVFSDIGAIQSLKRLVSYSTNGTKSALAKRALRLLGEEVPRPILPSVPSWKEAEVQTWLQQIGFSKYCESFREQQVDGDLLLRLTEEELQTDLGMKSGITRKRFFRELTELKTFANYSTCDRSNLADWLGSLDPRFRQYTYGLVSCGLDRSLLHRVSEQQLLEDCGIHLGVHRARILTAAREMLHSPLPCTGGKPSGDTPDVFISYRRNSGSQLASLLKVHLQLHGFSVFIDVEKLEAGKFEDKLIQSVMGARNFVLVLSPGALDKCMQDHDCKDWVHKEIVTALSCGKNIVPIIDGFEWPEPQVLPEDMQAVLTFNGIKWSHEYQEATIEKIIRFLQGRSSRDSSAGSDTSLEGAAPMGPT