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Target
AGAP001281-PB
Ligand
BDBM600756
Substrate
n/a
Meas. Tech.
thallium-flux assay
IC50
4600±n/a nM
Citation
 Swale, DR; Foil, LD Method for controlling hematophagous or sap-feeding arthropods US Patent  US11632953 Publication Date 4/25/2023 
Target
Name:
AGAP001281-PB
Synonyms:
n/a
Type:
Protein
Mol. Mass.:
49315.66
Organism:
African malaria mosquito
Description:
A7UVQ1
Residue:
426
Sequence:
MAAERPTLDEKKPLNRIFMRPGVIEEEPDSLDSVISNLPLTVVPSLARISTHGSAFSRQESVRSRALRPGTTRKYRRRAILKNGDCNIVLSKVSRQRLRFLQDIFTTLVDAQWRWTLLVFAFSFIGSWLFFGAIWWLIAFTHGDLEEMHLPKNQEESGWKPCVFNIESYTSAFLFSIETQTTIGYGYRTTTEECPEAIFIMCFQSIYGVMMQAFMVGFVFAKMTRPKHRTQTLLFSKHAVVCQRDGELSLMFRVGDMRKSHIIGANIRAQLIRTKLSREGEVMAQYQHELEVGADHCGSDLFFIWPQIVTHRINTESPFYNMSASDLLQDRFEIVVILEGTVESTGQSTQARSSYVNTEILWGHRFEPIVFYNKENQVYEINYSKFNETHSVDTPLCSARELAEFYKYQDDYRNQAEDHHHLQTPA
  
Inhibitor
Name:
BDBM600756
Synonyms:
US11632953, Compound 14 | VU0652934
Type:
Small organic molecule
Emp. Form.:
C18H18F3N3O2
Mol. Mass.:
365.3496
SMILES:
FC(F)(F)c1nn(CC(=O)N2CCOc3ccccc23)c2CCCCc12
Structure:
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