Reaction Details Report a problem with these data
Target
GTPase KRas [2-169,G12C,C51S,C80L,C118S]
Ligand
BDBM50572119
Substrate
n/a
Meas. Tech.
SOS-Catalyzed Nucleotide Exchange Assay
IC50
2.60±n/a nM
Citation
Bharathan, I; Gathiaka, S; Han, Y; Ma, X; Otte, RD; Sloman, DL; Graham, TH; Henderson, T; Hennessy, E; Palani, A Small Molecule Inhibitors of KRAS G12C Mutant US Patent US20240043448 Publication Date 2/8/2024
More Info.:
Target
Name:
GTPase KRas [2-169,G12C,C51S,C80L,C118S]
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
19160.36
Organism:
Human sapiens (Human)
Description:
P01116-2[2-169,G12C,C51S,C80L,C118S]
Residue:
168
Sequence:
TEYKLVVVGAGCVGKSALTIQLIQNHFVDEYDPTIEDSYRKQVVIDGETLLLDILDTAGQEEYSAMRDQYMRTGEGFLLVFAINNTKSFEDIHHYREQIKRVKDSEDVPMVLVGNKSDLPSRTVDTKQAQDLARSYGIPFIETSAKTRQGVDDAFYTLVREIRKHKEK