Reaction Details
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Target
Bifunctional 3'-5' exonuclease/ATP-dependent helicase WRN [517-1238]
Ligand
BDBM646427
Substrate
n/a
Meas. Tech.
In Vitro Enzymatic Activity Assay on WRN Helicase
IC50
40.0±n/a nM
Citation
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More Info.:
Target
Name:
Bifunctional 3'-5' exonuclease/ATP-dependent helicase WRN [517-1238]
Synonyms:
Bifunctional 3'-5' exonuclease/ATP-dependent helicase WRN (517-1238)
Type:
Enzyme Catalytic Domain
Mol. Mass.:
81717.91
Organism:
Homo sapiens (Human)
Description:
Q14191[517-1238]
Residue:
722
Sequence:
NEGEEDDDKDFLWPAPNEEQVTCLKMYFGHSSFKPVQWKVIHSVLEERRDNVAVMATGYGKSLCFQYPPVYVGKIGLVISPLISLMEDQVLQLKMSNIPACFLGSAQSENVLTDIKLGKYRIVYVTPEYCSGNMGLLQQLEADIGITLIAVDEAHCISEWGHDFRDSFRKLGSLKTALPMVPIVALTATASSSIREDIVRCLNLRNPQITCTGFDRPNLYLEVRRKTGNILQDLQPFLVKTSSHWEFEGPTIIYCPSRKMTQQVTGELRKLNLSCGTYHAGMSFSTRKDIHHRFVRDEIQCVIATIAFGMGINKADIRQVIHYGAPKDMESYYQEIGRAGRDGLQSSCHVLWAPADINLNRHLLTEIRNEKFRLYKLKMMAKMEKYLHSSRCRRQIILSHFEDKQVQKASLGIMGTEKCCDNCRSRLDHCYSMDDSEDTSWDFGPQAFKLLSAVDILGEKFGIGLPILFLRGSNSQRLADQYRRHSLFGTGKDQTESWWKAFSRQLITEGFLVEVSRYNKFMKICALTKKGRNWLHKANTESQSLILQANEELCPKKLLLPSSKTVSSGTKEHCYNQVPVELSTEKKSNLEKLYSYKPCDKISSGSNISKKSIMVQSPEKAYSSSQPVISAQEQETQIVLYGKLVEARQKHANKMDVPPAILATNKILVDMAKMRPTTVENVKRIDGVSEGKAAMLAPLLEVIKHFCQTNSVQTDLFSSTKP